Selectivity switch between FAK and Pyk2: Macrocyclization of FAK inhibitors improves Pyk2 potency von Farand, Julie, Mai, Nicholas, Chandrasekhar, Jayaraman, Newby, Zachary E., Van Veldhuizen, Josh, Loyer-Drew, Jennifer, Venkataramani, Chandrasekar, Guerrero, Juan, Kwok, Amy, Li, Ning, Zherebina, Yelena, Wilbert, Sibylle, Zablocki, Jeff, Phillips, Gary, Watkins, William J., Mourey, Robert, Notte, Gregory T.

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Kinetic Resolution and Double Stereodifferentiation in Catalytic Asymmetric C−H Activation of 2-Substituted Pyrrolidines von Davies, Huw M. L, Venkataramani, Chandrasekar

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Ex Vivo Profiling of PD-1 Blockade Using Organotypic Tumor Spheroids von Jenkins, Russell W, Aref, Amir R, Lizotte, Patrick H, Ivanova, Elena, Stinson, Susanna, Zhou, Chensheng W, Bowden, Michaela, Deng, Jiehui, Liu, Hongye, Miao, Diana, He, Meng Xiao, Walker, William, Zhang, Gao, Tian, Tian, Cheng, Chaoran, Wei, Zhi, Palakurthi, Sangeetha, Bittinger, Mark, Vitzthum, Hans, Kim, Jong Wook, Merlino, Ashley, Quinn, Max, Venkataramani, Chandrasekar, Kaplan, Joshua A, Portell, Andrew, Gokhale, Prafulla C, Phillips, Bart, Smart, Alicia, Rotem, Asaf, Jones, Robert E, Keogh, Lauren, Anguiano, Maria, Stapleton, Lance, Jia, Zhiheng, Barzily-Rokni, Michal, Cañadas, Israel, Thai, Tran C, Hammond, Marc R, Vlahos, Raven, Wang, Eric S, Zhang, Hua, Li, Shuai, Hanna, Glenn J, Huang, Wei, Hoang, Mai P, Piris, Adriano, Eliane, Jean-Pierre, Stemmer-Rachamimov, Anat O, Cameron, Lisa, Su, Mei-Ju, Shah, Parin, Izar, Benjamin, Thakuria, Manisha, LeBoeuf, Nicole R, Rabinowits, Guilherme, Gunda, Viswanath, Parangi, Sareh, Cleary, James M, Miller, Brian C, Kitajima, Shunsuke, Thummalapalli, Rohit, Miao, Benchun, Barbie, Thanh U, Sivathanu, Vivek, Wong, Joshua, Richards, William G, Bueno, Raphael, Yoon, Charles H, Miret, Juan, Herlyn, Meenhard, Garraway, Levi A, Van Allen, Eliezer M, Freeman, Gordon J, Kirschmeier, Paul T, Lorch, Jochen H, Ott, Patrick A, Hodi, F Stephen, Flaherty, Keith T, Kamm, Roger D, Boland, Genevieve M, Wong, Kwok-Kin, Dornan, David, Paweletz, Cloud Peter, Barbie, David A

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Discovery of GS-2278, a Potent and Selective LPAR1 Antagonist for the Treatment of Idiopathic Pulmonary Fibrosis von Tang, Doris T, Du, Zhimin, Yang, Kin S, Bestvater, Brian P, Kaplan, Joshua, Neubig, Megan E, Olen, Casey L, Phillips, Bart, Wang, Peiyuan, Hudson, Thomas, Marchand, Bruno, Chan, Julie, Sharma, Monika, Hu, Yiding, Matles, Mike, Nejati, Elham, Chojnacka, Maja, Adams, Clifton, Pong, Cassie, Holsapple, Kevin, Budas, Grant, Tsui, Vickie, Venkataramani, Chandrasekar, Lazerwith, Scott E, Notte, Gregory T, Watkins, William J, McGlinchey, Ellen, Zagorska, Anna, Farand, Julie

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Abstract 3696: GS-9716: A potent, selective and orally bioavailable small molecule inhibitor of MCL1 for the treatment of cancer von Matson, Clinton K., Kenney, Thomas, Steiner, Bart H., Deodato, Chloe R., Yahiaoui, Anella, Rubio, Claudia A., Chan, Julie T., Mollova, Nevena, Keegan, Kathleen S., Venkataramani, Chandrasekar

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Abstract 5161: Inhibition of TBK1/IKBKE impacts tumor growth of KRAS-mutant colorectal cancers von Stinson, Susanna, He, Jianhua, Jia, Zhiheng, Walker, Katie S., Cui, Zhi-Hua, Kaplan, Joshua A., Venkataramani, Chandrasekar, Wang, Yujin, Guevara, Fatima, Nelson, Timothy, Sicinska, Ewa, Ng, Kimmie, Fuchs, Charles S., Dornan, David

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New Strategic Reactions for Organic Synthesis:  Catalytic Asymmetric C−H Activation α to Nitrogen as a Surrogate for the Mannich Reaction von Davies, Huw M. L, Venkataramani, Chandrasekar, Hansen, Tore, Hopper, Darrin W

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Dirhodium Tetraprolinate-Catalyzed Asymmetric Cyclopropanations with High Turnover Numbers von Davies, Huw M. L, Venkataramani, Chandrasekar

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compostos inibidores da anilina cicloalquilcarbamato benzamida hdac von Chandrasekar Venkataramani

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COMBINATION MCL-1 INHIBITORS WITH ANTI-CANCER AGENTS von MATSON, Clinton, KENNEY, Thomas, VENKATARAMANI, Chandrasekar

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COMBINATION MCL-1 INHIBITORS WITH ANTI-CANCER AGENTS von MATSON, Clinton, KENNEY, Thomas, VENKATARAMANI, Chandrasekar

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Catalytic enantioselective synthesis of beta3-amino acids von Davies, Huw M L, Venkataramani, Chandrasekar

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Catalytic Enantioselective Synthesis of β2-Amino Acids von Davies, Huw M. L., Venkataramani, Chandrasekar

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Catalytic Enantioselective Synthesis of β2-Amino Acids This work was supported by the National Science Foundation (CHE 0092490) and the National Institutes of Health (GM57425) von Davies, Huw M. L., Venkataramani, Chandrasekar

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COMBINATION MCL-1 INHIBITORS WITH ANTI-BODY DRUG CONJUGATES von MATSON, Clinton K, KENNEY, Thomas F, VENKATARAMANI, Chandrasekar

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COMBINATION MCL-1 INHIBITORS WITH ANTI-CANCER AGENTS von KENNEY, Thomas, F, VENKATARAMANI, Chandrasekar, MATSON, Clinton, K

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Combination MCL-1 inhibitors with anti-cancer agents von Kenney, Thomas F, Venkataramani, Chandrasekar, Matson, Clinton K

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Combination MCL-1 inhibitors with anti-body drug conjugates von Kenney, Thomas F, Venkataramani, Chandrasekar, Matson, Clinton K

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LPA receptor antagonists and uses thereof von ZAGORSKA, Anna, VENKATARAMANI, Chandrasekar, YANG, Kin S, TANG, Doris T

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COMBINATION MCL-1 INHIBITORS WITH ANTI-BODY DRUG CONJUGATES von MATSON, Clinton K, KENNEY, Thomas F, VENKATARAMANI, Chandrasekar

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