Chemogenomics: Methods and Protocols von Merk, Daniel, Chaikuad, Apirat

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3D Spheroid Invasion Assay for High-Throughput Screening of Small-Molecule Libraries von Karve, Kunal, Poon, Stephanie, Prinos, Panagiotis, Ailles, Laurie

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NanoBRET™ Live-Cell Kinase Selectivity Profiling Adapted for High-Throughput Screening von Nieman, Amanda N., Dunn Hoffman, Kaitlin K., Dominguez, Elizabeth R., Wilkinson, Jennifer, Vasta, James D., Robers, Matthew B., Lam, Ngan

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Global Assessment of Drug Target Engagement and Selectivity of Covalent Cysteine-Reactive Inhibitors Using Alkyne-Functionalized Probes von Rothweiler, Elisabeth M., Huber, Kilian V. M.

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Annotation of the Effect of Chemogenomic Compounds on Cell Health Using High-Content Microscopy in Live-Cell Mode von Tjaden, Amelie, Knapp, Stefan, Müller, Susanne

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Characterization of Cellular Viability Using Label-Free Brightfield Live-Cell Imaging von Elson, Lewis, Tjaden, Amelie, Knapp, Stefan, Müller, Susanne

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Measuring Protein–Protein Interactions in Cells using Nanoluciferase Bioluminescence Resonance Energy Transfer (NanoBRET) Assay von Szewczyk, Magdalena M., Owens, Dominic D. G., Barsyte-Lovejoy, Dalia

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Developing a Kinase Chemogenomic Set: Facilitating Investigation into Kinase Biology by Linking Phenotypes to Targets von Wells, Carrow I., Drewry, David H.

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Quality Control of Chemogenomic Library Using LC-MS von Němec, Václav, Knapp, Stefan

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Live-Cell High-Throughput Screen for Monitoring Autophagy Flux von Cano-Franco, Sara, Ho-Xuan, Hung, Brunello, Lorene, Stolz, Alexandra

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Compilation of Custom Compound/Bioactivity Datasets from Public Repositories von Isigkeit, Laura, Merk, Daniel

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Target Deconvolution by Limited Proteolysis Coupled to Mass Spectrometry von Reber, Viviane, Gstaiger, Matthias

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Plate-Based Screening for DUB Inhibitors von Scherpe, Stephan, Sapmaz, Aysegul, Mulder, Monique P. C.

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A Fluorescence-Based Reporter Gene Assay to Characterize Nuclear Receptor Modulators von Schallmayer, Espen, Merk, Daniel

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Detection of Cellular Target Engagement for Small-Molecule Modulators of Striatal-Enriched Protein Tyrosine Phosphatase (STEP) von Han, Ye Na, Lambert, Lester J., De Backer, Laurent J. S., Wu, Jiaqian, Cosford, Nicholas D. P., Tautz, Lutz

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Phenotypic Chemical Screening in CD4+ T Cells to Identify Epigenetic Inhibitors von Cribbs, Adam P., Oppermann, Udo

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An Introduction to Chemogenomics von Chaikuad, Apirat, Merk, Daniel

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HiBiT Cellular Thermal Shift Assay (HiBiT CETSA) von Ramachandran, Sarath, Szewczyk, Magdalena, Barghout, Samir H., Ciulli, Alessio, Barsyte-Lovejoy, Dalia, Vu, Victoria

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Novel p38α MAP kinase inhibitors identified from yoctoReactor DNA-encoded small molecule library von Petersen, L. K, Blakskjær, P, Chaikuad, A, Christensen, A. B, Dietvorst, J, Holmkvist, J, Knapp, S, Ko ínek, M, Larsen, L. K, Pedersen, A. E, Röhm, S, Sløk, F. A, Hansen, N. J. V

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An Unusual Binding Model of the Methyl 9‑Anilinothiazolo[5,4‑f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphoryl... von Chaikuad, Apirat, Diharce, Julien, Schröder, Martin, Foucourt, Alicia, Leblond, Bertrand, Casagrande, Anne-Sophie, Désiré, Laurent, Bonnet, Pascal, Knapp, Stefan, Besson, Thierry

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