A Consensus Compound/Bioactivity Dataset for Data-Driven Drug Design and Chemogenomics von Isigkeit, Laura, Chaikuad, Apirat, Merk, Daniel

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Chemogenomics: Methods and Protocols von Merk, Daniel, Chaikuad, Apirat

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The Cysteinome of Protein Kinases as a Target in Drug Development von Chaikuad, Apirat, Koch, Pierre, Laufer, Stefan A., Knapp, Stefan

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The ins and outs of selective kinase inhibitor development von Müller, Susanne, Chaikuad, Apirat, Gray, Nathanael S, Knapp, Stefan

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An Introduction to Chemogenomics von Chaikuad, Apirat, Merk, Daniel

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Comparative structural analyses and nucleotide-binding characterization of the four KH domains of FUBP1 von Ni, Xiaomin, Knapp, Stefan, Chaikuad, Apirat

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Structural consequences of BMPR2 kinase domain mutations causing pulmonary arterial hypertension von Chaikuad, Apirat, Thangaratnarajah, Chancievan, von Delft, Frank, Bullock, Alex N.

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Discovery of an MLLT1/3 YEATS Domain Chemical Probe von Moustakim, Moses, Christott, Thomas, Monteiro, Octovia P., Bennett, James, Giroud, Charline, Ward, Jennifer, Rogers, Catherine M., Smith, Paul, Panagakou, Ioanna, Díaz‐Sáez, Laura, Felce, Suet Ling, Gamble, Vicki, Gileadi, Carina, Halidi, Nadia, Heidenreich, David, Chaikuad, Apirat, Knapp, Stefan, Huber, Kilian V. M., Farnie, Gillian, Heer, Jag, Manevski, Nenad, Poda, Gennady, Al‐awar, Rima, Dixon, Darren J., Brennan, Paul E., Fedorov, Oleg

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A new class of small molecule inhibitor of BMP signaling von Sanvitale, Caroline E, Kerr, Georgina, Chaikuad, Apirat, Ramel, Marie-Christine, Mohedas, Agustin H, Reichert, Sabine, Wang, You, Triffitt, James T, Cuny, Gregory D, Yu, Paul B, Hill, Caroline S, Bullock, Alex N

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Hepatitis Delta Virus histone mimicry drives the recruitment of chromatin remodelers for viral RNA replication von Abeywickrama-Samarakoon, Natali, Cortay, Jean-Claude, Sureau, Camille, Müller, Susanne, Alfaiate, Dulce, Guerrieri, Francesca, Chaikuad, Apirat, Schröder, Martin, Merle, Philippe, Levrero, Massimo, Dény, Paul

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Structural Basis of Intracellular TGF-β Signaling: Receptors and Smads von Chaikuad, Apirat, Bullock, Alex N

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Image-Based Annotation of Chemogenomic Libraries for Phenotypic Screening von Tjaden, Amelie, Chaikuad, Apirat, Kowarz, Eric, Marschalek, Rolf, Knapp, Stefan, Schröder, Martin, Müller, Susanne

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Defined PEG smears as an alternative approach to enhance the search for crystallization conditions and crystal-quality improvement in reduced screens von Chaikuad, Apirat, Knapp, Stefan, von Delft, Frank

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Development of Potent, Selective SRPK1 Inhibitors as Potential Topical Therapeutics for Neovascular Eye Disease von Batson, Jennifer, Toop, Hamish D, Redondo, Clara, Babaei-Jadidi, Roya, Chaikuad, Apirat, Wearmouth, Stephen F, Gibbons, Brian, Allen, Claire, Tallant, Cynthia, Zhang, Jingxue, Du, Chunyun, Hancox, Jules C, Hawtrey, Tom, Da Rocha, Joana, Griffith, Renate, Knapp, Stefan, Bates, David O, Morris, Jonathan C

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DFG‑1 Residue Controls Inhibitor Binding Mode and Affinity, Providing a Basis for Rational Design of Kinase Inhibitor Selectivity von Schröder, Martin, Bullock, Alex N, Fedorov, Oleg, Bracher, Franz, Chaikuad, Apirat, Knapp, Stefan

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Modulation of tau tubulin kinases (TTBK1 and TTBK2) impacts ciliogenesis von Bashore, Frances M., Marquez, Ariana B., Chaikuad, Apirat, Howell, Stefanie, Dunn, Andrea S., Beltran, Alvaro A., Smith, Jeffery L., Drewry, David H., Beltran, Adriana S., Axtman, Alison D.

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Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype von Walter, Anne, Chaikuad, Apirat, Helmer, Renate, Loaëc, Nadège, Preu, Lutz, Ott, Ingo, Knapp, Stefan, Meijer, Laurent, Kunick, Conrad

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Assessing reversible and irreversible binding effects of kinase covalent inhibitors through ADP-Glo assays von Schröder, Martin, Chaikuad, Apirat

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Lessons from LIMK1 enzymology and their impact on inhibitor design von Salah, Eidarus, Chatterjee, Deep, Beltrami, Alessandra, Tumber, Anthony, Preuss, Franziska, Canning, Peter, Chaikuad, Apirat, Knaus, Petra, Knapp, Stefan, Bullock, Alex N., Mathea, Sebastian

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Selective Inhibitors of Cyclin G Associated Kinase (GAK) as Anti-Hepatitis C Agents von Kovackova, Sona, Chang, Lei, Bekerman, Elena, Neveu, Gregory, Barouch-Bentov, Rina, Chaikuad, Apirat, Heroven, Christina, Šála, Michal, De Jonghe, Steven, Knapp, Stefan, Einav, Shirit, Herdewijn, Piet

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