Structural Determinants for Small-Molecule Activation of Skeletal Muscle AMPK α2β2γ1 by the Glucose Importagog SC4 von Ngoei, Kevin R.W., Langendorf, Christopher G., Ling, Naomi X.Y., Hoque, Ashfaqul, Varghese, Swapna, Camerino, Michelle A., Walker, Scott R., Bozikis, Ylva E., Dite, Toby A., Ovens, Ashley J., Smiles, William J., Jacobs, Roxane, Huang, He, Parker, Michael W., Scott, John W., Rider, Mark H., Foitzik, Richard C., Kemp, Bruce E., Baell, Jonathan B., Oakhill, Jonathan S.

Volltext

(+)-Fluorenylethylchloroformate (FLEC)--improved synthesis for application in chiral analysis and peptidomimetic synthesis von Camerino, Michelle A, Chalmers, David K, Thompson, Philip E

Volltext

The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interface von Camerino, Michelle A, Zhong, Nan, Dong, Aiping, Dickson, Bradley M, James, Lindsey I, Baughman, Brandi M, Norris, Jacqueline L, Kireev, Dmitri B, Janzen, William P, Arrowsmith, Cheryl H, Frye, Stephen V

Volltext

(S)-(−)-Fluorenylethylchloroformate (FLEC); preparation using asymmetric transfer hydrogenation and application to the analysis and resolution of amines von Amin, Mohammad A., Camerino, Michelle A., Mountford, Simon J., Ma, Xiao, Manallack, David T., Chalmers, David K., Wills, Martin, Thompson, Philip E.

Volltext

Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer von Sharma, Shikhar, Chung, Chi-Yeh, Uryu, Sean, Petrovic, Jelena, Cao, Joan, Rickard, Amanda, Nady, Nataliya, Greasley, Samantha, Johnson, Eric, Brodsky, Oleg, Khan, Showkhin, Wang, Hui, Wang, Zhenxiong, Zhang, Yong, Tsaparikos, Konstantinos, Chen, Lei, Mazurek, Anthony, Lapek, John, Kung, Pei-Pei, Sutton, Scott, Richardson, Paul F., Greenwald, Eric C., Yamazaki, Shinji, Jones, Rhys, Maegley, Karen A., Bingham, Patrick, Lam, Hieu, Stupple, Alexandra E., Kamal, Aileen, Chueh, Anderly, Cuzzupe, Anthony, Morrow, Benjamin J., Ren, Bin, Carrasco-Pozo, Catalina, Tan, Chin Wee, Bhuva, Dharmesh D., Allan, Elizabeth, Surgenor, Elliot, Vaillant, François, Pehlivanoglu, Havva, Falk, Hendrik, Whittle, James R., Newman, Janet, Cursons, Joseph, Doherty, Judy P., White, Karen L., MacPherson, Laura, Devlin, Mark, Dennis, Matthew L., Hattarki, Meghan K., De Silva, Melanie, Camerino, Michelle A., Butler, Miriam S., Dolezal, Olan, Pilling, Patricia, Foitzik, Richard, Stupple, Paul A., Lagiakos, H. Rachel, Walker, Scott R., Hediyeh-Zadeh, Soroor, Nuttall, Stewart, Spall, Sukhdeep K., Charman, Susan A., Connor, Theresa, Peat, Thomas S., Avery, Vicky M., Bozikis, Ylva E., Yang, Yuqing, Zhang, Ming, Monahan, Brendon J., Voss, Anne K., Thomas, Tim, Street, Ian P., Dawson, Sarah-Jane, Dawson, Mark A., Lindeman, Geoffrey J., Davis, Melissa J., Visvader, Jane E., Paul, Thomas A.

Volltext

Solid Phase Synthesis and Circular Dichroism Analysis of (i → i + 4) Cyclic Lactam Analogues of Kisspeptin von Camerino, Michelle A., Kong, David C. M., Chalmers, David K., Thompson, Philip E.

Volltext

Abstract 1130: First-in-class KAT6A/KAT6B inhibitor CTx-648 (PF-9363) demonstrates potent anti-tumor activity in ER+ breast cancer with KAT6A dysregulation von Sharma, Shikhar, Chung, Jay, Uryu, Sean, Rickard, Amanda, Nady, Natalie, Khan, Showkhin, Wang, Zhenxiong, Zhang, Yong, Zhang, Haikuo, Kung, Pei-Pei, Greenwald, Eric, Maegley, Karen, Bingham, Patrick, Lam, Hieu, Bozikis, Ylva E., Falk, Hendrik, Allan, Elizabeth, Avery, Vicky M., Butler, Miriam S., Camerino, Michelle A., Carrasco-Pozo, Catalina, Charman, Susan A., Davis, Melissa J., Dawson, Mark A., Sarah-Jane, Dawson, de Silva, Melanie, Dennis, Matthew L., Dolezal, Olan, Lagiakos, Rachel, Lindeman, Geoffrey J., MacPherson, Laura, Nuttall, Stewart, Peat, Thomas S., Ren, Bin, Stupple, Alexandra E., Surgenor, Elliot, Tan, Chin Wee, Thomas, Tim, Visvader, Jane E., Voss, Anne K., Vaillant, Francois, White, Karen L., Whittle, James, Yang, Yuqing, Hediyeh-Zadeh, Soroor, Stupple, Paul A., Street, Ian P., Monahan, Brendon J., Paul, Thomas

Volltext

(+)-Fluorenylethylchloroformate (FLEC) - improved synthesis for application in chiral analysis and peptidomimetic synthesisElectronic supplementary information (ESI) available: Ful... von Camerino, Michelle A, Chalmers, David K, Thompson, Philip E

Volltext

Abstract 5371: PRMT5 inhibitors as novel treatment for cancers von Falk, Hendrik, Foitzik, Richard C., Allan, Elizabeth, deSilva, Melanie, Yang, Hong, Bozikis, Ylva E., Nikac, Marica, Walker, Scott R., Camerino, Michelle A., Morrow, Ben J., Stupple, Alexandra E., Lagiakos, Rachel, Pinson, Jo-Anne, Lessene, Romina, Kersten, Wilhelmus JA, Ganame, Danny G., Holmes, Ian P., Lunniss, Gill E., Chung, Matthew, Hermans, Stefan J., Parker, Michael W., Thistlethwaite, Alison, White, Karen, Charman, Susan A., Monahan, Brendon J., Pilling, Patricia, Grusovin, Julian, Peat, Thomas S., Sonderegger, Stefan, Toulmin, Emma, Jane, Stephen M., Curtis, David J., Stupple, Paul A., Street, Ian P.

Volltext

The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interfaceElectronic supplementary information (ESI) available: Experimental procedures includin... von Camerino, Michelle A, Zhong, Nan, Dong, Aiping, Dickson, Bradley M, James, Lindsey I, Baughman, Brandi M, Norris, Jacqueline L, Kireev, Dmitri B, Janzen, William P, Arrowsmith, Cheryl H, Frye, Stephen V

Volltext

Synthesis of Benzyl 2-(4-(8-chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)piperazin-1-yl)acetate von Camerino, Michelle, Capuano, Ben, Crosby, Ian, Lloyd, Edward

Volltext

COMPOUND von MORROW BENJAMIN J, BOZIKIS YLVA E B, LAGIAKOS HELEN R, WALKER SCOTT R, FOITZIK RICHARD C, CAMERINO MICHELLE A, HEMLEY CATHERINE F, STUPPLE PAUL A

Volltext bestellen

High-resolution US of the facial vessels with new facial vein landmarks for reconstructive surgery and dermal injection von Pistoia, Federico, Camerino, Paola Lovino, Ioppi, Alessandro, Picasso, Riccardo, Zaottini, Federico, Caprioli, Simone, Mocellin, Davide, Ascoli, Alessandro, Pansecchi, Michelle, Carobbio, Andrea Luigi Camillo, Parrinello, Giampiero, Marchi, Filippo, Peretti, Giorgio, Martinoli, Carlo

Volltext

Crystal structures of human ENPP1 in apo and bound forms von Dennis, Matthew L., Newman, Janet, Dolezal, Olan, Hattarki, Meghan, Surjadi, Regina N., Nuttall, Stewart D., Pham, Tam, Nebl, Tom, Camerino, Michelle, Khoo, Poh Sim, Monahan, Brendon J., Peat, Thomas S.

Volltext

Compounds von HEMLEY, CATHERINE FAE, STUPPLE, PAUL ANTHONY, LAGIAKOS, HELEN RACHEL, MORROW, BENJAMIN JOSEPH, CAMERINO, MICHELLE ANG, WALKER, SCOTT RAYMOND, FOITZIK, RICHARD CHARLES, BOZIKIS, YLVA ELISABET BERGMAN

Volltext bestellen

Abstract 4029: BL-011256 is a novel VEGFR3 selective inhibitor, which suppresses tumor lymphatics and lymph node metastasis in an animal model of melanoma von Leske, Annabell, Foitzik, Richard, Beaumont, Donna, Bentley, John, Bergman, Ylva, Brown, Chloe, Camerino, Michelle, Charman, Susan, Choi, Neil, Silva, Melanie D., Chung, Matthew, Falk, Hendrik, Ganame, Danny, Gregg, Alison, Grusovin, Julian, Harvey, Andrew, Hemley, Catherine, Holmes, Ian, Huff, Belinda, Inglis, Daniel, Kersten, Wilhelmus, Lavranos, Tina, Lessene, Romina, Lunniss, Gillian, Monahan, Brendon, Morrow, Benjamin, Nikac, Marica, Nikolakopoulos, George, Paul, Dharam, Peat, Tom, Ripper, Justin, Scherer, Michaela, Stupple, Paul, White, Karen, Street, Ian, Kremmidiotis, Gabriel

Volltext

SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING von MORROW BENJAMIN JOSEPH, STEVENSON GRAEME IRVINE, WALKER SCOTT RAYMOND, STUPPLE PAUL ANTHONY, CAMERINO MICHELLE ANG

Volltext bestellen

Selective Inhibitors of Arginine Methyl Transferase 5 (PRMT5) As a Novel Treatment for β-Thalassemia and Sickle Cell Disease von Street, Ian, Monahan, Brendon, Falk, Hendrik, Allan, Elizabeth, Bergman, Ylva, Stupple, Paul, Holmes, Ian, Gregg, Alison, Charman, Susan, Lackovic, Kurt, Peat, Tom, Walker, Scott, Lowes, Kym, Kersten, Wilco, Alcindor, Jo, Chung, Matthew, Parker, Michael, Foitzik, Richard, Camerino, Michelle, Nikac, Marcia, Grusovin, Julian, Pilling, Pat, Sonderegger, Stefan, Tan, Yuen, Zhao, Quan, Curtis, David J., Jane, Stephen M

Volltext

BENZISOXAZOLE SULFONAMIDE DERIVATIVES von GREASLEY, SAMANTHA ELIZABETH, STUPPLE, PAUL ANTHONY, KUMPF, ROBERT ARNOLD, RICHARDSON, PAUL FRANCIS, KUNG, PEI-PEI, HOFFMAN, ROBERT LOUIS, CAMERINO, MICHELLE ANG, BRODSKY, OLEG, BOZIKIS, YLVA ELISABET BERGMAN, SUTTON, SCOTT CHANNING

Volltext bestellen

Benzisoxazole sulfonamide derivatives von GREASLEY, SAMANTHA ELIZABETH, STUPPLE, PAUL ANTHONY, KUMPF, ROBERT ARNOLD, RICHARDSON, PAUL FRANCIS, KUNG, PEI-PEI, HOFFMAN, ROBERT LOUIS, CAMERINO, MICHELLE ANG, BRODSKY, OLEG, BOZIKIS, YLVA ELISABET BERGMAN, SUTTON, SCOTT CHANNING

Volltext bestellen