Antagonizing the parathyroid calcium receptor stimulates parathyroid hormone secretion and bone formation in osteopenic rats von Gowen, M, Stroup, G B, Dodds, R A, James, I E, Votta, B J, Smith, B R, Bhatnagar, P K, Lago, A M, Callahan, J F, DelMar, E G, Miller, M A, Nemeth, E F, Fox, J

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Benzimidazole derivatives as arginine mimetics in 1,4-benzodiazepine nonpeptide vitronectin receptor (αvβ3) antagonists von Keenan, Richard M., Miller, William H., Lago, M.Amparo, Ali, Fadia E., Bondinell, William E., Callahan, James F., Calvo, Raul R., Cousins, Russell D., Hwang, Shing-Mei, Jakas, Dalia R., Ku, Thomas W., Kwon, Chet, Nguyen, Thomas T., Reader, Valerie A., Rieman, David J., Ross, Steven T., Takata, Dennis T., Uzinskas, Irene N., Yuan, Catherine C.K., Smith, Brian R.

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A Check on Rational Drug Design: Crystal Structure of a Complex of Human Immunodeficiency Virus Type 1 Protease with a Novel .gamma.-Turn Mimetic Inhibitor von Hoog, Susan S, Zhao, Baoguang, Winborne, Evon, Fisher, Seth, Green, David W, DesJarlais, Renee L, Newlander, Kenneth A, Callahan, James F, Abdel-Meguid, Sherin S, Moore, Michael L, Huffman, William F

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Structure−Activity Relationships of Novel Hematoregulatory Peptides von Bhatnagar, Pradip K, Agner, Erik K, Alberts, Doreen, Arbo, Bente E, Callahan, James F, Cuthbertson, Allan S, Engelsen, Steinar J, Fjerdingstad, Hege, Hartmann, Michael, Heerding, Dirk, Hiebl, Johann, Huffman, William F, Hysben, Mette, King, Andrew G, Kremminger, Peter, Kwon, Chet, LoCastro, Steve, Løvhaug, Dagfinn, Pelus, Louis M, Petteway, Steve, Takata, Joanne S

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Discovery of Orally Active Nonpeptide Vitronectin Receptor Antagonists Based on a 2-Benzazepine Gly-Asp Mimetic von Miller, William H, Alberts, Doreen P, Bhatnagar, Pradip K, Bondinell, William E, Callahan, James F, Calvo, Raul R, Cousins, Russell D, Erhard, Karl F, Heerding, Dirk A, Keenan, Richard M, Kwon, Chet, Manley, Peter J, Newlander, Kenneth A, Ross, Stephen T, Samanen, James M, Uzinskas, Irene N, Venslavsky, Joseph W, Yuan, Catherine C.-K, Haltiwanger, R. Curtis, Gowen, Maxine, Hwang, Shing-Mei, James, Ian E, Lark, Michael W, Rieman, David J, Stroup, George B, Azzarano, Leonard M, Salyers, Kevin L, Smith, Brian R, Ward, Keith W, Johanson, Kyung O, Huffman, William F

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A novel constrained reduced-amide inhibitor of HIV-1 protease derived from the sequential incorporation of .gamma.-turn mimetics into a model substrate von Newlander, Kenneth A, Callahan, James F, Moore, Michael L, Tomaszek, Thaddeus A, Huffman, William F

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Novel peptidomimetic hematoregulatory compounds von HEERDING, D. A, ABRUZZESE, M, TAKATA, J. S, BHATNAGAR, P. K, ALBERTS, D, BURGESS, J, CALLAHAN, J. F, HUFFMAN, W. F, KING, A. G, LOCASTRO, S, DEMARSH, P, PELUS, L. M

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Inhibition of Transforming Growth Factor (TGF)-β1–Induced Extracellular Matrix with a Novel Inhibitor of the TGF-β Type I Receptor Kinase Activity: SB-431542 von Laping, N. J., Grygielko, E., Mathur, A., Butter, S., Bomberger, J., Tweed, C., Martin, W., Fornwald, J., Lehr, R., Harling, J., Gaster, L., Callahan, J. F., Olson, B. A.

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Conformational Preferences in a Benzodiazepine Series of Potent Nonpeptide Fibrinogen Receptor Antagonists von Keenan, Richard M, Callahan, James F, Samanen, James M, Bondinell, William E, Calvo, Raul R, Chen, Lichong, DeBrosse, Charles, Eggleston, Drake S, Haltiwanger, R. Curtis, Hwang, Shing Mei, Jakas, Dalia R, Ku, Thomas W, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael F, Southhall, Linda S, Uzinskas, Irene, Vasko-Moser, Janice A, Venslavsky, Joseph W, Wong, Angela S, Huffman, William F

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Design and synthesis of a C7 mimetic for the predicted .gamma.-turn conformation found in several constrained RGD antagonists von Callahan, James F, Bean, John W, Burgess, Joelle L, Eggleston, Drake S, Hwang, Shing Mei, Kopple, Kenneth D, Koster, Paul F, Nichols, Andrew, Peishoff, Catherine E

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Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists von Samanen, James M, Ali, Fadia E, Barton, Linda S, Bondinell, William E, Burgess, Joelle L, Callahan, James F, Calvo, Raul R, Chen, Wenting, Chen, Lichong, Erhard, Karl, Feuerstein, Giora, Heys, Richard, Hwang, Shing-Mei, Jakas, Dalia R, Keenan, Richard M, Ku, Thomas W, Kwon, Chet, Lee, Chao-Pin, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael, Peishoff, Catherine E, Rhodes, Gerald, Ross, Steven, Shu, Arthur, Simpson, Richard, Takata, Dennis, Yellin, Tobias O, Uzsinskas, Irene, Venslavsky, Joseph W, Yuan, Chuan-Kui, Huffman, William F

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Structure-activity relationships of novel vasopressin antagonists containing C-terminal diaminoalkanes and (aminoalkyl)guanidines von Callahan, James F, Ashton-Shue, Daryl, Bryan, Heidemarie G, Bryan, William M, Heckman, Grace D, Kinter, Lewis B, McDonald, Jeanne E, Moore, Michael L, Schmidt, Dulcie B

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Inhibition of neuronally induced relaxation of canine lower esophageal sphincter by opioid peptides von Barnette, Mary S., Grous, Marilyn, Manning, Carol D., Callahan, James F., Barone, Frank C.

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Inhibition of hematopoietic progenitor cell growth by Tyr-MIF, an endogenous opiate modulator, and its degradation products von Horowitz, Daniel, Callahan, James F., Pelus, Louis M., Fukuda, Seiji, King, Andrew G.

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Discovery of Potent Nonpeptide Vitronectin Receptor (αVβ3) Antagonists von Keenan, Richard M, Miller, William H, Kwon, Chet, Ali, Fadia E, Callahan, James F, Calvo, Raul R, Hwang, Shing-Mei, Kopple, Kenneth D, Peishoff, Catherine E, Samanen, James M, Wong, Angela S, Yuan, Chuan-Kui, Huffman, William F

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Novel vasopressin analogs that help define a minimum effective antagonist pharmacophore von Huffman, William F, Ali, Fadia E, Bryan, William M, Callahan, James F, Moore, Michael L, Silvestri, Joanne S, Yim, Nelson C. F, Kinter, Lewis B, McDonald, Jeanne E

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SB-431542 is a potent and specific inhibitor of transforming growth factor-beta superfamily type I activin receptor-like kinase (ALK) receptors ALK4, ALK5, and ALK7 von Inman, Gareth J, Nicolás, Francisco J, Callahan, James F, Harling, John D, Gaster, Laramie M, Reith, Alastair D, Laping, Nicholas J, Hill, Caroline S

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Cyclic enkephalin analogues containing α-amino-β-mercapto-β,β-pentamethylenepropionic acid at positions 2 or 5 von BRYAN, W. M, CALLAHAN, J. F, CODD, E. E, LEMIEUX, C, MOORE, M. L, SCHILLER, P. W, WALKER, R. F, HUFFMAN, W. F

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Dicarbavasopressin antagonist analogs exhibit reduced in vivo agonist activity von Moore, Michael L, Albrightson, Christine, Brickson, Bridget, Bryan, Heidemarie G, Caldwell, Nancy, Callahan, James F, Foster, Jonathan, Kinter, Lewis B, Newlander, Kenneth A

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Chemical Structure and Skin Penetrating Capacity of a Short Series of Organic Phosphates and Phosphoric Acid von Marzulli, Francis N., Callahan, John F., Brown, D.W.C.

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