TRPA1 modulation by piperidine carboxamides suggests an evolutionarily conserved binding site and gating mechanism von Chernov-Rogan, Tania, Gianti, Eleonora, Liu, Chang, Villemure, Elisia, Cridland, Andrew P., Hu, Xiaoyu, Ballini, Elisa, Lange, Wienke, Deisemann, Heike, Li, Tianbo, Ward, Stuart I., Hackos, David H., Magnuson, Steven, Safina, Brian, Klein, Michael L., Volgraf, Matthew, Carnevale, Vincenzo, Chena, Jun

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Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic E... von Terrett, Jack A, Chen, Huifen, Shore, Daniel G, Villemure, Elisia, Larouche-Gauthier, Robin, Déry, Martin, Beaumier, Francis, Constantineau-Forget, Léa, Grand-Maître, Chantal, Lépissier, Luce, Ciblat, Stéphane, Sturino, Claudio, Chen, Yong, Hu, Baihua, Lu, Aijun, Wang, Yunli, Cridland, Andrew P, Ward, Stuart I, Hackos, David H, Reese, Rebecca M, Shields, Shannon D, Chen, Jun, Balestrini, Alessia, Riol-Blanco, Lorena, Lee, Wyne P, Liu, John, Suto, Eric, Wu, Xiumin, Zhang, Juan, Ly, Justin Q, La, Hank, Johnson, Kevin, Baumgardner, Matt, Chou, Kang-Jye, Rohou, Alexis, Rougé, Lionel, Safina, Brian S, Magnuson, Steven, Volgraf, Matthew

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Catalytic enantioselective electrocyclic cascades von Maciver, Eleanor E, Knipe, Peter C, Cridland, Andrew P, Thompson, Amber L, Smith, Martin D

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Optimization of Sphingosine-1-phosphate‑1 Receptor Agonists: Effects of Acidic, Basic, and Zwitterionic Chemotypes on Pharmacokinetic and Pharmacodynamic Profiles von Skidmore, John, Heer, Jag, Johnson, Christopher N, Norton, David, Redshaw, Sally, Sweeting, Jennifer, Hurst, David, Cridland, Andrew, Vesey, David, Wall, Ian, Ahmed, Mahmood, Rivers, Dean, Myatt, James, Giblin, Gerard, Philpott, Karen, Kumar, Umesh, Stevens, Alexander, Bit, Rino A, Haynes, Andrea, Taylor, Simon, Watson, Robert, Witherington, Jason, Demont, Emmanuel, Heightman, Tom D

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Studies on the Synthesis of the ABC Rings of (±)-Hexacyclinic Acid von Clarke, Paul A, Cridland, Andrew P, Rolla, Gabriele A, Iqbal, Mudassar, Bainbridge, Nigel P, Whitwood, Adrian C, Wilson, Claire

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A Racemic Synthesis of an AB-Ring System of Hexacyclinic Acid von Clarke, Paul A, Cridland, Andrew P

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Novel Conversion of 1,2-Disubstituted cis-Epoxides to One-Carbon Homologated Allylic Alcohols Using Dimethylsulfonium Methylide von Alcaraz, Lilian, Cridland, Andrew, Kinchin, Elizabeth

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Novel Enantioselective Synthesis of 1,3-Butadien-2-ylmethanols via Tandem Alkylbromide-epoxide Vinylations Using Dimethylsulfonium Methylide von Alcaraz, Lilian, Cox, Katherine, Cridland, Andrew P, Kinchin, Elizabeth, Morris, James, Thompson, Stewart P

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Small Molecule Inhibitors for Precise Inhibition of Alpha-Synuclein Oligomer Generation in Parkinson’s Disease (S32.002) von Thomson, John, Cridland, Andrew, Ball, Sarah, Staats, Roxine, Pandey, Samata, Cruz, Marta Castellana, Pisani, Katarina, Meisl, Georg, Kitchen-Smith, Isaac, Yang, Xiaoting, Mannini, Benedetta, Pollack, Scott, Rajah, Luke, Brewerton, Suzanne, Habchi, Johnny, Plowright, Alleyn

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Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models von Everett, Martin J., Davies, David T., Leiris, Simon, Sprynski, Nicolas, Llanos, Agustina, Castandet, Jérôme M., Lozano, Clarisse, LaRock, Christopher N., LaRock, Doris L., Corsica, Giuseppina, Docquier, Jean-Denis, Pallin, Thomas D., Cridland, Andrew, Blench, Toby, Zalacain, Magdalena, Lemonnier, Marc

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Catalytic enantioselective electrocyclic cascadesElectronic supplementary information (ESI) available: procedures and experimental data for all compounds and crystal structure data... von Maciver, Eleanor E, Knipe, Peter C, Cridland, Andrew P, Thompson, Amber L, Smith, Martin D

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An improved synthesis of (2 E,4 Z)-6-(benzyloxy)-4-bromohexa-2,4-dien-1-ol von Clarke, Paul A., Rolla, Gabriele A., Cridland, Andrew P., Gill, Andrew A.

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COMPOUNDS, COMPOSITIONS, AND MEZHODS OF TREATING DISORDERS ASSOCIATED WITH PROTEIN MISFOLDING von POPOVICI-MULLER, Janeta, PLOWRIGHT, Alleyn Thomas, CRIDLAND, Andrew Peter, JENKINS, Kerry, TAKLE, Andrew Kenneth, HOSHIKAWA, Tamaki

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4  Total synthesis highlights von Clarke, Paul A., Cridland, Andrew P.

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COMBINATION THERAPY von Leiris, Simon, Blench, Toby Jonathan, Davies, David Thomas, Clark, David Edward, Everett, Martin, Beyria, Lilha, Sprynski, Nicolas, Cridland, Andrew Peter, Elliott, Richard Leonard, Pallin, Thomas David

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CHEMICAL COMPOUNDS AS ANTIBIOTICS von PALLIN, THOMAS DAVID, CRIDLAND, ANDREW PETER, EVERETT, MARTIN, ELLIOTT, RICHARD LEONARD, BEYRIA, LILHA, CLARK, DAVID EDWARD, SPRYNSKI, NICOLAS, BLENCH, TOBY JONATHAN, SUTTON, JONATHAN MARK, DAVIES, DAVID THOMAS, LEIRIS, SIMON, BODNARCHUK, MICHAEL STEVEN

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COMBINATION THERAPY von BLENCH, Toby Jonathan, EVERETT, Martin, SPRYNSKI, Nicolas, LEIRIS, Simon, CLARK, David Edward, PALLIN, Thomas David, BEYRIA, Lilha, ELLIOTT, Richard Leonard, CRIDLAND, Andrew Peter, DAVIES, David Thomas

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CHEMICAL COMPOUNDS AS ANTIBIOTICS von BLENCH, Toby Jonathan, EVERETT, Martin, SPRYNSKI, Nicolas, LEIRIS, Simon, CLARK, David Edward, BODNARCHUK, Michael Steven, SUTTON, Jonathan Mark, PALLIN, Thomas David, BEYRIA, Lilha, ELLIOTT, Richard Leonard, CRIDLAND, Andrew Peter, DAVIES, David Thomas

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CHEMICAL COMPOUNDS AS ANTIBIOTICS von BLENCH, Toby Jonathan, EVERETT, Martin, SPRYNSKI, Nicolas, LEIRIS, Simon, CLARK, David Edward, BODNARCHUK, Michael Steven, SUTTON, Jonathan Mark, PALLIN, Thomas David, BEYRIA, Lilha, ELLIOTT, Richard Leonard, CRIDLAND, Andrew Peter, DAVIES, David Thomas

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S1PR4 RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF von GANCIA, Emanuela, BULL, Richard, JACKSON, Philip, KNIGHT, Jamie, LEVENSON, Jonathan Max, LARSON, Kelley Cronin, TATE, Barbara, JENNINGS, Neil, HYND, George, CRIDLAND, Andrew, MILLER, Thomas Allen, MARTENS, Lauren, BRUHN, Suzanne

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