PROTACs: past, present and future von Li, Ke, Crews, Craig M

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Proteolysis-Targeting Chimeras as Therapeutics and Tools for Biological Discovery von Burslem, George M., Crews, Craig M.

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Small-Molecule PROTACS: New Approaches to Protein Degradation von Toure, Momar, Crews, Craig M.

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Recent Developments in PROTAC‐Mediated Protein Degradation: From Bench to Clinic von Hu, Zhenyi, Crews, Craig M.

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PROTACs: An Emerging Therapeutic Modality in Precision Medicine von Nalawansha, Dhanusha A., Crews, Craig M.

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Waste disposal—An attractive strategy for cancer therapy von Salami, Jemilat, Crews, Craig M.

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Targeted Protein Degradation: from Chemical Biology to Drug Discovery von Cromm, Philipp M., Crews, Craig M.

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Major advances in targeted protein degradation: PROTACs, LYTACs, and MADTACs von Alabi, Shanique B., Crews, Craig M.

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Proteolysis-Targeting Chimeras: Induced Protein Degradation as a Therapeutic Strategy von Ottis, Philipp, Crews, Craig M

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MDM2-Recruiting PROTAC Offers Superior, Synergistic Antiproliferative Activity via Simultaneous Degradation of BRD4 and Stabilization of p53 von Hines, John, Lartigue, Schan, Dong, Hanqing, Qian, Yimin, Crews, Craig M

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Targeted Protein Degradation by Small Molecules von Bondeson, Daniel P, Crews, Craig M

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Differential PROTAC substrate specificity dictated by orientation of recruited E3 ligase von Smith, Blake E., Wang, Stephen L., Jaime-Figueroa, Saul, Harbin, Alicia, Wang, Jing, Hamman, Brian D., Crews, Craig M.

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Enhancing Antiproliferative Activity and Selectivity of a FLT‑3 Inhibitor by Proteolysis Targeting Chimera Conversion von Burslem, George M, Song, Jayoung, Chen, Xin, Hines, John, Crews, Craig M

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From epoxomicin to carfilzomib: chemistry, biology, and medical outcomes von Kim, Kyung Bo, Crews, Craig M

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Proteolysis targeting chimeras (PROTACs) come of age: entering the third decade of targeted protein degradation von Bond, Michael J, Crews, Craig M

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Targeting the C481S Ibrutinib-Resistance Mutation in Bruton’s Tyrosine Kinase Using PROTAC-Mediated Degradation von Buhimschi, Alexandru D, Armstrong, Haley A, Toure, Momar, Jaime-Figueroa, Saul, Chen, Timothy L, Lehman, Amy M, Woyach, Jennifer A, Johnson, Amy J, Byrd, John C, Crews, Craig M

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Modular PROTAC Design for the Degradation of Oncogenic BCR-ABL von Lai, Ashton C., Toure, Momar, Hellerschmied, Doris, Salami, Jemilat, Jaime-Figueroa, Saul, Ko, Eunhwa, Hines, John, Crews, Craig M.

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Small-Molecule Control of Intracellular Protein Levels through Modulation of the Ubiquitin Proteasome System von Buckley, Dennis L., Crews, Craig M.

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Targeted degradation of transcription factors by TRAFTACs: TRAnscription Factor TArgeting Chimeras von Samarasinghe, Kusal T.G., Jaime-Figueroa, Saul, Burgess, Michael, Nalawansha, Dhanusha A., Dai, Katherine, Hu, Zhenyi, Bebenek, Adrian, Holley, Scott A., Crews, Craig M.

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Targeting BCR-ABL1 in Chronic Myeloid Leukemia by PROTAC-Mediated Targeted Protein Degradation von Burslem, George M, Schultz, Anna Reister, Bondeson, Daniel P, Eide, Christopher A, Savage Stevens, Samantha L, Druker, Brian J, Crews, Craig M

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