Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P2-Modified, Orally Active Pept... von Cregge, Robert J, Durham, Sherrie L, Farr, Robert A, Gallion, Steven L, Hare, C. Michelle, Hoffman, Robert V, Janusz, Michael J, Kim, Hwa-Ok, Koehl, Jack R, Mehdi, Shujaath, Metz, William A, Peet, Norton P, Pelton, John T, Schreuder, Herman A, Sunder, Shyam, Tardif, Chantal

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Design, Synthesis, and Conformational Analysis of a Novel Macrocyclic HIV-Protease Inhibitor von Podlogar, Brent L, Farr, Robert A, Friedrich, Dirk, Tarnus, Celine, Huber, Edward W, Cregge, Robert J, Schirlin, Daniel

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Total synthesis of the indole alkaloids dl-eburnamonine and dl-vincamine von Herrmann, J. L, Cregge, R. J, Richman, J. E, Kieczykowski, G. R, Normandin, S. N, Quesada, M. L, Semmelhack, C. L, Poss, A. J, Schlessinger, R. H

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Conformationally restricted leukotriene antagonists. Asymmetric synthesis of some nor-leukotriene D4 analogs von SABOL, J. S, CREGGE, R. J

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High yield stereospecific total synthesis of vincamine von Herrmann, J. L, Cregge, R. J, Richman, J. E, Semmelhack, C. L, Schlessinger, R. H

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Conformationally restricted leukotriene antagonists. Synthesis of some leukotriene D4 analogs from D-xylose von SABOL, J. S, CREGGE, R. J

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1',3'-Dicyclohexylspiro[2H-1-benzopyran-2,4'-imidazolidine]-2',4(3H),5'-trione, C23H28N2O4 von Bates, R. B., Camou, F. A., Cregge, R. J.

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CoMFA, Synthesis, and Pharmacological Evaluation of (E)-3-(2-Carboxy-2-arylvinyl)-4,6-dichloro-1H-indole-2-carboxylic Acids: 3-[2-(3-Aminophenyl)-2-carboxyvinyl]-4,6-dichloro-1H-in... von Baron, B M, Cregge, R J, Farr, R A, Friedrich, D, Gross, R S, Harrison, B L, Janowick, DA, Matthews, D, McCloskey, T C, Meikrantz, S, Nyce, P L, Vaz, R, Metz, WA

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Large-scale synthesis of anticoagulant decapeptide MDL 28050 von Hoekstra, William J., Sunder, Shyam S., Cregge, Robert J., Ashton, Louis A., Stewart, Kenneth T., King, Chi-Hsin R.

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Conformationally restricted leukotriene antagonists. Stereoselective synthesis of some leukotriene D4 analogs von SABOL, J. S, WEINTRAUB, P. M, GIESKE, T. H, CREGGE, R. J

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Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P 2 -Modified, Orally Active Pe... von Cregge, Robert J., Durham, Sherrie L., Farr, Robert A., Gallion, Steven L., Hare, C. Michelle, Hoffman, Robert V., Janusz, Michael J., Kim, Hwa-Ok, Koehl, Jack R., Mehdi, Shujaath, Metz, William A., Peet, Norton P., Pelton, John T., Schreuder, Herman A., Sunder, Shyam, Tardif, Chantal

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Identification in man of urinary metabolites of a new bronchodilator, MDL 257, using triple stage quadrupole mass spectrometry-mass spectrometry von Coutant, John E., Barbuch, Robert J., Satonin, Darlene K., Cregge, Robert J.

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Synthesis of (E)-3-(2-carboxy-2-pyridyl-vinyl)-4,6-dichloro-1H-indole-2-carboxylic acids, glycine-site NMDA receptor antagonists, utilizing the Knoevenagel condensation reaction von Cregge, Robert J, Farr, Robert A, Friedrich, Dirk, Hulshof, Jos, Janowick, David A, Meikrantz, Scott, Metz, William A

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A convenient one flask procedure for ester alkylation von Cregge, R.J., Herrmann, J.L., Lee, C.S., Richman, J.E., Schlessinger, R.H.

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Comparative evaluation of the relaxant effects of MDL-257, its metabolites, and some related compounds on guinea pig tracheal cylindrical segments von ABDALLAH, A. H, BURNELL, J. W, CREGGE, R. J

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A versatile and reactive michael receptor for the synthesis of 1,4 -dicarbonyl compounds von Cregge, R.J., Herrmann, J.L., Schlessinger, R.H.

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Lipase-catalyzed transesterification in the synthesis of a new chiral unlabeled and carbon-14 labeled serotonin uptake inhibitor von Cregge, Robert J, Wagner, Eugene R, Freedman, Jules, Margolin, Alexey L

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Conformationally restricted leukotriene antagoniste: asymmetric synthesis of a nor-leukotriene D4 analog. II von SABOL, J. S, CREGGE, R. J

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The conjugate addition of a glyoxalate derived carbonyl anion equivalent and its application to the synthesis of 1,4-dicarbonyl compounds von Cregge, R.J., Herrmann, J.L., Richman, J.E., Romanet, R.F., Schlessinger, R.H.

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A convenient synthesis of peptidyl perfluoroalkyl ketones von Cregge, Robert J., Curran, Timothy T., Metz, William A.

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