Discovery of an Orally Bioavailable Benzimidazole Diacylglycerol Acyltransferase 1 (DGAT1) Inhibitor That Suppresses Body Weight Gain in Diet-Induced Obese Dogs and Postprandial Tr... von Nakajima, Katsumasa, Chatelain, Ricardo, Clairmont, Kevin B, Commerford, Renee, Coppola, Gary M, Daniels, Thomas, Forster, Cornelia J, Gilmore, Thomas A, Gong, Yongjin, Jain, Monish, Kanter, Aaron, Kwak, Youngshin, Li, Jingzhou, Meyers, Charles D, Neubert, Alan D, Szklennik, Paul, Tedesco, Vivienne, Thompson, James, Truong, David, Yang, Qing, Hubbard, Brian K, Serrano-Wu, Michael H

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Structure-Guided Design of Substituted Biphenyl Butanoic Acid Derivatives as Neprilysin Inhibitors von Kawanami, Toshio, Karki, Rajeshri G, Cody, Emma, Liu, Qian, Liang, Guiqing, Ksander, Gary M, Rigel, Dean F, Schiering, Nikolaus, Gong, Yongjin, Coppola, Gary M, Iwaki, Yuki, Sun, Robert, Neubert, Alan, Fan, Li, Ingles, Sara, D’Arcy, Allan, Villard, Frederic, Ramage, Paul, Jeng, Arco Y, Leung-Chu, Jennifer, Liu, Jing, Beil, Michael, Fu, Fumin, Chen, Wei, Cumin, Frederic, Wiesmann, Christian, Mogi, Muneto

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Intestinally Targeted Diacylglycerol Acyltransferase 1 (DGAT1) Inhibitors Robustly Suppress Postprandial Triglycerides von Serrano-Wu, Michael H, Coppola, Gary M, Gong, Yongjin, Neubert, Alan D, Chatelain, Ricardo, Clairmont, Kevin B, Commerford, Renee, Cosker, Theresa, Daniels, Thomas, Hou, Ying, Jain, Monish, Juedes, Marlene, Li, Lisha, Mullarkey, Tara, Rocheford, Erik, Sung, Moo Je, Tyler, Andrew, Yang, Qing, Yoon, Taeyoung, Hubbard, Brian K

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Perhydroquinolylbenzamides as Novel Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 von Coppola, Gary M, Kukkola, Paivi J, Stanton, James L, Neubert, Alan D, Marcopulos, Nicholas, Bilci, Natalie A, Wang, Hua, Tomaselli, Hollis C, Tan, Jenny, Aicher, Thomas D, Knorr, Douglas C, Jeng, Arco Y, Dardik, Beatriz, Chatelain, Ricardo E

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The chemistry of 4H-3,1-benzoxazin-4-ones von Coppola, Gary M.

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Synthesis and reactions of 2-hetero-4H-3,1-benzoxazin-4-ones von Coppola, Gary M.

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Biological evaluation of 1-alkyl-3-phenylthioureas as orally active HDL-elevating agents von Coppola, Gary M., Damon, Robert E., Eskesen, J. Bruce, France, Dennis S., Paterniti, James R.

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1-Hydroxyalkyl-3-phenylthioureas as novel HDL-elevating agents von Coppola, Gary M., Damon, Robert E., Eskesen, J. Bruce, France, Dennis S., Paterniti, James R.

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Secondary Amides of (R)-3,3,3-Trifluoro-2-hydroxy-2-methylpropionic Acid as Inhibitors of Pyruvate Dehydrogenase Kinase von Aicher, Thomas D, Anderson, Robert C, Gao, Jiaping, Shetty, Suraj S, Coppola, Gary M, Stanton, James L, Knorr, Douglas C, Sperbeck, Donald M, Brand, Leonard J, Vinluan, Christine C, Kaplan, Emma L, Dragland, Carol J, Tomaselli, Hollis C, Islam, Amin, Lozito, Robert J, Liu, Xilin, Maniara, Wieslawa M, Fillers, William S, DelGrande, Dominick, Walter, R. Eric, Mann, William R

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1-Aminomethylisoquinoline-4-carboxylates as novel dipeptidylpeptidase IV inhibitors von Coppola, Gary M, Zhang, Y.Larry, Schuster, Herbert F, Russell, Mary E, Hughes, Thomas E

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Thiourea-based gemfibrozil analogues as HDL-elevating agents von Coppola, Gary M, Damon, Robert E, Eskesen, J.Bruce, France, Dennis S, Paterniti, James R

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In Vitro Metabolism of N-(5-Chloro-2-methylphenyl)-N‘-(2-methylpropyl)thiourea:  Species Comparison and Identification of a Novel Thiocarbamide−Glutathione Adduct von Stevens, Gregory J, Hitchcock, Karen, Wang, Y. Karen, Coppola, Gary M, Versace, Richard W, Chin, Jefferson A, Shapiro, Michael, Suwanrumpha, Somchai, Mangold, Bonnie L. K

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A Mild and Efficient Preparation of Carbodiimides von Fell, Jay B., Coppola, Gary M.

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Amberlyst-15, A Superior Acid Catalyst for the Cleavage of Acetals von Coppola, Gary M.

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A new scavenger resin for amines von Coppola, Gary M.

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The Chemistry of 2H-3,1-Benzoxazine-2,4(1H)-dione (Isatoic Anhydride). 201. Synthesis and Wittig Reactions of Dimethyl (4-Oxo-1,4-dihydro-Quinolin-2-yl)methanephosphonates von Coppola, Gary M.

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Synthesis and reactions of 2‐hetero‐4 H ‐3,1‐benzoxazin‐4‐ones von Coppola, Gary M.

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The chemistry of 4 H ‐3,1‐benzoxazin‐4‐ones von Coppola, Gary M.

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(R)-3,3,3-Trifluoro-2-hydroxy-2-methylpropionamides Are Orally Active Inhibitors of Pyruvate Dehydrogenase Kinase von Aicher, Thomas D, Anderson, Robert C, Bebernitz, Gregory R, Coppola, Gary M, Jewell, Charles F, Knorr, Douglas C, Liu, Charles, Sperbeck, Donald M, Brand, Leonard J, Strohschein, Robert J, Gao, Jiaping, Vinluan, Christine C, Shetty, Suraj S, Dragland, Carol, Kaplan, Emma L, DelGrande, Dominick, Islam, Amin, Liu, Xilin, Lozito, Robert J, Maniara, Wieslawa M, Walter, R. Erik, Mann, William R

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Perhydroquinolylbenzamides as novel inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 von Coppola, Gary M, Kukkola, Paivi J, Stanton, James L, Neubert, Alan D, Marcopulos, Nicholas, Bilci, Natalie A, Wang, Hua, Tomaselli, Hollis C, Tan, Jenny, Aicher, Thomas D, Knorr, Douglas C, Jeng, Arco Y, Dardik, Beatriz, Chatelain, Ricardo E

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