Bioisosteric Replacements of the Pyrazole Moiety of Rimonabant:  Synthesis, Biological Properties, and Molecular Modeling Investigations of Thiazoles, Triazoles, and Imidazoles as... von Lange, Jos H. M, van Stuivenberg, Herman H, Coolen, Hein K. A. C, Adolfs, Tiny J. P, McCreary, Andrew C, Keizer, Hiskias G, Wals, Henri C, Veerman, Willem, Borst, Alice J. M, de Looff, Wouter, Verveer, Peter C, Kruse, Chris G

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Design, Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel Tacrine Derivatives with a Combination of Acetylcholinesterase Inhibition and Cannabinoid C... von Lange, Jos H. M, Coolen, Hein K. A. C, van der Neut, Martina A. W, Borst, Alice J. M, Stork, Bob, Verveer, Peter C, Kruse, Chris G

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Synthesis, Structure−Activity Relationships, and Biological Properties of 1-Heteroaryl-4-[ω-(1H-indol-3-yl)alkyl]piperazines, Novel Potential Antipsychotics Combining Potent Dopami... von Smid, Pieter, Coolen, Hein K. A. C, Keizer, Hiskias G, van Hes, Rolf, de Moes, Jan-Peter, den Hartog, Arnold P, Stork, Bob, Plekkenpol, Rob H, Niemann, Leonarda C, Stroomer, Cees N. J, Tulp, Martin Th. M, van Stuivenberg, Herman H, McCreary, Andrew C, Hesselink, Mayke B, Herremans, Arnoud H. J, Kruse, Chris G

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7-Azaindole derivatives as potential partial nicotinic agonists von Stoit, Axel R., den Hartog, Arnold P., Mons, Harry, van Schaik, Sjoerd, Barkhuijsen, Nynke, Stroomer, Cees, Coolen, Hein K.A.C., Reinders, Jan Hendrik, Adolfs, Tiny J.P., van der Neut, Martina, Keizer, Hiskias, Kruse, Chris G.

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Principal Component Analysis Differentiates the Receptor Binding Profiles of Three Antipsychotic Drug Candidates from Current Antipsychotic Drugs von Lange, Jos H. M, Reinders, Jan-Hendrik, Tolboom, Jeroen T. B. M, Glennon, Jeffrey C, Coolen, Hein K. A. C, Kruse, Chris G

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Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel 3,4-Diarylpyrazolines as Potent and Selective CB1 Cannabinoid Receptor Antagonists von Lange, Jos H. M, Coolen, Hein K. A. C, van Stuivenberg, Herman H, Dijksman, Jessica A. R, Herremans, Arnoud H. J, Ronken, Eric, Keizer, Hiskias G, Tipker, Koos, McCreary, Andrew C, Veerman, Willem, Wals, Henri C, Stork, Bob, Verveer, Peter C, den Hartog, Arnold P, de Jong, Natasja M. J, Adolfs, Tiny J. P, Hoogendoorn, Jan, Kruse, Chris G

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Novel 3,4-diarylpyrazolines as potent cannabinoid CB1 receptor antagonists with lower lipophilicity von LANGE, Jos H. M, VAN STUIVENBERG, Herman H, VEERMAN, Willem, WALS, Henri C, STORK, Bob, COOLEN, Hein K. A. C, MCCREARY, Andrew C, ADOLFS, Tiny J. P, KRUSE, Chris G

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Substrate Selective Catalysis by Rhodium Metallohosts von Coolen, Hein K. A. C, Meeuwis, Johannes A. M, van Leeuwen, Piet W. M. N, Nolte, Roeland J. M

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Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P5 receptor agonist chemotype von Stoit, Axel R., Lange, Jos H.M., Coolen, Hein K.A.C., Rensink, Annemieke, van den Hoogenband, Adri, den Hartog, Arnold P., van Schaik, Sjoerd, Kruse, Chris G.

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Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P 5 receptor agonist chemotype von Stoit, Axel R, Lange, Jos H M, Coolen, Hein K A C, Rensink, Annemieke, van den Hoogenband, Adri, den Hartog, Arnold P, van Schaik, Sjoerd, Kruse, Chris G

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Synthesis and Conformational Behavior of Rhodium(I) Metallohosts Derived from Diphenylglycoluril von Coolen, Hein K. A. C, van Leeuwen, Piet W. N. M, Nolte, Roeland J. M

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Design, Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel Tacrine Derivatives with a Combination of Acetylcholinesterase Inhibition and Cannabinoid C... von Lange, Jos H. M., Coolen, Hein K. A. C., van der Neut, Martina A. W., Borst, Alice J. M., Stork, Bob, Verveer, Peter C., Kruse, Chris G.

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Bioisosteric Replacements of the Pyrazole Moiety of Rimonabant:  Synthesis, Biological Properties, and Molecular Modeling Investigations of Thiazoles, Triazoles, and Imidazoles as... von Lange, Jos H. M., van Stuivenberg, Herman H., Coolen, Hein K. A. C., Adolfs, Tiny J. P., McCreary, Andrew C., Keizer, Hiskias G., Wals, Henri C., Veerman, Willem, Borst, Alice J. M., de Looff, Wouter, Verveer, Peter C., Kruse, Chris G.

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Synthesis, Structure−Activity Relationships, and Biological Properties of 1-Heteroaryl-4-[ω-(1 H -indol-3-yl)alkyl]piperazines, Novel Potential Antipsychotics Combining Potent Dopa... von Smid, Pieter, Coolen, Hein K. A. C., Keizer, Hiskias G., van Hes, Rolf, de Moes, Jan-Peter, den Hartog, Arnold P., Stork, Bob, Plekkenpol, Rob H., Niemann, Leonarda C., Stroomer, Cees N. J., Tulp, Martin Th. M., van Stuivenberg, Herman H., McCreary, Andrew C., Hesselink, Mayke B., Herremans, Arnoud H. J., Kruse, Chris G.

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Spiro-cyclic amine derivatives as S1P modulators von Stoit, Axel, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Leflemme, Nicolas J.-L. D, van Dongen, Maria J. P

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Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists von Lange, Jos H M, Coolen, Hein K A C, van Stuivenberg, Herman H, Dijksman, Jessica A R, Herremans, Arnoud H J, Ronken, Eric, Keizer, Hiskias G, Tipker, Koos, McCreary, Andrew C, Veerman, Willem, Wals, Henri C, Stork, Bob, Verveer, Peter C, den Hartog, Arnold P, de Jong, Natasja M J, Adolfs, Tiny J P, Hoogendoorn, Jan, Kruse, Chris G

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Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel 3,4-Diarylpyrazolines as Potent and Selective CB 1 Cannabinoid Receptor Antagonists von Lange, Jos H. M., Coolen, Hein K. A. C., van Stuivenberg, Herman H., Dijksman, Jessica A. R., Herremans, Arnoud H. J., Ronken, Eric, Keizer, Hiskias G., Tipker, Koos, McCreary, Andrew C., Veerman, Willem, Wals, Henri C., Stork, Bob, Verveer, Peter C., den Hartog, Arnold P., de Jong, Natasja M. J., Adolfs, Tiny J. P., Hoogendoorn, Jan, Kruse, Chris G.

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A RhI-Centered Cage Compound with Selective Catalytic Properties von Coolen, Hein K. A. C., van Leeuwen, Piet W. N. M., Nolte, Roeland J. M.

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Fused heterocyclic derivatives as S1P modulators von Smid, Pieter, den Hartog, Jacobus A. J, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Sliedregt, Leonardus A. J. M, van Dongen, Maria J. P

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Spiro-cyclic amine derivatives as S1P modulators von Stoit, Axel, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Leflemme, Nicolas J.-L. D, van Dongen, Maria J. P

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