Photoredox-catalyzed deuteration and tritiation of pharmaceutical compounds von Loh, Yong Yao, Nagao, Kazunori, Hoover, Andrew J., Hesk, David, Rivera, Nelo R., Colletti, Steven L., Davies, Ian W., MacMillan, David W. C.

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Cheminformatic analysis of natural product-based drugs and chemical probes von Stone, Samantha, Newman, David J, Colletti, Steven L, Tan, Derek S

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Chemoselective Peptide Modification via Photocatalytic Tryptophan β‑Position Conjugation von Yu, Younong, Zhang, Li-Kang, Buevich, Alexei V, Li, Guoqing, Tang, Haiqun, Vachal, Petr, Colletti, Steven L, Shi, Zhi-Cai

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Profiling and Application of Photoredox C(sp3)–C(sp2) Cross-Coupling in Medicinal Chemistry von Zhang, Rui, Li, Guoqing, Wismer, Michael, Vachal, Petr, Colletti, Steven L., Shi, Zhi-Cai

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International Union of Basic and Clinical Pharmacology. LXXXII: Nomenclature and Classification of Hydroxy-carboxylic Acid Receptors (GPR81, GPR109A, and GPR109B) von Offermanns, Stefan, Colletti, Steven L, Lovenberg, Timothy W, Semple, Graeme, Wise, Alan, IJzerman, Adriaan P

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Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40 von Lu, Jun, Byrne, Noel, Wang, John, Bricogne, Gerard, Brown, Frank K, Chobanian, Harry R, Colletti, Steven L, Di Salvo, Jerry, Thomas-Fowlkes, Brande, Guo, Yan, Hall, Dawn L, Hadix, Jennifer, Hastings, Nicholas B, Hermes, Jeffrey D, Ho, Thu, Howard, Andrew D, Josien, Hubert, Kornienko, Maria, Lumb, Kevin J, Miller, Michael W, Patel, Sangita B, Pio, Barbara, Plummer, Christopher W, Sherborne, Bradley S, Sheth, Payal, Souza, Sarah, Tummala, Srivanya, Vonrhein, Clemens, Webb, Maria, Allen, Samantha J, Johnston, Jennifer M, Weinglass, Adam B, Sharma, Sujata, Soisson, Stephen M

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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent von Pachanski, Michele J, Kirkland, Melissa E, Kosinski, Daniel T, Mane, Joel, Cheewatrakoolpong, Boonlert, Xue, Jiyan, Szeto, Daphne, Forrest, Gail, Miller, Corin, Bunzel, Michelle, Plummer, Christopher W, Chobanian, Harry R, Miller, Michael W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Li, Xiaoyan, Feng, Yue, Tatosian, Daniel A, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E

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Discovery of platencin, a dual FabF and FabH inhibitor with in vivo antibiotic properties von Wang, Jun, Kodali, Srinivas, Lee, Sang Ho, Galgoci, Andrew, Painter, Ronald, Dorso, Karen, Racine, Fred, Motyl, Mary, Hernandez, Lorraine, Tinney, Elizabeth, Colletti, Steven L, Herath, Kithsiri, Cummings, Richard, Salazar, Oscar, González, Ignacio, Basilio, Angela, Vicente, Francisca, Genilloud, Olga, Pelaez, Fernando, Jayasuriya, Hiranthi, Young, Katherine, Cully, Doris F, Singh, Sheo B

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GPR40 reduces food intake and body weight through GLP-1 von Gorski, Judith N, Pachanski, Michele J, Mane, Joel, Plummer, Christopher W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Cheewatrakoolpong, Boonlert, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E

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Medicinal Chemistry of siRNA Delivery von Stanton, Matthew G, Colletti, Steven L

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Palladium-Catalyzed Suzuki−Miyaura Coupling of Pyridyl-2-boronic Esters with Aryl Halides Using Highly Active and Air-Stable Phosphine Chloride and Oxide Ligands von Yang, David X, Colletti, Steven L, Wu, Kevin, Song, Maoying, Li, George Y, Shen, Hong C

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Systematic chemical modifications of single stranded siRNAs significantly improved CTNNB1 mRNA silencing von Chang, Wonsuk, Pei, Yi, Guidry, Erin N., Zewge, Daniel, Parish, Craig A., Sherer, Edward C., DiMuzio, Jillian, Zhang, Hangchun, South, Victoria J., Strapps, Walter R., Sepp-Lorenzino, Laura, Colletti, Steven L., Stanton, Matthew G.

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Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs von Pio, Barbara, Chobanian, Harry R., Guo, Yan, Josien, Hubert, Hagmann, William K., Miller, Michael, Trujillo, Maria E., Kirkland, Melissa, Kosinski, Daniel, Mane, Joel, Pachanski, Michele, Cheewatrakoolpong, Boonlert, Ashley, Eric, Orr, Robert, Wright, Michael J., Bugianesi, Randal, Souza, Sarah, Zhang, Xiaoping, Di Salvo, Jerry, Weinglass, Adam B., Tschirret-Guth, Richard, Samuel, Koppara, Chen, Qing, Shang, Jackie, Lamca, James, Ehrhart, Juliann, Nargund, Ravi, Howard, Andrew D., Colletti, Steven L.

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Synthesis of novel 2-azabicyclo[3.1.1]heptane-5-carboxylic acid von He, Shuwen, Hao, Jinsong, Ashley, Eric R., Chobanian, Harry R., Pio, Barbara, Colletti, Steven L., Miller, Michael

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Gold(I)-Catalyzed Regioselective Cyclizations of Silyl Ketene Amides and Carbamates with Alkynes von Minnihan, Ellen C, Colletti, Steven L, Toste, F. Dean, Shen, Hong C

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Endosomolytic Bioreducible Poly(amido amine disulfide) Polymer Conjugates for the in Vivo Systemic Delivery of siRNA Therapeutics von Parmar, Rubina Giare, Busuek, Marina, Walsh, Eileen S, Leander, Karen R, Howell, Bonnie J, Sepp-Lorenzino, Laura, Kemp, Eric, Crocker, Louis S, Leone, Anthony, Kochansky, Christopher J, Carr, Brian A, Garbaccio, Robert M, Colletti, Steven L, Wang, Weimin

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Structure–Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs von Chen, Helen Y., Plummer, Christopher W., Xiao, Dong, Chobanian, Harry R., DeMong, Duane, Miller, Michael, Trujillo, Maria E., Kirkland, Melissa, Kosinski, Daniel, Mane, Joel, Pachanski, Michele, Cheewatrakoolpong, Boonlert, Di Salvo, Jerry, Thomas-Fowlkes, Brande, Souza, Sarah, Tatosian, Daniel A., Chen, Qing, Hafey, Michael J., Houle, Robert, Nolting, Andrew F., Orr, Robert, Ehrhart, Juliann, Weinglass, Adam B., Tschirret-Guth, Richard, Howard, Andrew D., Colletti, Steven L.

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Novel Endosomolytic Poly(amido amine) Polymer Conjugates for Systemic Delivery of siRNA to Hepatocytes in Rodents and Nonhuman Primates von Parmar, Rubina Giare, Poslusney, Micheal, Busuek, Marina, Williams, J. Michael, Garbaccio, Robert, Leander, Karen, Walsh, Eileen, Howell, Bonnie, Sepp-Lorenzino, Laura, Riley, Sean, Patel, Mihir, Kemp, Eric, Latham, Andrew, Leone, Anthony, Soli, Eric, Burke, Rob S, Carr, Brian, Colletti, Steven L, Wang, Weimin

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(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic Acid (MK-1903): A Potent GPR109a Agonist that Lowers Free Fatty Acids in Humans von Boatman, P. Douglas, Lauring, Brett, Schrader, Thomas O, Kasem, Michelle, Johnson, Benjamin R, Skinner, Philip, Jung, Jae-Kyu, Xu, Jerry, Cherrier, Martin C, Webb, Peter J, Semple, Graeme, Sage, Carleton R, Knudsen, Jens, Chen, Ruoping, Luo, Wen-Lin, Caro, Luzelena, Cote, Josee, Lai, Eseng, Wagner, John, Taggart, Andrew K, Carballo-Jane, Ester, Hammond, Milton, Colletti, Steven L, Tata, James R, Connolly, Daniel T, Waters, M. Gerard, Richman, Jeremy G

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Development of a liver-targeted siRNA delivery platform with a broad therapeutic window utilizing biodegradable polypeptide-based polymer conjugates von Barrett, Stephanie E., Burke, Rob S., Abrams, Marc T., Bason, Carol, Busuek, Marina, Carlini, Edward, Carr, Brian A., Crocker, Louis S., Fan, Haihong, Garbaccio, Robert M., Guidry, Erin N., Heo, Jun H., Howell, Bonnie J., Kemp, Eric A., Kowtoniuk, Robert A., Latham, Andrew H., Leone, Anthony M., Lyman, Michael, Parmar, Rubina G., Patel, Mihir, Pechenov, Sergey Y., Pei, Tao, Pudvah, Nicole T., Raab, Conrad, Riley, Sean, Sepp-Lorenzino, Laura, Smith, Sheri, Soli, Eric D., Staskiewicz, Steven, Stern, Melissa, Truong, Quang, Vavrek, Marissa, Waldman, Jacob H., Walsh, Eileen S., Williams, J. Michael, Young, Stephanie, Colletti, Steven L.

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