Catalytic Asymmetric Synthesis of tert-Butanesulfinamide. Application to the Asymmetric Synthesis of Amines von Liu, Guangcheng, Cogan, Derek A, Ellman, Jonathan A

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Dihydrobenzisoxazole-4-one compounds are novel selective inhibitors of aldosterone synthase (CYP11B2) with in vivo activity von Meyers, Kenneth, Cogan, Derek A., Burke, Jennifer, Arenas, Raquel, Balestra, Michael, Brown, Nicholas F., Chen, Zhidong, Cerny, Matthew A., Clifford, Holly E., Colombo, Federico, Fader, Lee, Frederick, Kosea S., Guo, Xin, Goldberg, Daniel, Hornberger, Keith R., Kugler, Stanley, Lord, John, Marshall, Daniel R., Moss, Neil, Parmentier, Jean-Huges, Richman, Jeremy R., Schmenk, Jennifer, Weldon, Steven M., Yu, Maolin, Zhang, Michael

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Asymmetric Synthesis of α,α-Dibranched Amines by the Trimethylaluminum-Mediated 1,2-Addition of Organolithiums to tert-Butanesulfinyl Ketimines von Cogan, Derek A, Ellman, Jonathan A

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Catalytic Asymmetric Oxidation of tert-Butyl Disulfide. Synthesis of tert-Butanesulfinamides, tert-Butyl Sulfoxides, and tert-Butanesulfinimines von Cogan, Derek A, Liu, Guangcheng, Kim, Kyungjin, Backes, Bradley J, Ellman, Jonathan A

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Re-awakening Innate Immune Signaling in Cancer: The Development of Highly Potent ENPP1 Inhibitors von Cogan, Derek, Bakhoum, Samuel F.

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Discovery of potent and selective PKC-θ inhibitors von Cywin, Charles L., Dahmann, Georg, Prokopowicz, Anthony S., Young, Erick R.R., Magolda, Ronald L., Cardozo, Mario G., Cogan, Derek A., DiSalvo, Darren, Ginn, John D., Kashem, Mohammed A., Wolak, John P., Homon, Carol A., Farrell, Thomas M., Grbic, Heather, Hu, Hanbo, Kaplita, Paul V., Liu, Lisa H., Spero, Denice M., Jeanfavre, Deborah D., O’Shea, Kathy M., White, Della M., Woska, Joseph R., Brown, Maryanne L.

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Applications of Zr-Catalyzed Carbomagnesation and Mo-Catalyzed Macrocyclic Ring Closing Metathesis in Asymmetric Synthesis. Enantioselective Total Synthesis of Sch 38516 (Fluviruci... von Xu, Zhongmin, Johannes, Charles W, Houri, Ahmad F, La, Daniel S, Cogan, Derek A, Hofilena, Gloria E, Hoveyda, Amir H

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Discovery of potent, orally active KIF18A inhibitors targeting CIN-high cancer cells von Zhang, Rumin, Cogan, Derek, Eng, Christina, Phillips, Aaron, Carty, Marysol Chu, Feinberg, Tamar, Verma, Akanksha, Tourdot, Richard, Swiston, Albert, Bettigole, Sarah, Drutman, Scott, Su, Michael

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Cascade Catalysis in Synthesis. An Enantioselective Route to Sch 38516 (and Fluvirucin B1) Aglycon Macrolactam von Houri, Ahmad F, Xu, Zhongmin, Cogan, Derek A, Hoveyda, Amir H

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Selectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman Primates von Weldon, Steven M, Cerny, Matthew A, Gueneva-Boucheva, Kristina, Cogan, Derek, Guo, Xin, Moss, Neil, Parmentier, Jean-Hugues, Richman, Jeremy R, Reinhart, Glenn A, Brown, Nicholas F

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Abstract 517: Targeting chromosomally unstable tumors with a selective KIF18A inhibitor von Phillips, Aaron F., Zhang, Rumin, Verma, Akanksha, Feinberg, Tamar, Jaffe, Mia, Carty, Marysol Chu, Schulz, Ryan, Bettigole, Sarah, Andreu, Celia, Drutman, Scott, Su, Michael, Cogan, Derek, Eng, Christina H.

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TRICYCLIC SULFOXIMINE INHIBITORS OF ENPP1 von COGAN, Derek

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INDOLINE COMPOUNDS FOR INHIBITING KIF18A von COGAN, Derek A

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Indole RSK inhibitors. Part 1: Discovery and initial SAR von Boyer, Stephen J., Burke, Jennifer, Guo, Xin, Kirrane, Thomas M., Snow, Roger J., Zhang, Yunlong, Sarko, Chris, Soleymanzadeh, Lida, Swinamer, Alan, Westbrook, John, DiCapua, Frank, Padyana, Anil, Cogan, Derek, Gao, Amy, Xiong, Zhaoming, Madwed, Jeffrey B., Kashem, Mohammed, Kugler, Stanley, O’Neill, Margaret M.

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Spiro indoline inhibitors of kif18a von COGAN Derek A

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SPIRO INDOLINE INHIBITORS OF KIF18A von COGAN, Derek A

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COMPOUNDS FOR INHIBITING KIF18A von COGAN, Derek A

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COMPOUNDS FOR INHIBITING KIF18A von COGAN, Derek A

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Exploration of cathepsin S inhibitors characterized by a triazole P1–P2 amide replacement von Moss, Neil, Xiong, Zhaoming, Burke, Mike, Cogan, Derek, Gao, Donghong A., Haverty, Kathleen, Heim-Riether, Alexander, Hickey, Eugene R., Nagaraja, Raj, Netherton, Matthew, O’Shea, Kathy, Ramsden, Philip, Schwartz, Racheline, Shih, Daw-Tsun, Ward, Yancey, Young, Erick, Zhang, Qing

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INDOLINE COMPOUNDS FOR INHIBITING KIF18A von COGAN, Derek A

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