A highly productive, whole-cell DERA chemoenzymatic process for production of key lactonized side-chain intermediates in statin synthesis von Ošlaj, Matej, Cluzeau, Jérôme, Orkić, Damir, Kopitar, Gregor, Mrak, Peter, Casar, Zdenko

Volltext

Glasdegib Dimaleate: Synthesis, Characterization and Comparison of Its Properties with Monomaleate Analogue von Peklar, Boris, Perdih, Franc, Makuc, Damjan, Plavec, Janez, Cluzeau, Jérôme, Kitanovski, Zoran, Časar, Zdenko

Volltext

Concise Six-Step Asymmetric Approach to Ramelteon from an Acetophenone Derivative Using Ir, Rh, Cu, and Ni Catalysis von Cluzeau, Jérôme, Nettekoven, Ulrike, Kovačevič, Miroslav Planinc, Časar, Zdenko

Volltext

Development and optimization of a new synthetic process for lorcaserin von Cluzeau, Jérôme, Stavber, Gaj

Volltext

Structure–activity relationship study on small peptidic GPR54 agonists von Tomita, Kenji, Niida, Ayumu, Oishi, Shinya, Ohno, Hiroaki, Cluzeau, Jérôme, Navenot, Jean-Marc, Wang, Zi-xuan, Peiper, Stephen C., Fujii, Nobutaka

Volltext

SAR and QSAR Studies on the N-Terminally Acylated Pentapeptide Agonists for GPR54 von Tomita, Kenji, Oishi, Shinya, Cluzeau, Jérôme, Ohno, Hiroaki, Navenot, Jean-Marc, Wang, Zi-xuan, Peiper, Stephen C, Akamatsu, Miki, Fujii, Nobutaka

Volltext

Calcitonin Gene-Related Peptide Analogues with Aza and Indolizidinone Amino Acid Residues Reveal Conformational Requirements for Antagonist Activity at the Human Calcitonin Gene-Re... von Boeglin, Damien, Hamdan, Fadi F, Melendez, Rosa E, Cluzeau, Jérôme, Laperriere, Andre, Héroux, Madeleine, Bouvier, Michel, Lubell, William D

Volltext

Structure-Activity Relationships of Pyrazine-Based CK2 Inhibitors: Synthesis and Evaluation of 2,6-Disubstituted Pyrazines and 4,6-Disubstituted Pyrimidines von Suzuki, Yamato, Cluzeau, Jérôme, Hara, Takafumi, Hirasawa, Akira, Tsujimoto, Gozoh, Oishi, Shinya, Ohno, Hiroaki, Fujii, Nobutaka

Volltext

Structure−Activity Relationships of Cyclic Peptide-Based Chemokine Receptor CXCR4 Antagonists:  Disclosing the Importance of Side-Chain and Backbone Functionalities von Ueda, Satoshi, Oishi, Shinya, Wang, Zi-xuan, Araki, Takanobu, Tamamura, Hirokazu, Cluzeau, Jérôme, Ohno, Hiroaki, Kusano, Shuichi, Nakashima, Hideki, Trent, John O., Peiper, Stephen C., Fujii, Nobutaka

Volltext

Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists von Cluzeau, Jérôme, Oishi, Shinya, Ohno, Hiroaki, Wang, Zixuan, Evans, Barry, Peiper, Stephen C, Fujii, Nobutaka

Volltext

Design, synthesis, and application of azabicyclo[X.Y.0]alkanone amino acids as constrained dipeptide surrogates and peptide mimics von Cluzeau, Jérôme, Lubell, William D.

Volltext

Application of Chemoselective Pancreatin Powder-Catalyzed Deacetylation Reaction in the Synthesis of Key Statin Side Chain Intermediate (4R,6S)-4-(tert-Butyldimethylsilyloxy)-6-(hy... von Troiani, Vincent, Cluzeau, Jérôme, Časar, Zdenko

Volltext

Synthesis of enantiopure antiobesity drug lorcaserin von Smilovic, Ivana Gazic, Cluzeau, Jerome, Richter, Frank, Nerdinger, Sven, Schreiner, Erwin, Laus, Gerhard, Schottenberger, Herwig

Volltext

Conformationally Constrained Dipeptide Surrogates with Aromatic Side-Chains:  Synthesis of 4-Aryl Indolizidin-9-one Amino Acids by Conjugate Addition to a Common α,ω-Diaminoazelate... von Cluzeau, Jérôme, Lubell, William D

Volltext

Structure−Activity Study of the ORL1 Antagonist Ac-Arg-d-Cha-Qaa-d-Arg-d-p-ClPhe-NH2 von Van Cauwenberghe, Sylvia, Simonin, Frédéric, Cluzeau, Jérôme, Becker, Jérôme A. J, Lubell, William. D, Tourwé, Dirk

Volltext

Synthesis of optically pure N-Boc-protected (2 R,3 R)- and (2 R,3 S)-3-fluoroprolines von Demange, Luc, Cluzeau, Jérôme, Ménez, André, Dugave, Christophe

Volltext

A Highly Productive, Whole-Cell DERA Chemoenzymatic Process for Production of Key Lactonized Side-Chain Intermediates in Statin Synthesis. e62250 von Oslaj, Matej, Cluzeau, Jerome, Orkic, Damir, Kopitar, Gregor, Mrak, Peter, Casar, Zdenko

Volltext

PROCESSES FOR THE PREPARATION OF BETA-AMINOSULFONE COMPOUNDS von STAVBER, Gaj, CLUZEAU, Jerome

Volltext bestellen

Processes for the preparation of beta-aminosulfone compounds von Cluzeau, Jerome, Stavber, Gaj

Volltext bestellen

Processes For The Preparation Of Beta-Aminosulfone Compounds von Cluzeau Jerome, Stavber Gaj

Volltext bestellen