Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 von Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd

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Discovery of Vilaprisan (BAY 1002670): A Highly Potent and Selective Progesterone Receptor Modulator Optimized for Gynecologic Therapies von Möller, Carsten, Bone, Wilhelm, Cleve, Arwed, Klar, Ulrich, Rotgeri, Andrea, Rottmann, Antje, Schultze‐Mosgau, Marcus‐Hillert, Wagenfeld, Andrea, Schwede, Wolfgang

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BAY 1024767 blocks androgen receptor mutants found in castration-resistant prostate cancer patients von Sugawara, Tatsuo, Lejeune, Pascale, Köhr, Silke, Neuhaus, Roland, Faus, Hortensia, Gelato, Kathy A, Busemann, Matthias, Cleve, Arwed, Lücking, Ulrich, von Nussbaum, Franz, Brands, Michael, Mumberg, Dominik, Jung, Klaus, Stephan, Carsten, Haendler, Bernard

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Recent developments in antiandrogens and selective androgen receptor modulators von Haendler, Bernard, Cleve, Arwed

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Synthesis and Biological Activity of a Novel, Highly Potent Progesterone Receptor Antagonist von Fuhrmann, Ulrike, Hess-Stumpp, Holger, Cleve, Arwed, Neef, Günter, Schwede, Wolfgang, Hoffmann, Jens, Fritzemeier, Karl-Heinrich, Chwalisz, Kristof

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Inhibition of BUB1 Kinase by BAY 1816032 Sensitizes Tumor Cells toward Taxanes, ATR, and PARP Inhibitors In Vitro and In Vivo von Siemeister, Gerhard, Mengel, Anne, Fernández-Montalván, Amaury E, Bone, Wilhelm, Schröder, Jens, Zitzmann-Kolbe, Sabine, Briem, Hans, Prechtl, Stefan, Holton, Simon J, Mönning, Ursula, von Ahsen, Oliver, Johanssen, Sandra, Cleve, Arwed, Pütter, Vera, Hitchcock, Marion, von Nussbaum, Franz, Brands, Michael, Ziegelbauer, Karl, Mumberg, Dominik

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Front Cover: Discovery of Vilaprisan (BAY 1002670): A Highly Potent and Selective Progesterone Receptor Modulator Optimized for Gynecologic Therapies (ChemMedChem 21/2018) von Möller, Carsten, Bone, Wilhelm, Cleve, Arwed, Klar, Ulrich, Rotgeri, Andrea, Rottmann, Antje, Schultze‐Mosgau, Marcus‐Hillert, Wagenfeld, Andrea, Schwede, Wolfgang

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Abstract 4333: Identification and optimization of the first highly selective GLUT-1 inhibitors von Bauser, Marcus, Buchmann, Bernd, Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Mueller, Thomas, Kopitz, Charlotte Christine

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Abstract 287: BAY 1816032, a novel BUB1 kinase inhibitor with potent antitumor activity von Siemeister, Gerhard, Mengel, Anne, Bone, Wilhelm, Schröder, Jens, Zitzmann-Kolbe, Sabine, Briem, Hans, Fernández-Montalván, Amaury E., Holton, Simon, Mönning, Ursula, Ahsen, Oliver von, Johanssen, Sandra, Cleve, Arwed, Hitchcock, Marion, Meyer, Kirstin, Nussbaum, Franz von, Brands, Michael, Mumberg, Dominik, Ziegelbauer, Karl

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Cover Picture: Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 (ChemMedChem 20/2016) von Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd

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Abstract 1321: Castration-resistant prostate cancer: BAY 1024767 blocks function of mutated androgen receptor von Haendler, Bernard, Sugawara, Tatsuo, Lejeune, Pascale, Koehr, Silke, Faus, Hortensia, Busemann, Matthias, Cleve, Arwed, Luecking, Ulrich, von Nussbaum, Franz, Brands, Michael, Mumberg, Dominik

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방향족 술폰아미드 유도체 von HARDAKER ELIZABETH, HERBERT SIMON ANTHONY, CLEVE ARWED, WERNER STEFAN, LISHCHYNSKYI ANTON, MESCH STEFANIE, KOCH MARKUS, OSMERS MAREN, BRAEUER NICO, DAHLLOEF HENRIK

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New Roles for LTA4 Hydrolase, LTB4 and BLT1 in Multiple Sclerosis and Experimental Allergic Encephalomyelitis (48.9) von Parkinson, John F, Guilford, William J, Mendoza, Lisa M, Rosser, Mary, Post, Joseph, Schaefer, Caralee, Halks-Miller, Meredith, Kirkland, Tom, Cleve, Arwed, Lassmann, Hans, Reder, Anthony T

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Bub1 Benzyl substituted indazoles as BUB1 inhibitors von MOEWES MANFRED, HITCHCOCK MARION, SIEMEISTER GERHARD, SCHROEDER JENS, BAERFACKER LARS, FERNANDEZ MONTALVAN AMAURY ERNESTO, MUELLER THOMAS, KUHNKE JOACHIM, HOLTON SIMON, BONE WILHELM, CLEVE ARWED, LERCHEN HANS GEORG, BRIEM HANS, MOENNING URSULA, MENGEL ANNE

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BICYCLO 2,3-BENZODIAZEPINES AND SPIROCYCLICALLY SUBSTITUTED 2,3-BENZODIAZEPINES von KUHNKE JOACHIM, BAEURLE STEFAN, LEJEUNE PASCALE, CLEVE ARWED, FERNANDEZ MONTALVAN AMAURY ERNESTO, SIEGEL STEPHAN, HAENDLER BERNARD, KRAUSE SABINE, BUSEMANN MATTHIAS, MOENNING URSULA

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Beneficial effects of fluorine in the anti-progestin ZK 230211 von Cleve, Arwed, Klar, Ulrich, Schwede, Wolfgang

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SUSTITUTED (HETEROARYLMETHYL) THIOHYDANTOINS AS ANTICANCER DRUGS von KOEHR SILKE, CLEVE ARWED, IRLBACHER HORST, HAENDLER BERNARD, LUECKING ULRICH, FAUS GIMENEZ HORTENSIA

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AROMATIC SULFONAMIDE DERIVATIVES AS ANTAGONISTS OR NEGATIVE ALLOSTERIC MODULATORS OF P2X4 RECEPTOR von WERNER, Stefan, CLEVE, Arwed

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PROGESTERONE RECEPTOR ANTAGONISTS von PRUEHS STEFAN, MOELLER CARSTEN, GARKE GUNNAR, PETROV ORLIN, ROTTMANN ANTJE, CLEVE ARWED, SCHMIDT ANJA, HASSELMANN RAINER, FUHRMANN ULRIKE, SCHULTZE MOSGAU MARCUS, BRUDNY KLOEPPEL MARGARETE

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An Efficient Synthesis of 11β-(4-Aminophenyl)spiro[estr-4-ene-17β,2′(5′ H)-furan]-3,5′-dione von Geisler, Jens, Cleve, Arwed, Harre, Michael

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