Enantioselective Organocatalytic Construction of Pyrroloindolines by a Cascade Addition-Cyclization Strategy: Synthesis of (-)-Flustramine B von Austin, Joel F., Kim, Sung-Gon, Sinz, Christopher J., Xiao, Wen-Jing, David W. C. Mac Millan, Halpern, Jack

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Design, Synthesis, and Evaluation of Novel and Selective G‑protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists von Cox, Jason M, Chu, Hong D, Chelliah, Mariappan V, Debenham, John S, Eagen, Keith, Lan, Ping, Lombardo, Matthew, London, Clare, Plotkin, Michael A, Shah, Unmesh, Sun, Zhongxiang, Vaccaro, Henry M, Venkatraman, Srikanth, Suzuki, Takao, Wang, Nengxue, Ashley, Eric R, Crespo, Alejandro, Madeira, Maria, Leung, Dennis H, Alleyne, Candice, Ogawa, Aimie M, Souza, Sarah, Thomas-Fowlkes, Brande, Di Salvo, Jerry, Weinglass, Adam, Kirkland, Melissa, Pachanski, Michele, Powles, Mary Ann, Tozzo, Effie, Akiyama, Taro E, Ujjainwalla, Feroze, Tata, James R, Sinz, Christopher J

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Selective N7 Alkylation of 7-Azaindazoles von Lei, Zhiyu, Bao, Jianming, Cheng, Chen, Yu, Wensheng, Hu, Bin, Jin, Weichen, Jabri, Salman, Yang, Song, Zhao, Lianyun, Sinz, Christopher J, Duffy, Joseph L

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Seven transmembrane G protein-coupled receptor repertoire of gastric ghrelin cells von Engelstoft, Maja S, Park, Won-mee, Sakata, Ichiro, Kristensen, Line V, Husted, Anna Sofie, Osborne-Lawrence, Sherri, Piper, Paul K, Walker, Angela K, Pedersen, Maria H, Nøhr, Mark K, Pan, Jie, Sinz, Christopher J, Carrington, Paul E, Akiyama, Taro E, Jones, Robert M, Tang, Cong, Ahmed, Kashan, Offermanns, Stefan, Egerod, Kristoffer L, Zigman, Jeffrey M, Schwartz, Thue W

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Total synthesis of diazonamide A von Knowles, Robert R, Carpenter, Joseph, Blakey, Simon B, Kayano, Akio, Mangion, Ian K, Sinz, Christopher J, Macmillan, David W C

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The Direct and Enantioselective Organocatalytic α-Oxidation of Aldehydes von Brown, Sean P, Brochu, Michael P, Sinz, Christopher J, MacMillan, David W. C

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Modeling a Crowdsourced Definition of Molecular Complexity von Sheridan, Robert P, Zorn, Nicolas, Sherer, Edward C, Campeau, Louis-Charles, Chang, Charlie (Zhenyu), Cumming, Jared, Maddess, Matthew L, Nantermet, Philippe G, Sinz, Christopher J, O’Shea, Paul D

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Total synthesis of the polyene macrolide dermostatin A von Sinz, Christopher J, Rychnovsky, Scott D

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Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects von Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Discovery of Orally Bioavailable and Liver-Targeted Hypoxia-Inducible Factor Prolyl Hydroxylase (HIF-PHD) Inhibitors for the Treatment of Anemia von Liu, Ping, Wang, Liping, DuBois, Byron G, Colandrea, Vincent J, Liu, Rongqiang, Cai, Jiaqiang, Du, Xiaoxing, Quan, Weiguo, Morris, William, Bai, Jianwu, Bishwokarma, Bimjhana, Cheng, Mangeng, Piesvaux, Jennifer, Ray, Kallol, Alpert, Carla, Chiu, Chi-Sung, Zielstorff, Mark, Metzger, Joseph M, Yang, Liming, Leung, Dennis, Alleyne, Candice, Vincent, Stella H, Pucci, Vincenzo, Li, Xiaofang, Crespo, Alejandro, Stickens, Dominique, Hale, Jeffrey J, Ujjainwalla, Feroze, Sinz, Christopher J

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Small molecule activation of lecithin cholesterol acyltransferase modulates lipoprotein metabolism in mice and hamsters von Chen, Zhu, Wang, Sheng-ping, Krsmanovic, Mihajlo L, Castro-Perez, Jose, Gagen, Karen, Mendoza, Vivienne, Rosa, Ray, Shah, Vinit, He, Timothy, Stout, Steve J, Geoghagen, Neil S, Lee, Sang H, McLaren, David G, Wang, Liangsu, Roddy, Thomas P, Plump, Andrew S, Hubbard, Brian K, Sinz, Christopher J, Johns, Douglas G

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Corrigendum to “Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects” [Bioorg. Med. Chem. Lett. 26 (2016) 5724–5728]... von Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Discovery and Optimization of a Novel Triazole Series of GPR142 Agonists for the Treatment of Type 2 Diabetes von Guo, Liangqin, Parker, Dann L, Zang, Yi, Sweis, Ramzi F, Liu, Weiguo, Sherer, Edward C, Buist, Nicole, Terebetski, Jenna, Kelly, Terri, Bugianesi, Randal, Priest, Birgit T, Dingley, Karen H, Li, Xiaofang, Mitelman, Stan, Salituro, Gino, Trujillo, Maria E, Pachanski, Michele, Kirkland, Melissa, Powles, Mary Ann, Eiermann, George J, Feng, Yue, Shang, Jin, Howard, Andrew D, Ujjainwalla, Feroze, Sinz, Christopher J, Debenham, John S, Edmondson, Scott D, Nargund, Ravi P, Hagmann, William K, Li, Derun

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Total Synthesis of Dermostatin A von Sinz, Christopher J., Rychnovsky, Scott D.

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Total synthesis of diazonamide AElectronic supplementary information (ESI) available: Experimental procedures, structural proofs, and spectral data for all new compounds are provid... von Knowles, Robert R, Carpenter, Joseph, Blakey, Simon B, Kayano, Akio, Mangion, Ian K, Sinz, Christopher J, MacMillan, David W. C

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Abstract 17305: Activation of Soluble Guanylate Cyclase Ameliorates the Progression of Glucose Intolerance and Nephropathy in Obese ZSF1 Rats von da Cunha, Valdeci, Shah, Kashmira, Price, Olga, Sinz, Christopher J, Kim, Ronald M

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Diastereoselective synthesis of polypropionates: Cationic couplings of 4-acetoxy-1,3-dioxanes with crotyl-metal reagents von Rychnovsky, Scott D., Sinz, Christopher J.

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PLASMA KALLIKREIN INHIBITORS von CERNAKA, Natalija, LOPEZ, Jovan, Alexander, TIAN, Maoqun, MERCHANT, Rohan, Rajiv, SINZ, Christopher, J, OGAWA, Anthony, K, GAO, Ying-Duo, BAO, Jianming, TANG, Haiqun, MANDAL, Mihir, B, XIAO, Dong, CHENG, Alan, C, YANG, Song, SHARP, Phillip, Patrick, HE, Jiafang

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PLASMA KALLIKREIN INHIBITORS von CERNAKA, Natalija, JABRI, Salman, TIAN, Maoqun, OGAWA, Anthony Ken, OSLER, Skylar, K, SINZ, Christopher, J, GAO, Ying-Duo, SHARP, Phillip Patrick, BAO, Jianming, TANG, Haiqun, LOPEZ, Jovan Alexander, XIAO, Dong, CHENG, Alan, C, YANG, Song, MERCHANT, Rohan

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PLASMA KALLIKREIN INHIBITORS von TIAN, Maoqun, HICKS, Jacqueline, D, ZHAO, Zhiqiang, SINZ, Christopher, J, SHARP, Phillip Patrick, SHEARN-NANCE, Galen Paul, LOMBARDO, Matthew, J, BAO, Jianming, KUANG, Rongze, LOPEZ, Jovan Alexander, CHENG, Alan, C, YANG, Song, WU, Zhicai, MERCHANT, Rohan

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