N -Acetyl-3-aminopyrazoles block the non-canonical NF-kB cascade by selectively inhibiting NIK von Pippione, Agnese C, Sainas, Stefano, Federico, Antonella, Lupino, Elisa, Piccinini, Marco, Kubbutat, Michael, Contreras, Jean-Marie, Morice, Christophe, Barge, Alessandro, Ducime, Alex, Boschi, Donatella, Al-Karadaghi, Salam, Lolli, Marco L

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Moderately lipophilic 2-(Het)aryl-6-dithioacetals, 2-phenyl-1,4-benzodioxane-6-dithioacetals and 2-phenylbenzofuran-5-dithioacetals: Synthesis and primary evaluation as potential a... von Lepechkin-Zilbermintz, Veronica, Bareket, Daniel, Gonnord, Virginie, Steffen, Alexandre, Morice, Christophe, Michaut, Mathieu, Munder, Anna, Korshin, Edward E., Contreras, Jean-Marie, Cerasi, Erol, Sasson, Shlomo, Gruzman, Arie

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Discovery, Structure–Activity Relationship, and Antiparkinsonian Effect of a Potent and Brain-Penetrant Chemical Series of Positive Allosteric Modulators of Metabotropic Glutamate... von Charvin, Delphine, Pomel, Vincent, Ortiz, Millan, Frauli, Mélanie, Scheffler, Sophie, Steinberg, Edith, Baron, Luc, Deshons, Laurène, Rudigier, Rachel, Thiarc, Delphine, Morice, Christophe, Manteau, Baptiste, Mayer, Stanislas, Graham, Danielle, Giethlen, Bruno, Brugger, Nadia, Hédou, Gaël, Conquet, François, Schann, Stephan

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Chryso-lactams:Gold(I) derivatives of ampicillin with specific activity against Gram-positive pathogens von Michaut, Mathieu, Steffen, Alexandre, Contreras, Jean-Marie, Morice, Christophe, Paulen, Aurélie, Schalk, Isabelle J., Plésiat, Patrick, Mislin, Gaëtan L.A.

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1,2,3-Triazole-gold(I)-triethylposphine derivatives active against resistant Gram-positive pathogens von Michaut, Mathieu, Steffen, Alexandre, Contreras, Jean-Marie, Morice, Christophe, Schalk, Isabelle J., Plésiat, Patrick, Mislin, Gaëtan L.A.

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Toward the identification of viral cap-methyltransferase inhibitors by fluorescence screening assay von Aouadi, Wahiba, Eydoux, Cécilia, Coutard, Bruno, Martin, Baptiste, Debart, Françoise, Vasseur, Jean Jacques, Contreras, Jean Marie, Morice, Christophe, Quérat, Gilles, Jung, Marie-Louise, Canard, Bruno, Guillemot, Jean-Claude, Decroly, Etienne

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Approved drugs screening against the nsP1 capping enzyme of Venezuelan equine encephalitis virus using an immuno-based assay von Ferreira-Ramos, Ana S., Li, Changqing, Eydoux, Cécilia, Contreras, Jean Marie, Morice, Christophe, Quérat, Gilles, Gigante, Alba, Pérez Pérez, María-Jesús, Jung, Marie-Louise, Canard, Bruno, Guillemot, Jean-Claude, Decroly, Etienne, Coutard, Bruno

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Discovery of BNC375, a Potent, Selective, and Orally Available Type I Positive Allosteric Modulator of α7 nAChRs von Harvey, Andrew J, Avery, Thomas D, Schaeffer, Laurent, Joseph, Christophe, Huff, Belinda C, Singh, Rajinder, Morice, Christophe, Giethlen, Bruno, Grishin, Anton A, Coles, Carolyn J, Kolesik, Peter, Wagner, Stéphanie, Andriambeloson, Emile, Huyard, Bertrand, Poiraud, Etienne, Paul, Dharam, O’Connor, Susan M

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Porphyrin Derivatives Inhibit the Interaction between Receptor Activator of NF-[kappa]B and Its Ligand von Chypre, Mélanie, Madel, Maria-Bernadette, Chaloin, Olivier, Blin-Wakkach, Claudine, Morice, Christophe, Mueller, Christopher G

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4-Hydroxy- N -[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide: a novel inhibitor of the canonical NF-κB cascade von Pippione, Agnese C, Federico, Antonella, Ducime, Alex, Sainas, Stefano, Boschi, Donatella, Barge, Alessandro, Lupino, Elisa, Piccinini, Marco, Kubbutat, Michael, Contreras, Jean-Marie, Morice, Christophe, Al-Karadaghi, Salam, Lolli, Marco L

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Porphyrin Derivatives Inhibit the Interaction between Receptor Activator of NF‐κB and Its Ligand von Chypre, Mélanie, Madel, Maria‐Bernadette, Chaloin, Olivier, Blin‐Wakkach, Claudine, Morice, Christophe, Mueller, Christopher G.

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N-Acetyl-3-aminopyrazoles block the non-canonical NF-kB cascade by selectively inhibiting NIKElectronic supplementary information (ESI) available: Additional biochemical data, chem... von Pippione, Agnese C, Sainas, Stefano, Federico, Antonella, Lupino, Elisa, Piccinini, Marco, Kubbutat, Michael, Contreras, Jean-Marie, Morice, Christophe, Barge, Alessandro, Ducime, Alex, Boschi, Donatella, Al-Karadaghi, Salam, Lolli, Marco L

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Fragment pharmacophore-based screening: a powerful approach for efficient lead discovery von Deyon-Jung, Laurence, Morice, Christophe, Chéry, Florence, Gay, Julie, Langer, Thierry, Frantz, Marie-Céline, Rozot, Roger, Dalko-Csiba, Maria

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Fragment pharmacophore-based in silicoscreening: a powerful approach for efficient lead discovery von Deyon-Jung, Laurence, Morice, Christophe, Chery, Florence, Gay, Julie, Langer, Thierry, Frantz, Marie-Celine, Rozot, Roger, Dalko-Csiba, Maria

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Fragment pharmacophore-based in silico screening: a powerful approach for efficient lead discovery von Deyon-Jung, Laurence, Morice, Christophe, Chéry, Florence, Gay, Julie, Langer, Thierry, Frantz, Marie-Céline, Rozot, Roger, Dalko-Csiba, Maria

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4-Hydroxy-N-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide: a novel inhibitor of the canonical NF-κB cascadeElectronic supplementary information (ESI) available:... von Pippione, Agnese C, Federico, Antonella, Ducime, Alex, Sainas, Stefano, Boschi, Donatella, Barge, Alessandro, Lupino, Elisa, Piccinini, Marco, Kubbutat, Michael, Contreras, Jean-Marie, Morice, Christophe, Al-Karadaghi, Salam, Lolli, Marco L

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DIHYDRO[1,8]NAPHTHYRIDIN-7-ONE AND PYRIDO[3,2-B][1,4]OXAZIN-3-ONE FOR USE IN TREATING CANCER, AND METASTASES IN PARTICULAR von MORICE, Christophe, RIGUET, Eric

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DIHYDRO[1,8]NAPHTHYRIDIN-7-ONE AND PYRIDO[3,2-B][1,4]OXAZIN-3-ONE FOR USE IN TREATING CANCER, AND METASTASES IN PARTICULAR von MORICE, Christophe, RIGUET, Eric

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Structural, Magnetic, and Dynamic Characterization of the (d xz ,d y z )4(d x y )1 Ground-State Low-Spin Iron(III) Tetraphenylporphyrinate Complex [(p-TTP)Fe(2,6-XylylNC)2]CF3SO3 von Simonneaux, Gérard, Schünemann, Volker, Morice, Christophe, Carel, Laurence, Toupet, Loïc, Winkler, Heiner, Trautwein, Alfred X, Walker, F. Ann

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Palladium Assisted Substitution of 3-Benzo[b]furan Triflates von Morice, Christophe, Garrido, Fabrice, Mann, André, Suffert, Jean

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