The preclinical efficacy of the novel hypomethylating agent NTX-301 as a monotherapy and in combination with venetoclax in acute myeloid leukemia von Lim, Byungho, Yoo, Dabin, Chun, Younghwa, Go, Areum, Cho, Kyung-Jin, Choi, Daeun, Jung, Myoung Eun, Lee, Ha Young, Boohaker, Rebecca J., Lee, Jin Soo, Jung, DooYoung, Choi, Gildon

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Discovery of TRD‐93 as a novel DRAK2 inhibitor von Park, Sangjun, Kye, Seungmin, Jung, Myoung Eun, Chae, Chong Hak, Yang, Kyung‐Min, Kim, Seong‐Jin, Choi, Gildon, Lee, Kwangho

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Identification of TRD‐35 as Potent and Selective DRAK2 Inhibitor von Ali, Imran, Park, Sangjun, Jung, Myoung Eun, Lee, Nari, Bibi, Maimoona, Chae, Chong Hak, Yang, Kyung‐Min, Kim, Seong‐Jin, Choi, Gildon, Lee, Kwangho

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A bi-ligand co-functionalized gold nanoparticles-based calcium ion probe and its application to the detection of calcium ions in serum von Eom, Min Sik, Jang, Woojeong, Lee, Yoon Seo, Choi, Gildon, Kwon, Yong-Uk, Han, Min Su

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Identification of a New Morpholine Scaffold as a P2Y12 Receptor Antagonist von Ahn, Young Ha, Lee, Joo-Youn, Park, Hee Dong, Kim, Tae Hun, Park, Min Chul, Choi, Gildon, Kim, Sunghoon

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A guide for bioinformaticians: ‘omics-based drug discovery for precision oncology von Mun, Jihyeob, Choi, Gildon, Lim, Byungho

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Further optimization of novel pyrrole 3-carboxamides for targeting serotonin 5-HT2A, 5-HT2C, and the serotonin transporter as a potential antidepressant von SUK YOUN KANG, PARK, Eun-Jung, LEE, Jinhwa, PARK, Woo-Kyu, HYUN JUNG KIM, GILDON CHOI, MYUNG EUN JUNG, HEE JEONG SEO, MIN JU KIM, AE NIM PAE, KIM, Jeongmin

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Discovery of novel [1,2,4]triazolo[4,3-a]quinoxaline aminophenyl derivatives as BET inhibitors for cancer treatment von Ali, Imran, Lee, Jooyun, Go, Areum, Choi, Gildon, Lee, Kwangho

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Novel allosteric glutaminase 1 inhibitors with macrocyclic structure activity relationship analysis von Lee, Eun Ji, Duggirala, Krishna Babu, Lee, Yujin, Yun, Mi Ran, Jang, Jiyoon, Cyriac, Rajath, Jung, Myoung Eun, Choi, Gildon, Chae, Chong Hak, Cho, Byoung Chul, Lee, Kwangho

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Generation of human tonsil epithelial organoids as an ex vivo model for SARS-CoV-2 infection von Kim, Han Kyung, Kim, Hyeryeon, Lee, Myoung Kyu, Choi, Woo Hee, Jang, Yejin, Shin, Jin Soo, Park, Jun-Yeol, Bae, Dong Hyuck, Hyun, Seong-In, Kim, Kang Hyun, Han, Hyun Wook, Lim, Byungho, Choi, Gildon, Kim, Meehyein, Chang Lim, Young, Yoo, Jongman

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A Study on Preclinical Efficacy, Underlying Mechanisms, and Sensitivity Markers of a Novel Hypomethylating Agent Ntx-301 in Acute Myeloid Leukemia von Lim, Byungho, Yoo, Dabin, Cho, Kyung-jin, Choi, Daeun, Jung, Myoung Eun, Jung, Doo Young, Lee, Jin Soo, Chun, Younghwa, Go, Areum, Lee, Ha Young, Choi, Gildon

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Radicicol Inhibits Chikungunya Virus Replication by Targeting Nonstructural Protein 2 von Nam, Sangwoo, Ga, Yun Ji, Lee, Joo-Youn, Hwang, Woo-Yeon, Jung, Eunhye, Shin, Jin Soo, Chen, Weiyi, Choi, Gildon, Zhou, Bin, Yeh, Jung-Yong, Go, Yun Young

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DW71177: A novel [1,2,4]triazolo[4,3-a]quinoxaline-based potent and BD1-Selective BET inhibitor for the treatment of acute myeloid leukemia von Ali, Imran, Cha, Hyung Jin, Lim, Byungho, Chae, Chong Hak, Youm, Jihyun, Park, Whui Jung, Lee, Sang Ho, Kim, Jung Hwan, Jeong, Docgyun, Lim, Jae Kyung, Hwang, Yun-Ha, Roe, Jae-Seok, Woo, Jae-Sung, Lee, Kwangho, Choi, Gildon

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Novel allosteric glutaminase inhibitors with macrocyclic structure activity relationship analysis (part 2) von Lee, Eun Ji, Jang, Jiyoon, Cyriac, Rajath, Yun, Mi Ran, Kwon, Yeongju, Jung, Myoung Eun, Choi, Gildon, Chae, Chong Hak, Cho, Byoung Chul, Lee, Kwangho

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Synthesis and biological evaluation of (2‐aminosulfonylpyridin‐6‐yl)pyrazolopyrimidinone derivatives as Wee1 inhibitors for cancer treatment von Kim, Yeon Ju, Jung, Myoung Eun, Lee, Ju Yeong, Lee, Yun‐Han, Choi, Gildon, Jeon, Moon‐Kook

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Discovery of indirubin derivatives as new class of DRAK2 inhibitors from high throughput screening von Jung, Myoung Eun, Byun, Byung Jin, Kim, Hye-Mi, Lee, Joo Yun, Park, Jin-Hee, Lee, Nari, Son, You Hwa, Choi, Sang Un, Yang, Kyung-Min, Kim, Seong-Jin, Lee, Kwangho, Kim, Yong-Chul, Choi, Gildon

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Biological evaluation of tanshindiols as EZH2 histone methyltransferase inhibitors von Woo, Jimin, Kim, Hyun-Young, Byun, Byung Jin, Chae, Chong-Hak, Lee, Ji Young, Ryu, Shi Yong, Park, Woo-Kyu, Cho, Heeyeong, Choi, Gildon

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Integrative Analyses Reveal the Anticancer Mechanisms and Sensitivity Markers of the Next-Generation Hypomethylating Agent NTX-301 von Lim, Byungho, Yoo, Dabin, Chun, Younghwa, Go, Areum, Kim, Ji Yeon, Lee, Ha Young, Boohaker, Rebecca J, Cho, Kyung-Jin, Ahn, Sunjoo, Lee, Jin Soo, Jung, DooYoung, Choi, Gildon

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Allosteric Inhibitor TREA‐0236 Containing Non‐hydrolysable Quinazoline‐4‐one for EGFR T790M/C797S Mutants Inhibition von Lee, Seoyoung, Kim, Jiwon, Duggirala, Krishna Babu, Go, Areum, Shin, Inji, Cho, Byoung Chul, Choi, Gildon, Chae, Chong Hak, Lee, Kwangho

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Discovery of a potent small molecule SIRT1/2 inhibitor with anticancer effects von CHOI, GILDON, LEE, JONGKOOK, JI, JEONG YEON, WOO, JIMIN, KANG, NAM SOOK, CHO, SUNG YUN, KIM, HYOUNG RAE, HA, JAE DU, HAN, SUN-YOUNG

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