Decarboxylative borylation von Li, Chao, Wang, Jie, Barton, Lisa M., Yu, Shan, Tian, Maoqun, Peters, David S., Kumar, Manoj, Yu, Antony W., Johnson, Kristen A., Chatterjee, Arnab K., Yan, Ming, Baran, Phil S.

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A high-throughput phenotypic screen identifies clofazimine as a potential treatment for cryptosporidiosis von Love, Melissa S, Beasley, Federico C, Jumani, Rajiv S, Wright, Timothy M, Chatterjee, Arnab K, Huston, Christopher D, Schultz, Peter G, McNamara, Case W

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Antimalarial drug discovery — approaches and progress towards new medicines von Flannery, Erika L., Chatterjee, Arnab K., Winzeler, Elizabeth A.

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Antitumor activity of a systemic STING-activating non-nucleotide cGAMP mimetic von Chin, Emily N., Yu, Chenguang, Vartabedian, Vincent F., Jia, Ying, Kumar, Manoj, Gamo, Ana M., Vernier, William, Ali, Sabrina H., Kissai, Mildred, Lazar, Daniel C., Nhan Nguyen, Pereira, Laura E., Benish, Brent, Woods, Ashley K., Joseph, Sean B., Chu, Alan, Johnson, Kristen A., Sander, Philipp N., Martinez-Pena, Francisco, Hampton, Eric N., Young, Travis S., Wolan, Dennis W., Chatterjee, Arnab K., Schultz, Peter G., Petrassi, H. Michael, Teijaro, John R., Lairson, Luke L.

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Auranofin exerts broad-spectrum bactericidal activities by targeting thiol-redox homeostasis von Harbut, Michael B., Vilchèze, Catherine, Luo, Xiaozhou, Hensler, Mary E., Guo, Hui, Yang, Baiyuan, Chatterjee, Arnab K., Nizet, Victor, Jacobs, William R., Schultz, Peter G., Wang, Feng

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A metabolite-derived protein modification integrates glycolysis with KEAP1–NRF2 signalling von Bollong, Michael J., Lee, Gihoon, Coukos, John S., Yun, Hwayoung, Zambaldo, Claudio, Chang, Jae Won, Chin, Emily N., Ahmad, Insha, Chatterjee, Arnab K., Lairson, Luke L., Schultz, Peter G., Moellering, Raymond E.

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The ReFRAME library as a comprehensive drug repurposing library and its application to the treatment of cryptosporidiosis von Janes, Jeff, Young, Megan E., Chen, Emily, Rogers, Nicole H., Burgstaller-Muehlbacher, Sebastian, Hughes, Laura D., Love, Melissa S., Hull, Mitchell V., Kuhen, Kelli L., Woods, Ashley K., Joseph, Sean B., Petrassi, H. Michael, McNamara, Case W., Tremblay, Matthew S., Su, Andrew I., Schultz, Peter G., Chatterjee, Arnab K.

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Commonly used surfactants sodium dodecyl sulphate, cetylpyridinium chloride and sodium laureth sulphate and their effects on antioxidant defence system and oxidative stress indices... von Bhattacharya, Ritwick, Chatterjee, Arnab, Chatterjee, Soumendranath, Saha, Nimai Chandra

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Drug repurposing screens identify chemical entities for the development of COVID-19 interventions von Bakowski, Malina A., Beutler, Nathan, Wolff, Karen C., Kirkpatrick, Melanie G., Chen, Emily, Nguyen, Tu-Trinh H., Riva, Laura, Shaabani, Namir, Parren, Mara, Ricketts, James, Gupta, Anil K., Pan, Kastin, Kuo, Peiting, Fuller, MacKenzie, Garcia, Elijah, Teijaro, John R., Yang, Linlin, Sahoo, Debashis, Chi, Victor, Huang, Edward, Vargas, Natalia, Roberts, Amanda J., Das, Soumita, Ghosh, Pradipta, Woods, Ashley K., Joseph, Sean B., Hull, Mitchell V., Schultz, Peter G., Burton, Dennis R., Chatterjee, Arnab K., McNamara, Case W., Rogers, Thomas F.

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Multistep Synthesis of Analogues of Remdesivir: Incorporating Heterocycles at the C‑1′ Position von Cardoza, Savio, Shrivash, Manoj Kumar, Riva, Laura, Chatterjee, Arnab K., Mandal, Ajay, Tandon, Vibha

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Drug repurposing screen identifies lonafarnib as respiratory syncytial virus fusion protein inhibitor von Sake, Svenja M., Zhang, Xiaoyu, Rajak, Manoj Kumar, Urbanek-Quaing, Melanie, Carpentier, Arnaud, Gunesch, Antonia P., Grethe, Christina, Matthaei, Alina, Rückert, Jessica, Galloux, Marie, Larcher, Thibaut, Le Goffic, Ronan, Hontonnou, Fortune, Chatterjee, Arnab K., Johnson, Kristen, Morwood, Kaycie, Rox, Katharina, Elgaher, Walid A. M., Huang, Jiabin, Wetzke, Martin, Hansen, Gesine, Fischer, Nicole, Eléouët, Jean-Francois, Rameix-Welti, Marie-Anne, Hirsch, Anna K. H., Herold, Elisabeth, Empting, Martin, Lauber, Chris, Schulz, Thomas F., Krey, Thomas, Haid, Sibylle, Pietschmann, Thomas

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The combined treatment of Molnupiravir and Favipiravir results in a potentiation of antiviral efficacy in a SARS-CoV-2 hamster infection model von Abdelnabi, Rana, Foo, Caroline S., Kaptein, Suzanne J.F., Zhang, Xin, Do, Thuc Nguyen Dan, Langendries, Lana, Vangeel, Laura, Breuer, Judith, Pang, Juanita, Williams, Rachel, Vergote, Valentijn, Heylen, Elisabeth, Leyssen, Pieter, Dallmeier, Kai, Coelmont, Lotte, Chatterjee, Arnab K., Mols, Raf, Augustijns, Patrick, De Jonghe, Steven, Jochmans, Dirk, Weynand, Birgit, Neyts, Johan

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Reprogramming of Protein-Targeted Small-Molecule Medicines to RNA by Ribonuclease Recruitment von Zhang, Peiyuan, Liu, Xiaohui, Abegg, Daniel, Tanaka, Toru, Tong, Yuquan, Benhamou, Raphael I, Baisden, Jared, Crynen, Gogce, Meyer, Samantha M, Cameron, Michael D, Chatterjee, Arnab K, Adibekian, Alexander, Childs-Disney, Jessica L, Disney, Matthew D

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Antiviral drug screen identifies DNA-damage response inhibitor as potent blocker of SARS-CoV-2 replication von Garcia, Gustavo, Sharma, Arun, Ramaiah, Arunachalam, Sen, Chandani, Purkayastha, Arunima, Kohn, Donald B., Parcells, Mark S., Beck, Sebastian, Kim, Heeyoung, Bakowski, Malina A., Kirkpatrick, Melanie G., Riva, Laura, Wolff, Karen C., Han, Brandon, Yuen, Constance, Ulmert, David, Purbey, Prabhat K., Scumpia, Philip, Beutler, Nathan, Rogers, Thomas F., Chatterjee, Arnab K., Gabriel, Gülsah, Bartenschlager, Ralf, Gomperts, Brigitte, Svendsen, Clive N., Betz, Ulrich A.K., Damoiseaux, Robert D., Arumugaswami, Vaithilingaraja

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Scalable Thiol Reactivity Profiling Identifies Azetidinyl Oxadiazoles as Cysteine-Targeting Electrophiles von Ghorbani, Fereshte, You, Shaochen, Grabovyi, Gennadii A., Hong, Mannkyu, Lindsey, Garrett, Chatterjee, Arnab K., Bollong, Michael J.

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Allosteric nanobodies reveal the dynamic range and diverse mechanisms of G-protein-coupled receptor activation von Staus, Dean P., Strachan, Ryan T., Manglik, Aashish, Pani, Biswaranjan, Kahsai, Alem W., Kim, Tae Hun, Wingler, Laura M., Ahn, Seungkirl, Chatterjee, Arnab, Masoudi, Ali, Kruse, Andrew C., Pardon, Els, Steyaert, Jan, Weis, William I., Prosser, R. Scott, Kobilka, Brian K., Costa, Tommaso, Lefkowitz, Robert J.

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Neratinib protects pancreatic beta cells in diabetes von Ardestani, Amin, Li, Sijia, Annamalai, Karthika, Lupse, Blaz, Geravandi, Shirin, Dobrowolski, Aleksandra, Yu, Shan, Zhu, Siying, Baguley, Tyler D., Surakattula, Murali, Oetjen, Janina, Hauberg-Lotte, Lena, Herranz, Raquel, Awal, Sushil, Altenhofen, Delsi, Nguyen-Tran, Van, Joseph, Sean, Schultz, Peter G., Chatterjee, Arnab K., Rogers, Nikki, Tremblay, Matthew S., Shen, Weijun, Maedler, Kathrin

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2‑Sulfonylpyridines as Tunable, Cysteine-Reactive Electrophiles von Zambaldo, Claudio, Vinogradova, Ekaterina V, Qi, Xiaotian, Iaconelli, Jonathan, Suciu, Radu M, Koh, Minseob, Senkane, Kristine, Chadwick, Stormi R, Sanchez, Brittany B, Chen, Jason S, Chatterjee, Arnab K, Liu, Peng, Schultz, Peter G, Cravatt, Benjamin F, Bollong, Michael J

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Identification of a small molecule with activity against drug-resistant and persistent tuberculosis von Wang, Feng, Sambandan, Dhinakaran, Halder, Rajkumar, Wang, Jianing, Batt, Sarah M, Weinrick, Brian, Ahmad, Insha, Yang, Pengyu, Zhang, Yong, Kim, John, Hassani, Morad, Huszar, Stanislav, Trefzer, Claudia, Ma, Zhenkun, Kaneko, Takushi, Mdluli, Khisi E, Franzblau, Scott, Chatterjee, Arnab K, Johnsson, Kai, Johnson, Kai, Mikusova, Katarina, Besra, Gurdyal S, Fütterer, Klaus, Robbins, Scott H, Barnes, S Whitney, Walker, John R, Jacobs, Jr, William R, Schultz, Peter G

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Cell-based medicinal chemistry optimization of high-throughput screening (HTS) hits for orally active antimalarials. Part 1: challenges in potency and absorption, distribution, met... von Chatterjee, Arnab K

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