Quinoline 3-sulfonamides inhibit lactate dehydrogenase A and reverse aerobic glycolysis in cancer cells von Billiard, Julia, Dennison, Jennifer B, Briand, Jacques, Annan, Roland S, Chai, Deping, Colón, Mariela, Dodson, Christopher S, Gilbert, Seth A, Greshock, Joel, Jing, Junping, Lu, Hong, McSurdy-Freed, Jeanelle E, Orband-Miller, Lisa A, Mills, Gordon B, Quinn, Chad J, Schneck, Jessica L, Scott, Gilbert F, Shaw, Anthony N, Waitt, Gregory M, Wooster, Richard F, Duffy, Kevin J

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An efficient, asymmetric solid-phase synthesis of benzothiadiazine-substituted tetramic acids: Potent inhibitors of the hepatitis C virus RNA-dependent RNA polymerase von Evans, Karen A., Chai, Deping, Graybill, Todd L., Burton, George, Sarisky, Robert T., Lin-Goerke, Juili, Johnston, Victor K., Rivero, Ralph A.

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Synthesis of (25 R)-26-hydroxycholesterol von Williams, John R, Chai, Deping, Wright, Dominic

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3-(1,1-Dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones, Potent Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase von Tedesco, Rosanna, Shaw, Antony N, Bambal, Ramesh, Chai, Deping, Concha, Nestor O, Darcy, Michael G, Dhanak, Dashyant, Fitch, Duke M, Gates, Adam, Gerhardt, Warren G, Halegoua, Dina L, Han, Chao, Hofmann, Glenn A, Johnston, Victor K, Kaura, Arun C, Liu, Nannan, Keenan, Richard M, Lin-Goerke, Juili, Sarisky, Robert T, Wiggall, Kenneth J, Zimmerman, Michael N, Duffy, Kevin J

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Substituted benzothiadizine inhibitors of Hepatitis C virus polymerase von Shaw, Antony N., Tedesco, Rosanna, Bambal, Ramesh, Chai, Deping, Concha, Nestor O., Darcy, Michael G., Dhanak, Dashyant, Duffy, Kevin J., Fitch, Duke M., Gates, Adam, Johnston, Victor K., Keenan, Richard M., Lin-Goerke, Juili, Liu, Nannan, Sarisky, Robert T., Wiggall, Kenneth J., Zimmerman, Michael N.

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Abstract 5418: Rapid LDH5 inhibition reverses malignant metabolic phenotype and impairs survival of hepatocellular carcinoma cells von Billiard, Julia, Annan, Roland, Ariazi, Jennifer, Briand, Jacques, Brown, Kristin, Campobasso, Nino, Chakravorty, Subhas, Chai, Deping, Colón, Mariela, Davenport, Elizabeth, Dodson, Christopher, Gaul, Nathan, Gilbert, Seth, Jurewicz, Anthony, Lu, Hong, McNulty, Dean, McSurdy-Freed, Jeanelle, Miller, Lisa, Nurse, Kelvin, Rao Nuthulaganti, Paru, Quinn, Chad, Schneck, Jessica, Scott, Gilbert, Shaw, Tony, Sherk, Christian, Smallwood, Angela, Sweitzer, Sharon, Villa, James, Waitt, Gregory, Wooster, Richard, Duffy, Kevin

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A Highly Efficient, Asymmetric Synthesis of Benzothiadiazine-Substituted Tetramic Acids:  Potent Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase von Fitch, Duke M, Evans, Karen A, Chai, Deping, Duffy, Kevin J

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Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzothiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitors von Tedesco, Rosanna, Chai, Deping, Darcy, Michael G., Dhanak, Dashyant, Fitch, Duke M., Gates, Adam, Johnston, Victor K., Keenan, Richard M., Lin-Goerke, Juili, Sarisky, Robert T., Shaw, Antony N., Valko, Klara L., Wiggall, Kenneth J., Zimmerman, Michael N., Duffy, Kevin J.

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Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295 von Qian, Xiangping, McDonald, Andrew, Zhou, Han-Jie, Adams, Nicholas D, Parrish, Cynthia A, Duffy, Kevin J, Fitch, Duke M, Tedesco, Rosanna, Ashcraft, Luke W, Yao, Bing, Jiang, Hong, Huang, Jennifer K, Marin, Melchor V, Aroyan, Carrie E, Wang, Jianchao, Ahmed, Seyed, Burgess, Joelle L, Chaudhari, Amita M, Donatelli, Carla A, Darcy, Michael G, Ridgers, Lance H, Newlander, Ken A, Schmidt, Stanley J, Chai, Deping, Colón, Mariela, Zimmerman, Michael N, Lad, Latesh, Sakowicz, Roman, Schauer, Stephen, Belmont, Lisa, Baliga, Ramesh, Pierce, Daniel W, Finer, Jeffrey T, Wang, Zhengping, Morgan, Bradley P, Morgans, David J, Auger, Kurt R, Sung, Chiu-Mei, Carson, Jeff D, Luo, Lusong, Hugger, Erin D, Copeland, Robert A, Sutton, David, Elliott, John D, Jackson, Jeffrey R, Wood, Kenneth W, Dhanak, Dashyant, Bergnes, Gustave, Knight, Steven D

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Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzo-thiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitor... von TEDESCO, Rosanna, DEPING CHAI, SHAW, Antony N, VALKO, Klara L, WIGGALL, Kenneth J, ZIMMERMAN, Michael N, DUFFY, Kevin J, DARCY, Michael G, DHANAK, Dashyant, FITCH, Duke M, GATES, Adam, JOHNSTON, Victor K, KEENAN, Richard M, LIN-GOERKE, Juili, SARISKY, Robert T

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Synthesis of the aglycone of 26- O-deacetyl pavoninin-5 von Williams, John R, Chai, Deping, Bloxton, James D, Gong, Hua, Solvibile, William R

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Studies toward the synthesis of the shark repellent pavoninin‐5 von Williams, John R., Chai, Deping, Gong, Hua, Zhao, Wei, Wright, Dominic

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PROLYL HYDROXYLASE INHIBITORS von CHAI, DEPING

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PROLYL HYDROXYLASE INHIBITORS von FITCH, DUKE, M, CHAI, DEPING

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PROLYL HYDROXYLASE INHIBITORS von CHAI DEPING, FITCH DUKE M

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PROLYL HYDROXYLASE INHIBITORS von FITCH, DUKE, M, CHAI, DEPING

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PROLYL HYDROXYLASE INHIBITORS von FITCH, DUKE, M, CHAI, DEPING

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PROLYL HYDROXYLASE INHIBITORS von FITCH, DUKE, M, CHAI, DEPING

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PROLYL HYDROXYLASE INHIBITORS von CHAI DEPING, FITCH DUKE M

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PROLYL HYDROXYLASE INHIBITORS von FITCH, DUKE, M, CHAI, DEPING

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