Novel hematopoietic progenitor kinase 1 inhibitor KHK-6 enhances T-cell activation von Ahn, Min Jeong, Kim, Eun Hye, Choi, Yunha, Chae, Chong Hak, Kim, Pilho, Kim, Seong Hwan

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A novel aminothiazole KY-05009 with potential to inhibit Traf2- and Nck-interacting kinase (TNIK) attenuates TGF-β1-mediated epithelial-to-mesenchymal transition in human lung aden... von Kim, Jiyeon, Moon, Seong-Hee, Kim, Bum Tae, Chae, Chong Hak, Lee, Joo Yun, Kim, Seong Hwan

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Discovery of TRD‐93 as a novel DRAK2 inhibitor von Park, Sangjun, Kye, Seungmin, Jung, Myoung Eun, Chae, Chong Hak, Yang, Kyung‐Min, Kim, Seong‐Jin, Choi, Gildon, Lee, Kwangho

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Biological evaluation of tanshindiols as EZH2 histone methyltransferase inhibitors von Woo, Jimin, Kim, Hyun-Young, Byun, Byung Jin, Chae, Chong-Hak, Lee, Ji Young, Ryu, Shi Yong, Park, Woo-Kyu, Cho, Heeyeong, Choi, Gildon

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The Predictive QSAR Model for hERG Inhibitors Using Bayesian and Random Forest Classification Method von Kim, Jun-Hyoung, Chae, Chong-Hak, Kang, Shin-Myung, Lee, Joo-Yon, Lee, Gil-Nam, Hwang, Soon-Hee, Kang, Nam-Sook

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Novel QSAR Models for Molecular Initiating Event Modeling in Two Intersecting Adverse Outcome Pathways Based Pulmonary Fibrosis Prediction for Biocidal Mixtures von Seo, Myungwon, Chae, Chong Hak, Lee, Yuno, Kim, Ha Ryong, Kim, Jongwoon

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A novel IRAK4/PIM1 inhibitor ameliorates rheumatoid arthritis and lymphoid malignancy by blocking the TLR/MYD88-mediated NF-κB pathway von Yoon, Sae-Bom, Hong, Hyowon, Lim, Hee-Jong, Choi, Ji Hye, Choi, Yoon Pyo, Seo, Seong Wook, Lee, Hyuk Woo, Chae, Chong Hak, Park, Woo-Kyu, Kim, Hyun Young, Jeong, Daeyoung, De, Tran Quang, Myung, Chang-Seon, Cho, Heeyeong

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Rational Design, Synthesis and Evaluation of Novel C6‐Bicycloalkaneimidazole Containing Imidazo[1,2‐b]pyridazines for ASK1 Inhibition von Lee, Yujin, Jang, Jiyoon, Bibi, Maimoona, Duggirala, Krishna Babu, Ji, Sang Hee, Lee, Ji Hun, Ahn, Sunjoo, Song, Jin Sook, Chae, Chong Hak, Kim, Seong Hwan, Lee, Kwangho

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Identification of a novel turn-on albumin binding small-molecule bioprobe in live zebrafish and its potential application in drug discovery von Chun, Hang-Suk, Han, Seo-Jung, Shin, Dae-Seop, Pagire, Haushabhau S., Pagire, Suvarna H., Lee, Gwi Bin, Chae, Chong Hak, Pak, Boryeong, Jin, Suk-Won, Chang, Young-Tae, Park, Seung Bum, Ahn, Jin Hee, Bae, Myung Ae

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Discovery and Characterization of a Novel MASTL Inhibitor MKI-2 Targeting MASTL-PP2A in Breast Cancer Cells and Oocytes von Kang, Minsung, Kim, Chijung, Leem, Jiyeon, Kim, Ye-hyun, Kwon, Young-ju, Yoon, Yi Na, Chae, Chong Hak, Ahn, Jiyeon, Jung, Kwan-Young, Oh, Jeong Su, Kim, Jae-Sung

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Chemical inhibitors destabilize HuR binding to the AU-rich element of TNF-α mRNA von Chae, Min-Ju, Sung, Hye Youn, Kim, Eun-Hye, Lee, Mira, Kwak, Hojoong, Chae, Chong Hak, Kim, Sunwoo, Park, Woong-Yang

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Identification of new pyrrole alkaloids from the fruits of Lycium chinense von Youn, Ui Joung, Lee, Joo Yun, Kil, Yun-Seo, Han, Ah-Reum, Chae, Chong Hak, Ryu, Shi Yong, Seo, Eun-Kyoung

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A novel assessment of nefazodone-induced hERG inhibition by electrophysiological and stereochemical method von Shin, Dae-Seop, Park, Myoung Joo, Lee, Hyang-Ae, Lee, Joo Yun, Chung, Hee-Chung, Yoo, Dae Seok, Chae, Chong Hak, Park, Sang-Joon, Kim, Ki-Suk, Bae, Myung Ae

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Fluorinated pyridinium oximes as potential reactivators for acetylcholinesterases inhibited by paraoxon organophosphorus agent von Jeong, Hee Chun, Park, No-Joong, Chae, Chong Hak, Musilek, Kamil, Kassa, Jiri, Kuca, Kamil, Jung, Young-Sik

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Docking-based 3D-QSAR study for selectivity of DPP4, DPP8, and DPP9 inhibitors von Kang, Nam Sook, Ahn, Jin Hee, Kim, Sung Soo, Chae, Chong Hak, Yoo, Sung-Eun

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Identification of 3-acyl-2-phenylamino-1,4-dihydroquinolin-4-one derivatives as inhibitors of the phosphatase SerB653 in Porphyromonas gingivalis, implicated in periodontitis von Jung, Suk-Kyeong, Ko, Youngkyung, Yu, Keum Ran, Kim, Ju Hee, Lee, Joo-Youn, Chae, Chong Hak, Ji, Suk, Kim, Chang Hyen, Lee, Hyeon Kyu, Choi, Eun Bok, Kim, Bo Yeon, Erikson, Raymond L., Chung, Sang J., Kim, Seung Jun

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Development and structure-activity relationship study of SHP2 inhibitor containing 3,4,6-trihydroxy-5-oxo-5H-benzo[7]annulene von Kim, Bohee, Jo, Seungjin, Park, Sung Bum, Chae, Chong Hak, Lee, Kwangho, Koh, Byumseok, Shin, Inji

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Novel allosteric glutaminase 1 inhibitors with macrocyclic structure activity relationship analysis von Lee, Eun Ji, Duggirala, Krishna Babu, Lee, Yujin, Yun, Mi Ran, Jang, Jiyoon, Cyriac, Rajath, Jung, Myoung Eun, Choi, Gildon, Chae, Chong Hak, Cho, Byoung Chul, Lee, Kwangho

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Synthesis and evaluation of tirbanibulin derivatives: a detailed exploration of the structure-activity relationship for anticancer activity von Park, Jaebeom, Kang, Minji, Lim, Ahyoung, Cho, Kyung-Jin, Chae, Chong Hak, Koh, Byumseok, Jeon, Hongjun

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Front Cover: Rotational Variance‐Based Data Augmentation in 3D Graph Convolutional Network (Chem. Asian J. 18/2021) von Kim, Jihoo, Kim, Yeji, Lee, Eok Kyun, Chae, Chong Hak, Lee, Kwangho, Kim, Won June, Choi, Insung S.

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