Ligand and Target Discovery by Fragment-Based Screening in Human Cells von Parker, Christopher G., Galmozzi, Andrea, Wang, Yujia, Correia, Bruno E., Sasaki, Kenji, Joslyn, Christopher M., Kim, Arthur S., Cavallaro, Cullen L., Lawrence, R. Michael, Johnson, Stephen R., Narvaiza, Iñigo, Saez, Enrique, Cravatt, Benjamin F.

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Microscale purification in support of high-throughput medicinal chemistry von Barhate, Chandan L, Donnell, Andrew F, Davies, Merrill, Li, Ling, Zhang, Yong, Yang, Fukang, Black, Regina, Zipp, Greg, Zhang, Yingru, Cavallaro, Cullen L, Priestley, E. Scott, Weller, Harold N

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Ni/Photoredox-Catalyzed C(sp2)–C(sp3) Cross-Coupling of Alkyl Pinacolboronates and (Hetero)Aryl Bromides von Cauley, Anthony N., Ramirez, Antonio, Barhate, Chandan L., Donnell, Andrew F., Khandelwal, Purnima, Sezen-Edmonds, Melda, Sherwood, Trevor C., Sloane, Jack L., Cavallaro, Cullen L., Simmons, Eric M.

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Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N‑Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-B... von Nimje, Roshan Y, Vytla, Devaiah, Kuppusamy, Prakasam, Velayuthaperumal, Rajeswari, Jarugu, Lokesh Babu, Reddy, China Anki, Chikkananjaiah, Nanjundaswamy Kanikahalli, Rampulla, Richard A, Cavallaro, Cullen L, Li, Jianqing, Mathur, Arvind, Gupta, Anuradha, Roy, Amrita

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Synthesis of Differentially Protected Azatryptophan Analogs via Pd 2 (dba) 3 /XPhos Catalyzed Negishi Coupling of N -Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected t... von Nimje, Roshan Y, Vytla, Devaiah, Kuppusamy, Prakasam, Velayuthaperumal, Rajeswari, Jarugu, Lokesh Babu, Reddy, China Anki, Chikkananjaiah, Nanjundaswamy Kanikahalli, Rampulla, Richard A, Cavallaro, Cullen L, Li, Jianqing, Mathur, Arvind, Gupta, Anuradha, Roy, Amrita

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Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists von Harikrishnan, Lalgudi S., Gill, Patrice, Kamau, Muthoni G., Qin, Lan-Ying, Ruan, Zheming, O'Malley, Daniel, Huynh, Tram, Stachura, Sylwia, Cavallaro, Cullen L., Lu, Zhonghui, J.-W. Duan, James, Weigelt, Carolyn A., Sack, John S., Ruzanov, Max, Khan, Javed, Gururajan, Murali, Wong, Jessica J., Huang, Yanling, Yarde, Melissa, Li, Zhuyin, Chen, Cliff, Sun, Huadong, Borowski, Virna, Murtaza, Anwar, Fink, Brian E.

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Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ von Myers, Michael C., Bilder, Donna M., Cavallaro, Cullen L., Chao, Hannguang J., Su, Shun, Burford, Neil T., Nayeem, Akbar, Wang, Tao, Yan, Mujing, Langish, Robert A., Dabros, Marta, Li, Yi-Xin, Rose, Anne V., Behnia, Kamelia, Onorato, Joelle M., Gargalovic, Peter S., Wexler, Ruth R., Lawrence, R. Michael

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Substituted diaryl ether compounds as retinoic acid-related orphan Receptor-γt (RORγt) agonists von Ruan, Zheming, Park, Peter K., Wei, Donna, Purandare, Ashok, Wan, Honghe, O'Malley, Daniel, Stachura, Sylwia, Perez, Heidi, Cavallaro, Cullen L., Weigelt, Carolyn A., Sack, John S., Ruzanov, Max, Khan, Javed, Gururajan, Murali, Wong, Jessica J., Huang, Yanling, Yarde, Melissa, Li, Zhuyin, Chen, Cliff, Sun, Huadong, Borowski, Virna, Xie, Jenny H., Anthony, Monique, Agler, Michele, Fink, Brian E., Harikrishnan, Lalgudi S.

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A compact, practical photoreactor for multi-reaction arrays von Brown, Gregory D, Batalla, Daniel, Cavallaro, Cullen L, Perez, Heidi L, Wrobleski, Stephen T, Sherwood, Trevor C

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Developing Adnectins That Target SRC Co-Activator Binding to PXR: A Structural Approach toward Understanding Promiscuity of PXR von Khan, Javed A., Camac, Daniel M., Low, Simon, Tebben, Andrew J., Wensel, David L., Wright, Martin C., Su, Julie, Jenny, Victoria, Gupta, Ruchira Das, Ruzanov, Max, Russo, Katie A., Bell, Aneka, An, Yongmi, Bryson, James W., Gao, Mian, Gambhire, Pallavi, Baldwin, Eric T., Gardner, Daniel, Cavallaro, Cullen L., Duncia, John V., Hynes, John

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Rapid Preparation of Variously Protected Glycals Using Titanium(III) von Spencer, Roxanne P, Cavallaro, Cullen L, Schwartz, Jeffrey

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Discovery and Lead Optimization of a Novel Series of CC Chemokine Receptor 1 (CCR1)-Selective Piperidine Antagonists via Parallel Synthesis von Cavallaro, Cullen L, Briceno, Stephanie, Chen, Jing, Cvijic, Mary Ellen, Davies, Paul, Hynes, John, Liu, Rui-Qin, Mandlekar, Sandhya, Rose, Anne V, Tebben, Andrew J, Van Kirk, Katy, Watson, Andrew, Wu, Hong, Yang, Guchen, Carter, Percy H

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Catalytic Dechlorination of Polychlorinated Biphenyls von Liu, Yumin, Schwartz, Jeffrey, Cavallaro, Cullen L

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Visible-light enabled one-pot three-component Petasis reaction for synthesis of α-substituted secondary sulfonamides/amides/hydrazides von Vytla, Devaiah, Emmadi, Jithendra, Velayuthaperumal, Rajeswari, Shaw, Parinita, Cavallaro, Cullen L., Mathur, Arvind, Roy, Amrita

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Increasing saturation: development of broadly applicable photocatalytic C sp2 –C sp3 cross-couplings of alkyl trifluoroborates and (hetero)aryl bromides for array synthesis von Cauley, Anthony N., Sezen-Edmonds, Melda, Simmons, Eric M., Cavallaro, Cullen L.

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Preparation of Aldehydo Sugars and Sugar Acids via Ozonolysis of Sugar Hydrazones von Spencer, Roxanne P, Bae Yu, Hye Kyung, Cavallaro, Cullen L, Schwartz, Jeffrey

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A Rapid Synthesis of Pyranoid Glycals from Glycosyl Bromides von Cavallaro, Cullen L, Schwartz, Jeffrey

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Increasing saturation: development of broadly applicable photocatalytic C-C cross-couplings of alkyl trifluoroborates and (hetero)aryl bromides for array synthesis von Cauley, Anthony N, Sezen-Edmonds, Melda, Simmons, Eric M, Cavallaro, Cullen L

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Increasing saturation: development of broadly applicable photocatalytic Csp2–Csp3 cross-couplings of alkyl trifluoroborates and (hetero)aryl bromides for array synthesis von Cauley, Anthony N, Sezen-Edmonds, Melda, Simmons, Eric M, Cavallaro, Cullen L

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Reduction of Glycosyl Bromides to Anhydroalditols by Titanocene Borohydride von Cavallaro, Cullen L, Schwartz, Jeffrey

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