Antitubercular drugs for an old target: GSK693 as a promising InhA direct inhibitor von Martínez-Hoyos, María, Perez-Herran, Esther, Gulten, Gulcin, Encinas, Lourdes, Álvarez-Gómez, Daniel, Alvarez, Emilio, Ferrer-Bazaga, Santiago, García-Pérez, Adolfo, Ortega, Fátima, Angulo-Barturen, Iñigo, Rullas-Trincado, Joaquin, Blanco Ruano, Delia, Torres, Pedro, Castañeda, Pablo, Huss, Sophie, Fernández Menéndez, Raquel, González del Valle, Silvia, Ballell, Lluis, Barros, David, Modha, Sundip, Dhar, Neeraj, Signorino-Gelo, François, McKinney, John D., García-Bustos, Jose Francisco, Lavandera, Jose Luis, Sacchettini, James C., Jimenez, M. Soledad, Martín-Casabona, Nuria, Castro-Pichel, Julia, Mendoza-Losana, Alfonso

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N-Benzyl-4-((heteroaryl)methyl)benzamides: A New Class of Direct NADH-Dependent 2-trans Enoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors with Antitubercular Activity von Guardia, Ana, Gulten, Gulcin, Fernandez, Raquel, Gómez, Jesus, Wang, Feng, Convery, Maire, Blanco, Delia, Martínez, María, Pérez-Herrán, Esther, Alonso, Marta, Ortega, Fátima, Rullás, Joaquín, Calvo, David, Mata, Lydia, Young, Robert, Sacchettini, James C., Mendoza-Losana, Alfonso, Remuiñán, Modesto, Ballell Pages, Lluís, Castro-Pichel, Julia

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4-Substituted Thioquinolines and Thiazoloquinolines: Potent, Selective, and Tween-80 in vitro Dependent Families of Antitubercular Agents with Moderate in vivo Activity von Escribano, Jaime, Rivero-Hernández, Cristina, Rivera, Hilda, Barros, David, Castro-Pichel, Julia, Pérez-Herrán, Esther, Mendoza-Losana, Alfonso, Angulo-Barturen, Íñigo, Ferrer-Bazaga, Santiago, Jiménez-Navarro, Elena, Ballell, Lluís

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Mycobacterium tuberculosis Decaprenylphosphoryl-β‑d‑ribose Oxidase Inhibitors: Expeditious Reconstruction of Suboptimal Hits into a Series with Potent in Vivo Activity von Borthwick, Jennifer A, Alemparte, Carlos, Wall, Ian, Whitehurst, Benjamin C, Argyrou, Argyrides, Burley, Glenn, de Dios-Anton, Paco, Guijarro, Laura, Monteiro, Maria Candida, Ortega, Fatima, Suckling, Colin J, Pichel, Julia Castro, Cacho, Monica, Young, Robert J

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Encoded Library Technology as a Source of Hits for the Discovery and Lead Optimization of a Potent and Selective Class of Bactericidal Direct Inhibitors of Mycobacterium tuberculos... von Encinas, Lourdes, O’Keefe, Heather, Neu, Margarete, Remuiñán, Modesto J, Patel, Amish M, Guardia, Ana, Davie, Christopher P, Pérez-Macías, Natalia, Yang, Hongfang, Convery, Maire A, Messer, Jeff A, Pérez-Herrán, Esther, Centrella, Paolo A, Álvarez-Gómez, Daniel, Clark, Matthew A, Huss, Sophie, O’Donovan, Gary K, Ortega-Muro, Fátima, McDowell, William, Castañeda, Pablo, Arico-Muendel, Christopher C, Pajk, Stane, Rullás, Joaquín, Angulo-Barturen, Iñigo, Álvarez-Ruíz, Emilio, Mendoza-Losana, Alfonso, Ballell Pages, Lluís, Castro-Pichel, Julia, Evindar, Ghotas

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An improved one-pot method for the stereoselective synthesis of the (2S,3R)-3-amino-2-hydroxy acids: key intermediates for bestatin and amastatin von Herranz, Rosario, Castro-Pichel, Julia, Vinuesa, Soledad, Garcia-Lopez, M. Teresa

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Cyclopropyl Carboxamides: A New Oral Antimalarial Series Derived from the Tres Cantos Anti-Malarial Set (TCAMS) von Rueda, Lourdes, Castellote, Isabel, Castro-Pichel, Julia, Chaparro, Maria J, de la Rosa, Juan Carlos, Garcia-Perez, Adolfo, Gordo, Mariola, Jimenez-Diaz, Maria Belen, Kessler, Albane, Macdonald, Simon J.F, Martinez, Maria Santos, Sanz, Laura M, Gamo, Francisco Javier, Fernandez, Esther

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Release of 50 new, drug-like compounds and their computational target predictions for open source anti-tubercular drug discovery: e0142293 von Rebollo-Lopez, Maria Jose, Lelievre, Joeel, Alvarez-Gomez, Daniel, Castro-Pichel, Julia, Martinez-Jimenez, Francisco, Papadatos, George, Kumar, Vinod, Colmenarejo, Gonzalo, Mugumbate, Grace, Hurle, Mark

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Tributyltin Cyanide, a Novel Reagent for the Stereoselective Preparation of 3-Amino-2-hydroxy Acids via Cyanohydrin Intermediates von Herranz, Rosario, Castro-Pichel, Julia, García-López, Teresa

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ANTITUBERCULOSIS AGENT von BATES, ROBERT H, ESQUIVIAS PROVENCIO, JORGE, BALLELL PAGES, LLUIS, BARROS AGUIRRE, DAVID, PETHE, KEVIN, CASTRO PICHEL, JULIA

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Ketomethylenebestatin: Synthesis and Aminopeptidase Inhibition von Herranz, Rosario, Castro-Pichel, Julia, García-López, M. Teresa, Gómez-Monterrey, Isabel, Pérez, Concepción, Vinuesa, Soledad

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ANTITUBERCULOSIS AGENT von BATES, ROBERT H, ESQUIVIAS PROVENCIO, JORGE, BALLELL PAGES, LLUIS, BARROS AGUIRRE, DAVID, PETHE, KEVIN, CASTRO PICHEL, JULIA

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ANTITUBERCULOSIS AGENT von BARROS AGUIRRE, David, BATES, Robert H, CASTRO PICHEL, Julia, BALLELL PAGES, Lluis, ESQUIVIAS PROVENCIO, Jorge, PETHE, Kevin

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ANTITUBERCULOSIS AGENT von BALLELL PAGES Lluis, BARROS AGUIRRE David, CASTRO PICHEL Julia, ESQUIVIAS PROVENCIO Jorge, PETHE Kevin, BATES Robert H

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ANTITUBERCULOSIS AGENT von BATES, ROBERT H, BALLELL, PAGES, LLUIS, CASTRO, PICHEL, JULIA, ESQUIVIAS, PROVENCIO, JORGE, PETHE, KEVIN, BARROS, AGUIRRE, DAVID

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ANTITUBERCULOSIS AGENT von BARROS AGUIRRE, David, BATES, Robert H, CASTRO PICHEL, Julia, BALLELL PAGES, Lluis, ESQUIVIAS PROVENCIO, Jorge, PETHE, Kevin

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Anti-tuberkulosemiddel von BARROS AGUIRRE, David, BATES, Robert H, CASTRO PICHEL, Julia, BALLELL PAGES, Lluis, ESQUIVIAS PROVENCIO, Jorge, PETHE, Kevin

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ANTITUBERCULOSIS AGENT von BARROS AGUIRRE, David, BATES, Robert, H, CASTRO PICHEL, Julia, BALLELL PAGES, Lluis, ESQUIVIAS PROVENCIO, Jorge, PETHE, Kevin

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Antituberculosis agent von Pethe, Kevin, Bates, Robert H, Ballell Pages, Lluis, Barros Aguirre, David, Esquivias Provencio, Jorge, Castro Pichel, Julia

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Synthesis of pyrimidine analogues of the nucleoside antibiotic ascamycin von Castro-Pichel, Julia, García-López, M. Teresa, De las Heras, Federico G., Herranz, Rosario

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