Defining the minimum inhibitory concentration of 22 rifamycins in iron limited, physiologic medium against Acinetobacter baumannii, Escherichia coli, and Klebsiella pneumoniae clin... von Lu, Peggy, Alletto, Francesco, Lee, Bosul, Burk, Elizabeth, Martinez, Jasmine, Prati, Fabio, Caselli, Emilia, Spellberg, Brad, Luna, Brian

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The β-Lactamase Inhibitor Boronic Acid Derivative SM23 as a New Anti- Pseudomonas aeruginosa Biofilm von Peppoloni, Samuele, Pericolini, Eva, Colombari, Bruna, Pinetti, Diego, Cermelli, Claudio, Fini, Francesco, Prati, Fabio, Caselli, Emilia, Blasi, Elisabetta

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Deciphering the Evolution of Cephalosporin Resistance to Ceftolozane-Tazobactam in Pseudomonas aeruginosa von Barnes, Melissa D, Taracila, Magdalena A, Rutter, Joseph D, Bethel, Christopher R, Galdadas, Ioannis, Hujer, Andrea M, Caselli, Emilia, Prati, Fabio, Dekker, John P, Papp-Wallace, Krisztina M, Haider, Shozeb, Bonomo, Robert A

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Fragment-guided design of subnanomolar β-lactamase inhibitors active in vivo von Eidam, Oliv, Romagnoli, Chiara, Dalmasso, Guillaume, Barelier, Sarah, Caselli, Emilia, Bonnet, Richard, Shoichet, Brian K, Prati, Fabio

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A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening von McGovern, Susan L, Caselli, Emilia, Grigorieff, Nikolaus, Shoichet, Brian K

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Biochemical and Structural Analysis of Inhibitors Targeting the ADC‑7 Cephalosporinase of Acinetobacter baumannii von Powers, Rachel A., Swanson, Hollister C., Taracila, Magdalena A., Florek, Nicholas W., Romagnoli, Chiara, Caselli, Emilia, Prati, Fabio, Bonomo, Robert A., Wallar, Bradley J.

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Insights Into the Inhibition of MOX-1 β-Lactamase by S02030, a Boronic Acid Transition State Inhibitor von Ishikawa, Tatsuya, Furukawa, Nayuta, Caselli, Emilia, Prati, Fabio, Taracila, Magdalena A, Bethel, Christopher R, Ishii, Yoshikazu, Shimizu-Ibuka, Akiko, Bonomo, Robert A

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One-Pot Synthesis of Imidazole-4-Carboxylates by Microwave-Assisted 1,5-Electrocyclization of Azavinyl Azomethine Ylides von Preti, Lisa, Attanasi, Orazio A., Caselli, Emilia, Favi, Gianfranco, Ori, Claudia, Davoli, Paolo, Felluga, Fulvia, Prati, Fabio

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Interactions of Oximino-Substituted Boronic Acids and β-Lactams with the CMY-2-Derived Extended-Spectrum Cephalosporinases CMY-30 and CMY-42 von KOTSAKIS, Stathis D, CASELLI, Emilia, TZOUVELEKIS, Leonidas S, PETINAKI, Efi, PRATI, Fabio, MIRIAGOU, Vivi

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Sulfonamidoboronic Acids as "Cross-Class" Inhibitors of an Expanded-Spectrum Class C Cephalosporinase, ADC-33, and a Class D Carbapenemase, OXA-24/40: Strategic Compound Design to... von Introvigne, Maria Luisa, Beardsley, Trevor J, Fernando, Micah C, Leonard, David A, Wallar, Bradley J, Rudin, Susan D, Taracila, Magdalena A, Rather, Philip N, Colquhoun, Jennifer M, Song, Shaina, Fini, Francesco, Hujer, Kristine M, Hujer, Andrea M, Prati, Fabio, Powers, Rachel A, Bonomo, Robert A, Caselli, Emilia

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Structures of FOX-4 Cephamycinase in Complex with Transition-State Analog Inhibitors von Lefurgy, Scott T, Caselli, Emilia, Taracila, Magdalena A, Malashkevich, Vladimir N, Biju, Beena, Papp-Wallace, Krisztina M, Bonanno, Jeffrey B, Prati, Fabio, Almo, Steven C, Bonomo, Robert A

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Straightforward synthesis of chiral non-racemic α-boryl isocyanides von Fini, Francesco, Zanni, Alessandro, Introvigne, Maria Luisa, Stucchi, Mattia, Caselli, Emilia, Prati, Fabio

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Synthesis of [(1,2,3-Triazol-1-yl)methyl]boronic Acids Through Click Chemistry: Easy Access to a Potential Scaffold for Protease Inhibitors von Romagnoli, Chiara, Caselli, Emilia, Prati, Fabio

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α‐Triazolylboronic Acids: A Novel Scaffold to Target FLT3 in AML von Introvigne, Maria Luisa, Destro, Lorenza, Mologni, Luca, Crippa, Valentina, Zardi, Paolo, Fini, Francesco, Prati, Fabio, Caselli, Emilia, Zambon, Alfonso

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Click Chemistry in Lead Optimization of Boronic Acids as β‑Lactamase Inhibitors von Caselli, Emilia, Romagnoli, Chiara, Vahabi, Roza, Taracila, Magdalena A., Bonomo, Robert A., Prati, Fabio

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Enantiomeric excess of 1,2-diols by formation of cyclic boronates: an improved method von Morandi, Stefania, Caselli, Emilia, Forni, Arrigo, Bucciarelli, Maria, Torre, Giovanni, Prati, Fabio

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Negative Epistasis and Evolvability in TEM-1 β-Lactamase—The Thin Line between an Enzyme's Conformational Freedom and Disorder von Dellus-Gur, Eynat, Elias, Mikael, Caselli, Emilia, Prati, Fabio, Salverda, Merijn L.M., de Visser, J. Arjan G.M., Fraser, James S., Tawfik, Dan S.

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Natural protein engineering in the Ω-loop: the role of Y221 in ceftazidime and ceftolozane resistance in Pseudomonas -derived cephalosporinase von Mack, Andrew R, Kumar, Vijay, Taracila, Magdalena A, Mojica, Maria F, O'Shea, Margaret, Schinabeck, William, Silver, Galen, Hujer, Andrea M, Papp-Wallace, Krisztina M, Chen, Shuang, Haider, Shozeb, Caselli, Emilia, Prati, Fabio, van den Akker, Focco, Bonomo, Robert A

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Synthesis of 1,2,3-triazol-1-yl-methaneboronic acids via click chemistry: an easy access to a new potential scaffold for protease inhibitors von Romagnoli, Chiara, Caselli, Emilia, Prati, Fabio

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α‐Triazolylboronic Acids: A Promising Scaffold for Effective Inhibitors of KPCs von Introvigne, Maria Luisa, Taracila, Magdalena A., Prati, Fabio, Caselli, Emilia, Bonomo, Robert A.

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