In vitro methods for estimating eye irritancy of cleaning products. I: Preliminary assessment von BOOMAN, K. A, CASCIERI, T. M, SEDLAK, R. I, DEMETRULIAS, J, DRIEDGER, A, GRIFFITH, J. F, GROCHOSKI, G. T, KONG, B, MCCORMICK, W. C. III, NORTH-ROOT, H, ROZEN, M. G

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Identification, localization and receptor characterization of novel mammalian substance P-like peptides von Kurtz, Marc M, Wang, Ruiping, Clements, Michelle K, Cascieri, Margaret A, Austin, Christopher P, Cunningham, Barry R, Chicchi, Gary G, Liu, Qingyun

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Distinct Mechanism for Antidepressant Activity by Blockade of Central Substance P Receptors von Kramer, Mark S., Cutler, Neal, Feighner, John, Shrivastava, Ram, Carman, John, Sramek, John J., Reines, Scott A., Liu, Guanghan, Snavely, Duane, Wyatt-Knowles, Edwina, Hale, Jeffrey J., Mills, Sander G., MacCoss, Malcolm, Swain, Christopher J., Harrison, Timothy, Hill, Raymond G., Hefti, Franz, Scolnick, Edward M., Cascieri, Margaret A., Chicchi, Gary G., Sadowski, Sharon, Williams, Angela R., Hewson, Louise, Smith, David, Carlson, Emma J., Hargreaves, Richard J., Nadia M. J. Rupniak

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The chemokine/chemokine-receptor family: potential and progress for therapeutic intervention von Cascieri, Margaret A, Springer, Martin S

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Structural Optimization Affording 2-(R)-(1-(R)-3,5-Bis(trifluoromethyl)phenylethoxy)-3-(S)-(4-fluoro)phenyl-4- (3-oxo-1,2,4-triazol-5-yl)methylmorpholine, a Potent, Orally Active,... von Hale, Jeffrey J, Mills, Sander G, MacCoss, Malcolm, Finke, Paul E, Cascieri, Margaret A, Sadowski, Sharon, Ber, Elzbieta, Chicchi, Gary G, Kurtz, Marc, Metzger, Joseph, Eiermann, George, Tsou, Nancy N, Tattersall, F. David, Rupniak, Nadia M. J, Williams, Angela R, Rycroft, Wayne, Hargreaves, Richard, MacIntyre, D. Euan

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Substituted Imidazoles as Glucagon Receptor Antagonists von Chang, Linda L., Sidler, Kelly L., Cascieri, Margaret A., de Laszlo, Stephen, Koch, Greg, Li, Bing, MacCoss, Malcolm, Mantlo, Nathan, O'Keefe, Stephen, Pang, Margaret, Rolando, Anna, Hagmann, William K.

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Amino-aromatic interaction between histidine 197 of the neurokinin-1 receptor and CP 96345 von Ming Fong, Tung, Cascieri, Margaret A, Yu, Hong, Bansal, Alka, Swain, Christopher, Strader, Catherine D

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Potent, orally absorbed glucagon receptor antagonists von de Laszlo, Stephen E., Hacker, Candice, Li, Bing, Kim, Dooseop, MacCoss, Malcolm, Mantlo, Nathan, Pivnichny, James V., Colwell, Larry, Koch, Gregory E., Cascieri, Margaret A., Hagmann, William K.

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The potential for novel anti-inflammatory therapies for coronary artery disease von Cascieri, Margaret A

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Molecular cloning and characterization of a new receptor for galanin von Howard, Andrew D, Tan, Carina, Shiao, Lin-Lin, Palyha, Oksana C, McKee, Karen Kulju, Weinberg, David H, Feighner, Scott D, Cascieri, Margaret A, Smith, Roy G, Van Der Ploeg, Lex H.T, Sullivan, Kathleen A

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Receptor for Motilin Identified in the Human Gastrointestinal System von Feighner, Scott D., Tan, Carina P., McKee, Karen Kulju, Palyha, Oksana C., Hreniuk, Donna L., Pong, Sheng-Shung, Austin, Christopher P., Figueroa, David, MacNeil, Douglas, Cascieri, Margaret A., Nargund, Ravi, Bakshi, Raman, Abramovitz, Mark, Stocco, Rino, Kargman, Stacia, O'Neill, Gary, Lex H. T. Van Der Ploeg, Evans, Jilly, Patchett, Arthur A., Smith, Roy G., Howard, Andrew D.

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Cloning and Expression of a Novel Neuropeptide Y Receptor von Weinberg, David H., Sirinathsinghji, Dalip J.S., Tan, Carina P., Shiao, Lin-Lin, Morin, Nancy, Rigby, Michael R., Heavens, Robert H., Rapoport, Davida R., Bayne, Marvin L., Cascieri, Margaret A., Strader, Catherine D., Linemeyer, David L., MacNeil, Douglas J.

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Peroxisome proliferator-activated receptors gamma and alpha mediate in vivo regulation of uncoupling protein (UCP-1, UCP-2, UCP-3) gene expression von Kelly, L J, Vicario, P P, Thompson, G M, Candelore, M R, Doebber, T W, Ventre, J, Wu, M S, Meurer, R, Forrest, M J, Conner, M W, Cascieri, M A, Moller, D E

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Phosphorylated Morpholine Acetal Human Neurokinin-1 Receptor Antagonists as Water-Soluble Prodrugs von Hale, Jeffrey J, Mills, Sander G, MacCoss, Malcolm, Dorn, Conrad P, Finke, Paul E, Budhu, Richard J, Reamer, Robert A, Huskey, Su-Er W, Luffer-Atlas, Debra, Dean, Brian J, McGowan, Erin M, Feeney, William P, Chiu, Shuet-Hing Lee, Cascieri, Margaret A, Chicchi, Gary G, Kurtz, Marc M, Sadowski, Sharon, Ber, Elzbieta, Tattersall, F. David, Rupniak, Nadia M. J, Williams, Angela R, Rycroft, Wayne, Hargreaves, Richard, Metzger, Joseph M, MacIntyre, D. Euan

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An Orally Active, Water-Soluble Neurokinin-1 Receptor Antagonist Suitable for Both Intravenous and Oral Clinical Administration von Harrison, Timothy, Owens, Andrew P, Williams, Brian J, Swain, Christopher J, Williams, Angela, Carlson, Emma J, Rycroft, Wayne, Tattersall, F. David, Cascieri, Margaret A, Chicchi, Gary G, Sadowski, Sharon, Rupniak, Nadia M. J, Hargreaves, Richard J

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Human β 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides von Brockunier, Linda L, Parmee, Emma R, Ok, Hyun O, Candelore, Mari R, Cascieri, Margaret A, Colwell, Lawrence F, Deng, Liping, Feeney, William P, Forrest, Michael J, Hom, Gary J, MacIntyre, D.Euan, Tota, Laurie, Wyvratt, Matthew J, Fisher, Michael H, Weber, Ann E

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The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L-758,298, inhibit acute and delayed cisplatin-induced emesis in ferrets von TATTERSALL, F. D, RYCROFT, W, SADOWSKI, S, BER, E, CASCIERI, M, HILL, R. G, MACINTYRE, D. E, HARGREAVES, R. J, CUMBERBATCH, M, MASON, G, TYE, S, WILLIAMSON, D. J, HALE, J. J, MILLS, S. G, FINKE, P. E, MACCOSS, M

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In vitro and in vivo predictors of the anti-emetic activity of tachykinin NK1 receptor antagonists von RUPNIAK, N. M. J, TATTERSALL, F. D, MACCOSS, M, SEWARD, E, HUSCROFT, I, OWEN, S, SWAIN, C. J, HILL, R. G, HARGREAVES, R. J, WILLIAMS, A. R, RYCROFT, W, CARLSON, E. J, CASCIERI, M. A, SADOWSKI, S, BER, E, HALE, J. J, MILLS, S. G

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Characterization of a Novel, Non-peptidyl Antagonist of the Human Glucagon Receptor von Cascieri, M A, Koch, G E, Ber, E, Sadowski, S J, Louizides, D, de Laszlo, S E, Hacker, C, Hagmann, W K, MacCoss, M, Chicchi, G G, Vicario, P P

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Discovery of 3,5-bis(trifluoromethyl)benzyl l-arylglycinamide based potent CCR2 antagonists von Yang, Lihu, Zhou, Changyou, Guo, Liangqin, Morriello, Gregori, Butora, Gabor, Pasternak, Alexander, Parsons, William H., Mills, Sander G., MacCoss, Malcolm, Vicario, Pasquale P., Zweerink, Hans, Ayala, Julia M., Goyal, Shefali, Hanlon, William A., Cascieri, Margaret A., Springer, Marty S.

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