ACE and LRPAP1 Insertion-Deletion Polymorphisms in a Northern Ivory Coast Population von Santovito, A., Bulgarello, C., Caravatti, G. A., Ouattará, M., Cervella, P., Pisano, G., Salvarani, B., Delpero, M.

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AEE788: A dual family epidermal growth factor receptor/ErbB2 and vascular endothelial growth factor receptor tyrosine kinase inhibitor with antitumor and antiangiogenic activity von TRAXLER, Peter, ALLEGRINI, Peter R, MEYER, Thomas, TANG, Careen, WARTMANN, Markus, WOOD, Jeanette, CARAVATTI, Giorgio, BRANDT, Ralf, BRUEGGEN, Josef, COZENS, Robert, FABBRO, Doriano, GROSIOS, Konstantina, LANE, Heidi A, MCSHEEHY, Paul, MESTAN, Jürgen

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A derivative of staurosporine (CGP 41 251) shows selectivity for protein kinase C inhibition and In vitro anti‐proliferative as well as In vivo anti‐tumor activity von Meyer, Thomas, Regenass, Urs, Fabbro, Doriano, Alteri, Enrica, Röusel, Johannes, Möller, Marcel, Caravatti, Giorgio, Matter, Alex

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Tyrosine kinase inhibitors: From rational design to clinical trials von Traxler, Peter, Bold, Guido, Buchdunger, Elisabeth, Caravatti, Giorgio, Furet, Pascal, Manley, Paul, O'Reilly, Terence, Wood, Jeanette, Zimmermann, Juerg

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Erythrocyte polymorphisms in five ethnic groups of Northern Côte d'Ivoire von Santovito, A., Burgarello, C., Cervella, P., Ouattara, M., Caravatti, G. A., Salvarani, B., Delpero, M.

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Potent Antagonists of the SH2 Domain of Grb2:  Optimization of the X+1 Position of 3-Amino-Z-Tyr(PO3H2)-X+1-Asn-NH2 von García-Echeverría, Carlos, Furet, Pascal, Gay, Brigitte, Fretz, Heinz, Rahuel, Joseph, Schoepfer, Joseph, Caravatti, Giorgio

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Protein kinases as targets for anticancer agents: from inhibitors to useful drugs von Fabbro, Doriano, Ruetz, Stephan, Buchdunger, Elisabeth, Cowan-Jacob, Sandra W, Fendrich, Gabriele, Liebetanz, Janis, Mestan, Jürgen, O'Reilly, Terence, Traxler, Peter, Chaudhuri, Bhabatosh, Fretz, Heinz, Zimmermann, Jürg, Meyer, Thomas, Caravatti, Giorgio, Furet, Pascal, Manley, Paul W

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Structural basis for specificity of GRB2-SH2 revealed by a novel ligand binding mode von Rahuel, Joseph, Gay, Brigitte, Erdmann, Dirk, Strauss, André, García-Echeverría, Carlos, Furet, Pascal, Caravatti, Giorgio, Fretz, Heinz, Schoepfer, Joseph, Grütter, Markus G

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COL1A2 gene deletion polymorphism in an Italian and an Ivorian populations von Santovito, A., Burgarello, C., Cervella, P., Caravatti, G. A., Ouattara, M., Salvarani, B., Delpero, M.

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In vitro trypanocidal activities of new S-adenosylmethionine decarboxylase inhibitors von BRUN, R, BÜHLER, Y, CARAVATTI, G, FREI, J, STANEK, J, METT, H, SANDMEIER, U, KAMINSKY, R, BACCHI, C. J, RATTENDI, D, LANE, S, CROFT, S. L, SNOWDON, D, YARDLEY, V

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Antileukemic Effects of Novel First- and Second-Generation FLT3 Inhibitors: Structure-Affinity Comparison von Weisberg, Ellen, Roesel, Johannes, Furet, Pascal, Bold, Guido, Imbach, Patricia, Flörsheimer, Andreas, Caravatti, Georgio, Jiang, Jingrui, Manley, Paul, Ray, Arghya, Griffin, James D

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The Total Synthesis and Biological Assessment of trans-Epothilone A von Altmann, Karl-Heinz, Bold, Guido, Caravatti, Giorgio, Denni, Donatienne, Flörsheimer, Andreas, Schmidt, Alfred, Rihs, Grety, Wartmann, Markus

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Selective GRB2 SH2 inhibitors as anti‐Ras therapy von Gay, Brigitte, Suarez, Stéphanie, Caravatti, Giorgio, Furet, Pascal, Meyer, Thomas, Schoepfer, Joseph

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Synthesis and biological evaluation of highly potent analogues of epothilones B and D von Altmann, Karl-Heinz, Bold, Guido, Caravatti, Giorgio, Flörsheimer, Andreas, Guagnano, Vito, Wartmann, Markus

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Structure-Based Design and Synthesis of High Affinity Tripeptide Ligands of the Grb2-SH2 Domain von Furet, Pascal, Gay, Brigitte, Caravatti, Giorgio, García-Echeverría, Carlos, Rahuel, Joseph, Schoepfer, Joseph, Fretz, Heinz

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Author errata von Lydon, N, Mett, H, Mueller, M, Becker, M, Cozens, R M, Daniels, D, Traxler, P, Buchdunger, E, Stover, D

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Effect of Potent and Selective Inhibitors of the Grb2 SH2 Domain on Cell Motility von Gay, Brigitte, Suarez, Stéphanie, Weber, Christine, Rahuel, Joseph, Fabbro, Doriano, Furet, Pascal, Caravatti, Giorgio, Schoepfer, Joseph

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Structural basis for the high affinity of amino-aromatic SH2 phosphopeptide ligands von Rahuel, Joseph, Garcı́a-Echeverrı́a, Carlos, Furet, Pascal, Strauss, André, Caravatti, Giorgio, Fretz, Heinz, Schoepfer, Joseph, Gay, Brigitte

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Discovery of 3-Aminobenzyloxycarbonyl as an N-Terminal Group Conferring High Affinity to the Minimal Phosphopeptide Sequence Recognized by the Grb2-SH2 Domain von Furet, Pascal, Gay, Brigitte, García-Echeverría, Carlos, Rahuel, Joseph, Fretz, Heinz, Schoepfer, Joseph, Caravatti, Giorgio

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Highly potent inhibitors of the Grb2-SH2 domain von Schoepfer, Joseph, Fretz, Heinz, Gay, Brigitte, Furet, Pascal, García-Echeverría, Carlos, End, Nicole, Caravatti, Giorgio

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