The synthesis and structure–activity relationship of substituted N-phenyl anthranilic acid analogs as amyloid aggregation inhibitors von Simons, Lloyd J., Caprathe, Bradley W., Callahan, Michael, Graham, James M., Kimura, Takenori, Lai, Yingjie, LeVine, Harry, Lipinski, William, Sakkab, Annette T., Tasaki, Yoshikazu, Walker, Lary C., Yasunaga, Tomoyuki, Ye, Yuyang, Zhuang, Nian, Augelli-Szafran, Corinne E.

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2-Amino-4H-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease von Hays, Sheryl J, Caprathe, Bradley W, Gilmore, John L, Amin, Nilam, Emmerling, Mark R, Michael, Walter, Nadimpalli, Ravi, Nath, Rathna, Raser, Kadee J, Stafford, Daniel, Watson, Desiree, Wang, Kevin, Jaen, Juan C

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Design and Synthesis of m1-Selective Muscarinic Agonists:  (R)-(−)-(Z)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-(3‘-Methoxyphenyl)-2-propynyl)- oxime Maleate (CI-1017), a Functionally... von Tecle, Haile, Barrett, Stephen D, Lauffer, David J, Augelli-Szafran, Corinne, Brann, Mark R, Callahan, Michael J, Caprathe, Bradley. W, Davis, Robert E, Doyle, Patricia D, Eubanks, David, Lipiniski, William, Mirzadegan, Tara, Moos, Walter H, Moreland, D. W, Nelson, Carrie B, Pavia, Michael R, Raby, Charlotte, Schwarz, Roy D, Spencer, Carolyn J, Thomas, Anthony J, Jaen, Juan C

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The Discovery and Structure-Activity Relationships of 1,2,3,6-Tetrahydro-4-phenyl-1-[(arylcyclohexenyl)alkyl]pyridines. Dopamine Autoreceptor Agonists and Potential Antipsychotic A... von Wright, Jon L, Caprathe, Bradley W, Downing, Dennis M, Glase, Shelly A, Heffner, Thomas G, Jaen, Juan C, Johnson, Stephen J, Kesten, Suzanne R, MacKenzie, Robert G

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4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties von Jaen, Juan C, Wise, Lawrence D, Caprathe, Bradley W, Tecle, Haile, Bergmeier, Stephen, Humblet, Christine C, Heffner, Thomas G, Meltzer, Leonard T, Pugsley, Thomas A

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Kynurenic Acid Derivatives Inhibit the Binding of Nerve Growth Factor (NGF) to the Low-Affinity p75 NGF Receptor von Jaen, Juan C, Laborde, Edgardo, Bucsh, Ruth A, Caprathe, Bradley W, Sorenson, Roderick J, Fergus, James, Spiegel, Katharyn, Marks, James, Dickerson, Melvin R, Davis, Robert E

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Evaluation of the effects of the enantiomers of reduced haloperidol, azaperol, and related 4-amino-1-arylbutanols on dopamine and .sigma. receptors von Jaen, Juan C, Caprathe, Bradley W, Pugsley, Thomas A, Wise, Lawrence D, Akunne, Hyacinth

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Identification of a 3-Hydroxylated Tacrine Metabolite in Rat and Man:  Metabolic Profiling Implications and Pharmacology von Pool, William F, Woolf, Thomas F, Reily, Michael D, Caprathe, Bradley W, Emmerling, Mark R, Jaen, Juan C

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Dopamine autoreceptor agonists as potential antipsychotics. 3. 6-Propyl-4,5,5a,6,7,8-hexahydrothiazolo[4,5-f]quinolin-2-amine von Caprathe, Bradley W, Jaen, Juan C, Wise, Lawrence D, Heffner, Thomas G, Pugsley, Thomas A, Meltzer, Leonard T, Parvez, Masood

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Amnesia-reversal activity of a series of cyclic imides von Butler, Donald E, Leonard, James D, Caprathe, Bradley W, L'Italien, Yvon J, Pavia, Michael R, Hershenson, Fred M, Poschel, Paul H, Marriott, John G

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Nitrones by heterolytic fragmentation of .gamma.-N-hydroxyamino sulfonates. Conversion of a decahydroquinoline to a perhydroazaazulene von LeBel, Norman A, Caprathe, Bradley W

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Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitors von Gilmore, John L., Hays, Sheryl J., Caprathe, Bradley W., Lee, Chitase, Emmerling, Mark R., Michael, Walter, Jaen, Juan C.

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2-Amino-4 H -3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease von Hays, Sheryl J., Caprathe, Bradley W., Gilmore, John L., Amin, Nilam, Emmerling, Mark R., Michael, Walter, Nadimpalli, Ravi, Nath, Rathna, Raser, Kadee J., Stafford, Daniel, Watson, Desiree, Wang, Kevin, Jaen, Juan C.

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Synthesis of the enantiomers of reduced haloperidol von JAEN, J. C, CAPRATHE, B. W, PRIEBE, S, WISE, L. D

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EFFICIENT SYNTHESIS OF EXO-1-AZABICYCLO[2.2.1]HEPTAN-3-OL von Barrett, Stephen D., Jaen, Juan C., Caprathe, Bradley W., Thomas, Anthony J., Tecle, Haile

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Synthesis and pharmacological evaluation of the enantiomers of the dopamine autoreceptor agonist PD 135385 von Jaén, Juan C., Caprathe, Bradley W., Wise, Lawrence D., Meltzer, Leonard T., Pugsley, Thomas A., Huffner, Thomas G.

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PYRIMIDINE TRICYCLIC ENONE DERIVATIVES FOR INHIBITION OF ROR[gamma] AND OTHER USES von CAPRATHE BRADLEY W, SHELDON ZACHARY S, LEE CHITASE, HOTEMA MARTHA R, BENDER CHRISTOPHER F, JIANG XIN, VISNICK MELEAN, BOLTON GARY, KORNBERG BRIAN

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Synthesis and dopaminergic activity of the enantiomers of 6-methyl-4,5a,6,7,8-hexahydrothiazolo[4,5-f]quinolin-2-amine (PD 128483) von Jaen, Juan C., Caprathe, Bradley W., Wise, Lawrence D., Pugsley, Thomas A., Meltzer, Leonard T., Heffner, Thomas G.

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Piperidine Derivatives von CAPRATHE BRADLEY W, JENNINGS REX A, SIMONS LLOYD J, GOGLIOTTI ROCCO D

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Novel 4,5,6,7-tetrahydrobenzothiazole dopamine agonists display very low stereoselectivity in their interaction with dopamine receptors von Jaen, Juan C., Caprathe, Bradley W., Wise, Lawrence D., Smith, Sarah J., Pugsley, Thomas A., Heffner, Thomas G., Meltzer, Leonard T.

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