The synthesis and structure–activity relationship of substituted N-phenyl anthranilic acid analogs as amyloid aggregation inhibitors von Simons, Lloyd J., Caprathe, Bradley W., Callahan, Michael, Graham, James M., Kimura, Takenori, Lai, Yingjie, LeVine, Harry, Lipinski, William, Sakkab, Annette T., Tasaki, Yoshikazu, Walker, Lary C., Yasunaga, Tomoyuki, Ye, Yuyang, Zhuang, Nian, Augelli-Szafran, Corinne E.

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2-Amino-4H-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease von Hays, Sheryl J, Caprathe, Bradley W, Gilmore, John L, Amin, Nilam, Emmerling, Mark R, Michael, Walter, Nadimpalli, Ravi, Nath, Rathna, Raser, Kadee J, Stafford, Daniel, Watson, Desiree, Wang, Kevin, Jaen, Juan C

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Design and Synthesis of m1-Selective Muscarinic Agonists:  (R)-(−)-(Z)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-(3‘-Methoxyphenyl)-2-propynyl)- oxime Maleate (CI-1017), a Functionally... von Tecle, Haile, Barrett, Stephen D, Lauffer, David J, Augelli-Szafran, Corinne, Brann, Mark R, Callahan, Michael J, Caprathe, Bradley. W, Davis, Robert E, Doyle, Patricia D, Eubanks, David, Lipiniski, William, Mirzadegan, Tara, Moos, Walter H, Moreland, D. W, Nelson, Carrie B, Pavia, Michael R, Raby, Charlotte, Schwarz, Roy D, Spencer, Carolyn J, Thomas, Anthony J, Jaen, Juan C

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4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties von Jaen, Juan C, Wise, Lawrence D, Caprathe, Bradley W, Tecle, Haile, Bergmeier, Stephen, Humblet, Christine C, Heffner, Thomas G, Meltzer, Leonard T, Pugsley, Thomas A

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Succinic acid amides as P2–P3 replacements for inhibitors of interleukin-1β converting enzyme (ICE or caspase 1) von Galatsis, Paul, Caprathe, Bradley, Gilmore, John, Thomas, Anthony, Linn, Kristin, Sheehan, Susan, Harter, William, Kostlan, Catherine, Lunney, Elizabeth, Stankovic, Charles, Rubin, John, Brady, Kenneth, Allen, Hamish, Talanian, Robert

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Kynurenic Acid Derivatives Inhibit the Binding of Nerve Growth Factor (NGF) to the Low-Affinity p75 NGF Receptor von Jaen, Juan C, Laborde, Edgardo, Bucsh, Ruth A, Caprathe, Bradley W, Sorenson, Roderick J, Fergus, James, Spiegel, Katharyn, Marks, James, Dickerson, Melvin R, Davis, Robert E

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The Discovery and Structure-Activity Relationships of 1,2,3,6-Tetrahydro-4-phenyl-1-[(arylcyclohexenyl)alkyl]pyridines. Dopamine Autoreceptor Agonists and Potential Antipsychotic A... von Wright, Jon L, Caprathe, Bradley W, Downing, Dennis M, Glase, Shelly A, Heffner, Thomas G, Jaen, Juan C, Johnson, Stephen J, Kesten, Suzanne R, MacKenzie, Robert G

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Evaluation of the effects of the enantiomers of reduced haloperidol, azaperol, and related 4-amino-1-arylbutanols on dopamine and .sigma. receptors von Jaen, Juan C, Caprathe, Bradley W, Pugsley, Thomas A, Wise, Lawrence D, Akunne, Hyacinth

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Identification of a 3-Hydroxylated Tacrine Metabolite in Rat and Man:  Metabolic Profiling Implications and Pharmacology von Pool, William F, Woolf, Thomas F, Reily, Michael D, Caprathe, Bradley W, Emmerling, Mark R, Jaen, Juan C

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The design and synthesis of sulfonamides as caspase-1 inhibitors von Harter, William G., Albrect, Hans, Brady, Kenneth, Caprathe, Bradley, Dunbar, James, Gilmore, John, Hays, Sheryl, Kostlan, Catherine R., Lunney, Beth, Walker, Nigel

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Inhibition of interleukin-1β converting enzyme (ICE or caspase 1) by aspartyl acyloxyalkyl ketones and aspartyl amidooxyalkyl ketones von Galatsis, Paul, Caprathe, Bradley, Downing, Dennis, Gilmore, John, Harter, William, Hays, Sheryl, Kostlan, Catherine, Linn, Kristin, Lunney, Elizabeth, Para, Kim, Thomas, Anthony, Warmus, Joseph, Allen, Hamish, Brady, Kenneth, Talanian, Robert, Walker, Nigel

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Dopamine autoreceptor agonists as potential antipsychotics. 3. 6-Propyl-4,5,5a,6,7,8-hexahydrothiazolo[4,5-f]quinolin-2-amine von Caprathe, Bradley W, Jaen, Juan C, Wise, Lawrence D, Heffner, Thomas G, Pugsley, Thomas A, Meltzer, Leonard T, Parvez, Masood

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Inhibition of interteukin-1β converting enzyme (ICE or caspase 1) by aspartyl acyloxyalkyl ketones and aspartyl amidooxyalkyl ketones von GALATSIS, Paul, CAPRATHE, Bradley, THOMAS, Anthony, WARMUS, Joseph, ALLEN, Hamish, BRADY, Kenneth, TALANIAN, Robert, WALKER, Nigel, DOWNING, Dennis, GILMORE, John, HARTER, William, HAYS, Sheryl, KOSTLAN, Catherine, LINN, Kristin, LUNNEY, Elizabeth, PARA, Kim

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Design, Synthesis, and Biological Activity of Novel Polycyclic Aza-Amide FKBP12 Ligands von Hudack, Raymond A, Barta, Nancy S, Guo, Chuangxing, Deal, Judith, Dong, Liming, Fay, Lorraine K, Caprathe, Bradley, Chatterjee, Arindam, Vanderpool, Darin, Bigge, Christopher, Showalter, Richard, Bender, Steve, Augelli-Szafran, Corinne E, Lunney, Elizabeth, Hou, Xinjun

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Amnesia-reversal activity of a series of cyclic imides von Butler, Donald E, Leonard, James D, Caprathe, Bradley W, L'Italien, Yvon J, Pavia, Michael R, Hershenson, Fred M, Poschel, Paul H, Marriott, John G

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BIARYL AMIDES WITH MODIFIED SUGAR GROUPS FOR TREATMENT OF DISEASES ASSOCIATED WITH HEAT SHOCK PROTEIN PATHWAY von BOLTON, Gary, BENDER, Christopher F, CAPRATHE, Bradley, JIANG, Xin, VISNICK, Melean, LEE, Chitase

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Biaryl amides with modified sugar groups for treatment of diseases associated with heat shock protein pathway von BOLTON, Gary, BENDER, Christopher F, CAPRATHE, Bradley, JIANG, Xin, VISNICK, Melean, LEE, Chitase

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BIARYL AMIDES WITH MODIFIED SUGAR GROUPS FOR TREATMENT OF DISEASES ASSOCIATED WITH HEAT SHOCK PROTEIN PATHWAY von BOLTON, Gary, BENDER, Christopher F, CAPRATHE, Bradley, JIANG, Xin, VISNICK, Melean, LEE, Chitase

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PYRAZOLE AND IMIDAZOLE COMPOUNDS FOR INHIBITION OF IL-17 AND RORGAMMA von BOLTON, Gary, BENDER, Christopher F, CAPRATHE, Bradley, HOTEMA, Martha R, JIANG, Xin, KORNBERG, Brian, O'BRIEN, Patrick, VISNICK, Melean, LEE, Chitase

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Biaryl amides with modified sugar groups for treatment of diseases associated with heat shock protein pathway von Jiang, Xin, Lee, Chitase, Bender, Christopher F, Bolton, Gary, Caprathe, Bradley, Visnick, Melean

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