Oxadiazolone bioisosteres of pregabalin and gabapentin von Wustrow, David J., Belliotti, Thomas R., Capiris, Thomas, Kneen, Clare O., Bryans, Justin S., Field, Mark J., Williams, Dic, El-Kattan, Ayman, Buchholz, Lisa, Kinsora, Jack J., Lotarski, Susan M., Vartanian, Mark G., Taylor, Charles P., Donevan, Sean D., Thorpe, Andrew J., Schwarz, Jacob B.

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Structure-activity relationships of pregabalin and analogues that target the alpha(2)-delta protein von Belliotti, Thomas R, Capiris, Thomas, Ekhato, I Victor, Kinsora, Jack J, Field, Mark J, Heffner, Thomas G, Meltzer, Leonard T, Schwarz, Jacob B, Taylor, Charles P, Thorpe, Andrew J, Vartanian, Mark G, Wise, Lawrence D, Zhi-Su, Ti, Weber, Mark L, Wustrow, David J

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Structure−Activity Relationships of Pregabalin and Analogues That Target the α2-δ Protein von Belliotti, Thomas R, Capiris, Thomas, Ekhato, I. Victor, Kinsora, Jack J, Field, Mark J, Heffner, Thomas G, Meltzer, Leonard T, Schwarz, Jacob B, Taylor, Charles P, Thorpe, Andrew J, Vartanian, Mark G, Wise, Lawrence D, Zhi-Su, Ti, Weber, Mark L, Wustrow, David J

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The preparation of optically active α-amino 4H-[1,2,4]oxadiazol-5-ones from optically active α-amino acids von MANGETTE, John E, JOHNSON, Matthew R, LE, Van-Duc, SHENOY, Rajesh A, ROARK, Howard, STIER, Michael, BELLIOTTI, Thomas, CAPIRIS, Thomas, GUZZO, Peter R

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The preparation of optically active α-amino 4 H-[1,2,4]oxadiazol-5-ones from optically active α-amino acids von Mangette, John E., Johnson, Matthew R., Le, Van-Duc, Shenoy, Rajesh A., Roark, Howard, Stier, Michael, Belliotti, Thomas, Capiris, Thomas, Guzzo, Peter R.

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Carboxylate bioisosteres of gabapentin von Burgos-Lepley, Carmen E., Thompson, Lisa R., Kneen, Clare O., Osborne, Simon A., Bryans, Justin S., Capiris, Thomas, Suman-Chauhan, Nirmala, Dooley, David J., Donovan, Cindy M., Field, Mark J., Vartanian, Mark G., Kinsora, Jack J., Lotarski, Susan M., El-Kattan, Ayman, Walters, Karen, Cherukury, Madhu, Taylor, Charles P., Wustrow, David J., Schwarz, Jacob B.

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Chromeno[3,4- c ]pyridin-5-ones:  Selective Human Dopamine D 4 Receptor Antagonists as Potential Antipsychotic Agents von Unangst, Paul C., Capiris, Thomas, Connor, David T., Heffner, Thomas G., MacKenzie, Robert G., Miller, Steven R., Pugsley, Thomas A., Wise, Lawrence D.

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Chromeno[3,4-c]pyridin-5-ones:  Selective Human Dopamine D4 Receptor Antagonists as Potential Antipsychotic Agents von Unangst, Paul C, Capiris, Thomas, Connor, David T, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D

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Pyrazolo[1,5-a]pyrimidine CRF-1 receptor antagonists von Wustrow, David J., Capiris, Thomas, Rubin, Ronald, Knobelsdorf, James A., Akunne, Hyacinth, Davis, M.Duff, MacKenzie, Robert, Pugsley, Thomas A., Zoski, Kim T., Heffner, Thomas G., Wise, Lawrence D.

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Structure−Activity Relationships of Pregabalin and Analogues That Target the α 2 -δ Protein von Belliotti, Thomas R., Capiris, Thomas, Ekhato, I. Victor, Kinsora, Jack J., Field, Mark J., Heffner, Thomas G., Meltzer, Leonard T., Schwarz, Jacob B., Taylor, Charles P., Thorpe, Andrew J., Vartanian, Mark G., Wise, Lawrence D., Zhi-Su, Ti, Weber, Mark L., Wustrow, David J.

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Carboxylate bioisosteres of gabapentin Dedicated to David W. Robertson in memory of his outstanding contributions as a mentor and drug hunter von Burgos-Lepley, Carmen E, Thompson, Lisa R, Kneen, Clare O, Osborne, Simon A, Bryans, Justin S, Capiris, Thomas, Suman-Chauhan, Nirmala, Dooley, David J, Donovan, Cindy M, Field, Mark J, Vartanian, Mark G, Kinsora, Jack J, Lotarski, Susan M, El-Kattan, Ayman, Walters, Karen, Cherukury, Madhu, Taylor, Charles P, Wustrow, David J, Schwarz, Jacob B

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(Aryloxy)alkylamines as Selective Human Dopamine D4 Receptor Antagonists:  Potential Antipsychotic Agents von Unangst, Paul C, Capiris, Thomas, Connor, David T, Doubleday, Robert, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D

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(Aryloxy)alkylamines as Selective Human Dopamine D 4 Receptor Antagonists:  Potential Antipsychotic Agents von Unangst, Paul C., Capiris, Thomas, Connor, David T., Doubleday, Robert, Heffner, Thomas G., MacKenzie, Robert G., Miller, Steven R., Pugsley, Thomas A., Wise, Lawrence D.

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Hydroxylamine analogs of 2,6 di- t-butylphenols: Dual inhibitors of cyclooxygenase and 5-lipoxygenase or selective 5-lipoxygenase inhibitors von Kramer, James B., Capiris, Thomas, Sircar, Jagadish C., Connor, David T., Bornemeier, Dirk A., Dyer, Richard D., Kuipers, Paul J., Kennedy, John A., Wright, Clifford D., Okonkwo, Godwin C.N., Lesch, Mark E., Schrier, Denis J., Boschelli, Diane H.

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ChemInform Abstract: The Preparation of Optically Active α-Amino 4H-[1,2,4]Oxadiazol-5-ones from Optically Active α-Amino Acids von Mangette, John E., Johnson, Matthew R., Le, Van-Duc, Shenoy, Rajesh A., Roark, Howard, Stier, Michael, Belliotti, Thomas, Capiris, Thomas, Guzzo, Peter R.

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Synthesis of 4-hydroxy-N-[5-(hydroxymethyl)-3-isoxazolyl]-2-methyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide and [(5-methyl-3-isoxazolyl)amino]oxoacetic acid. Major metabolite... von Sircar, Jagadish C., Capiris, Thomas, Bobovski, Thomas P., Schwender, Charles F.

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Thiophene-2-carboxamidotetrazoles and pharmaceutical use thereof von CONNOR, DAVID T, CAPIRIS, THOMAS

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((CYCLO)ALKYL SUBSTITUTED)-GAMMA-AMINOBUTYRIC ACID DERIVATIVES (=GABA ANALOGUES), THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS von HORWELL, DAVID CHRISTOPHER, BELLIOTTI, THOMAS RICHARD, KNEEN, CLARE OCTAVIA, CAPIRIS, THOMAS, BRYANS, JUSTIN STEPHEN, WUSTROW, DAVID JUERGEN

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Pyrazolo[5,1-b]quinazolin-9-ones: a new series of antiallergic agents von Sircar, Jagadish C, Capiris, Thomas, Kesten, Stephen J, Herzig, David J

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4-HYDROXY-N-(5-((SUBSTITUTED HETERO)METHYL)-3- ISOXAZOLYL)-2H- 1,2-BENZOTHIAZINE-3-CARBOXAMIDE, 1, 1-DIOXIDE AND 4-HYDROXY-2-METHYL-N-(5- ((SUBSTITUTED HETERO)METHYL)-3-ISOXAZOLYL)... von SIRCAR, JAGADISH C, CAPIRIS, THOMAS

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