Palladium-Catalyzed Domino Direct Arylation/N-Arylation: Convenient Synthesis of Phenanthridines von Candito, David A, Lautens, Mark

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Development of an Intramolecular Aryne Ene Reaction and Application to the Formal Synthesis of (±)-Crinine von Candito, David A, Dobrovolsky, Dennis, Lautens, Mark

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Formal Synthesis of Nitidine and NK109 via Palladium-Catalyzed Domino Direct Arylation/N-Arylation of Aryl Triflates von Blanchot, Mathieu, Candito, David A, Larnaud, Florent, Lautens, Mark

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Exploiting the Divergent Reactivity of Aryl-Palladium Intermediates for the Rapid Assembly of Fluorene and Phenanthrene Derivatives von Zhao, Ya-Bin, Mariampillai, Brian, Candito, David A, Laleu, Benoît, Li, Mengzhou, Lautens, Mark

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Exploiting the Chemistry of Strained Rings: Synthesis of Indoles via Domino Reaction of Aryl Iodides with 2H-Azirines von Candito, David A, Lautens, Mark

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Palladium-Catalyzed Reductive ortho-Arylation: Evidence for the Decomposition of 1,2-Dimethoxyethane and Subsequent Arylpalladium(II) Reduction von Martins, Andrew, Candito, David A, Lautens, Mark

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Intramolecular Aryne–Ene Reaction: Synthetic and Mechanistic Studies von Candito, David A, Panteleev, Jane, Lautens, Mark

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Lessons from the Synthetic Chemist Nature von Jürjens, Gerrit, Kirschning, Andreas, Candito, David A

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Development of a Flexible and Robust Synthesis of Tetrahydrofuro[3,4‑b]furan Nucleoside Analogues von Candito, David A, Ye, Yingchun, Quiroz, Ryan V, Reutershan, Michael H, Witter, David, Gadamsetty, Surendra B, Li, Hongming, Saurí, Josep, Schneider, Sebastian E, Lam, Yu-hong, Palte, Rachel L

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Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors as Preclinical Immunotherapy Tool Compounds von Vara, Brandon A, Levi, Samuel M, Achab, Abdelghani, Candito, David A, Fradera, Xavier, Lesburg, Charles A, Kawamura, Shuhei, Lacey, Brian M, Lim, Jongwon, Methot, Joey L, Xu, Zangwei, Xu, Haiyan, Smith, Dustin M, Piesvaux, Jennifer A, Miller, J. Richard, Bittinger, Mark, Ranganath, Sheila H, Bennett, David J, DiMauro, Erin F, Pasternak, Alexander

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Exploiting the Chemistry of Strained Rings: Synthesis of Indoles via Domino Reaction of Aryl Iodides with 2 H -Azirines von Candito, David A., Lautens, Mark

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SYNTHESIS OF (S,S)-DIISOPROPYL TARTRATE (E)-CROTYLBORONATE AND ITS REACTION WITH ALDEHYDES: (2R,3R,4R)-1,2-DIDEOXY-2-ETHENYL-4,5-O-(1-METHYLETHYLIDENE)-XYLITOL von Sun, Huikai, Roush, William R, Candito, David A, Blanchot, Mathieu, Lautens, Mark

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Palladium‐Catalyzed Domino Direct Arylation/N‐Arylation: Convenient Synthesis of Phenanthridines von Candito, David A., Lautens, Mark

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Racemic Synthesis of a Key 1,4-Dihydro-2 H -spiro[isoquinoline-3,4′-piperidin]-3′-ol Building Block von Candito, David A., Martinot, Theodore A., Su, Jing, Saurí, Josep, Lam, Yu-hong, Joyce, Leo A., Silverman, Steven M., Sloman, David L., Maddess, Matthew L., Machacek, Michelle R.

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Racemic Synthesis of a Key 1,4-Dihydro‑2H‑spiro[isoquinoline-3,4′-piperidin]-3′-ol Building Block von Candito, David A., Martinot, Theodore A., Su, Jing, Saurí, Josep, Lam, Yu-hong, Joyce, Leo A., Silverman, Steven M., Sloman, David L., Maddess, Matthew L., Machacek, Michelle R.

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Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1‑Heteroaryl‑1H‑Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson’s Disease von Candito, David A., Simov, Vladimir, Gulati, Anmol, Kattar, Solomon, Chau, Ryan W., Lapointe, Blair T., Methot, Joey L., DeMong, Duane E., Graham, Thomas H., Kurukulasuriya, Ravi, Keylor, Mitchell H., Tong, Ling, Morriello, Gregori J., Acton, John J., Pio, Barbara, Liu, Weiguo, Scott, Jack D., Ardolino, Michael J., Martinot, Theodore A., Maddess, Matthew L., Yan, Xin, Gunaydin, Hakan, Palte, Rachel L., McMinn, Spencer E., Nogle, Lisa, Yu, Hongshi, Minnihan, Ellen C., Lesburg, Charles A., Liu, Ping, Su, Jing, Hegde, Laxminarayan G., Moy, Lily Y., Woodhouse, Janice D., Faltus, Robert, Xiong, Tina, Ciaccio, Paul, Piesvaux, Jennifer A., Otte, Karin M., Kennedy, Matthew E., Bennett, David Jonathan, DiMauro, Erin F., Fell, Matthew J., Neelamkavil, Santhosh, Wood, Harold B., Fuller, Peter H., Ellis, J. Michael

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Discovery and Optimization of Potent, Selective, and Brain-Penetrant 1-Heteroaryl-1 H -Indazole LRRK2 Kinase Inhibitors for the Treatment of Parkinson's Disease von Candito, David A, Simov, Vladimir, Gulati, Anmol, Kattar, Solomon, Chau, Ryan W, Lapointe, Blair T, Methot, Joey L, DeMong, Duane E, Graham, Thomas H, Kurukulasuriya, Ravi, Keylor, Mitchell H, Tong, Ling, Morriello, Gregori J, Acton, John J, Pio, Barbara, Liu, Weiguo, Scott, Jack D, Ardolino, Michael J, Martinot, Theodore A, Maddess, Matthew L, Yan, Xin, Gunaydin, Hakan, Palte, Rachel L, McMinn, Spencer E, Nogle, Lisa, Yu, Hongshi, Minnihan, Ellen C, Lesburg, Charles A, Liu, Ping, Su, Jing, Hegde, Laxminarayan G, Moy, Lily Y, Woodhouse, Janice D, Faltus, Robert, Xiong, Tina, Ciaccio, Paul, Piesvaux, Jennifer A, Otte, Karin M, Kennedy, Matthew E, Bennett, David Jonathan, DiMauro, Erin F, Fell, Matthew J, Neelamkavil, Santhosh, Wood, Harold B, Fuller, Peter H, Ellis, J Michael

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ChemInform Abstract: Development of an Intramolecular Aryne Ene Reaction and Application to the Formal Synthesis of (.+-.)-Crinine von Candito, David A., Dobrovolsky, Dennis, Lautens, Mark

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ChemInform Abstract: Intramolecular Aryne-Ene Reaction: Synthetic and Mechanistic Studies von Candito, David A., Panteleev, Jane, Lautens, Mark

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ChemInform Abstract: Stereoselective Nickel-Catalyzed [2 + 2 + 2] Cycloaddition of Enynes and Arynes von Candito, David A., Lautens, Mark

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