INHIBITORS OF (ALPHA-V)(BETA-6) INTEGRIN von Day, Tyler, Dowling, James E, Sosa, Brian, Svensson, Mats A, Troast, Dawn M, Rogers, Bruce N, Qiao, Qi, Bortolato, Andrea, Konze, Kyle D, Harrison, Bryce A, Hickey, Eugene, Lin, Fu-Yang, Bursavich, Matthew M, Kim, Byungchan, Zhong, Cheng, Gerasyuto, Aleksey I, Lippa, Blaise S

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N-benzenesulfonyl substituted anilino-pyrimidine analogs von SUM FUK-WAH,POWELL DENNIS W.,ZHANG YIXIAN,CHEN LIJING,KINCAID SCOTT L.,JENNINGS LEE D.,HU YONGBO,GILBERT ADAM M.,BURSAVICH MATTHEW G

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Designing Non-Peptide Peptidomimetics in the 21st Century:  Inhibitors Targeting Conformational Ensembles von Bursavich, Matthew G, Rich, Daniel H

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Identification and Characterization of Acidic Mammalian Chitinase Inhibitors von Cole, Derek C, Olland, Andrea M, Jacob, Jaison, Brooks, Jon, Bursavich, Matthew G, Czerwinski, Robert, DeClercq, Charlene, Johnson, Mark, Joseph-McCarthy, Diane, Ellingboe, John W, Lin, Laura, Nowak, Pawel, Presman, Ella, Strand, James, Tam, Amy, Williams, Cara M. M, Yao, Shihua, Tsao, Désirée H. H, Fitz, Lori J

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ERK5 Is Required for Tumor Growth and Maintenance Through Regulation of the Extracellular Matrix in Triple Negative Breast Cancer von Van T Hoang, Matossian, Margarite D., Ucar, Deniz A., Elliott, Steven, La, Jacqueline, Wright, Maryl K., Burks, Hope E., Perles, Aaron, Hossain, Fokhrul, King, Connor T., Browning, Valentino E., Bursavich, Jacob, Fang, Fang, Del Valle, Luis, Bhatt, Akshita B., Cavanaugh, Jane E., Flaherty, Patrick T., Anbalagan, Muralidharan, Rowan, Brian G., Bratton, Melyssa R., Nephew, Kenneth P., Miele, Lucio, Collins-Burow, Bridgette M., Martin, Elizabeth C., Burow, Matthew E.

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Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors von Vijay Kumar, D., Hoarau, Christophe, Bursavich, Matthew, Slattum, Paul, Gerrish, David, Yager, Kraig, Saunders, Michael, Shenderovich, Mark, Roth, Bruce L., McKinnon, Rena, Chan, Ashley, Cimbora, Daniel M., Bradford, Chad, Reeves, Leslie, Patton, Scott, Papac, Damon I., Williams, Brandi L., Carlson, Robert O.

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N-((8-Hydroxy-5-substituted-quinolin-7-yl)(phenyl)methyl)-2-phenyloxy/amino-acetamide inhibitors of ADAMTS-5 (Aggrecanase-2) von Gilbert, Adam M., Bursavich, Matthew G., Lombardi, Sabrina, Georgiadis, Katy E., Reifenberg, Erica, Flannery, Carl R., Morris, Elisabeth A.

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5-((1 H-Pyrazol-4-yl)methylene)-2-thioxothiazolidin-4-one inhibitors of ADAMTS-5 von Gilbert, Adam M., Bursavich, Matthew G., Lombardi, Sabrina, Georgiadis, Katy E., Reifenberg, Erica, Flannery, Carl R., Morris, Elisabeth A.

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Novel purine and pyrazolo[3,4- d]pyrimidine inhibitors of PI3 kinase-α: Hit to lead studies von Gilbert, Adam M., Nowak, Pawel, Brooijmans, Natasja, Bursavich, Matthew G., Dehnhardt, Christoph, Santos, Efren Delos, Feldberg, Larry R., Hollander, Irwin, Kim, Stephen, Lombardi, Sabrina, Park, Kaapjoo, Venkatesan, Aranapakam M., Mallon, Robert

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Expedient Parallel Synthesis of 2-Amino-4-heteroarylpyrimidines von Bursavich, Matthew G, Lombardi, Sabrina, Gilbert, Adam M

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5'-Phenyl-3'H-spiro[indoline-3,2'-[1,3,4]thiadiazol]-2-one inhibitors of ADAMTS-5 (aggrecanase-2) von Bursavich, Matthew G, Gilbert, Adam M, Lombardi, Sabrina, Georgiadis, Katy E, Reifenberg, Erica, Flannery, Carl R, Morris, Elisabeth A

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Synthesis and evaluation of aryl thioxothiazolidinone inhibitors of ADAMTS-5 (Aggrecanase-2) von Bursavich, Matthew G., Gilbert, Adam M., Lombardi, Sabrina, Georgiadis, Katy E., Reifenberg, Erica, Flannery, Carl R., Morris, Elisabeth A.

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5′-Phenyl-3′H-spiro[indoline-3,2′-[1,3,4]thiadiazol]-2-one inhibitors of ADAMTS-5 (Aggrecanase-2) von Bursavich, Matthew G., Gilbert, Adam M., Lombardi, Sabrina, Georgiadis, Katy E., Reifenberg, Erica, Flannery, Carl R., Morris, Elisabeth A.

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2-Anilino-4-aryl-1,3-thiazole inhibitors of valosin-containing protein (VCP or p97) von Bursavich, Matthew G., Parker, Daniel P., Willardsen, J. Adam, Gao, Zhong-Hua, Davis, Thaylon, Ostanin, Kirill, Robinson, Rosann, Peterson, Ashley, Cimbora, Daniel M., Zhu, Ju-Fen, Richards, Burt

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3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: Hit to lead studies von Gilbert, Adam M., Bursavich, Matthew G., Lombardi, Sabrina, Adedoyin, Adedayo, Dwyer, Jason M., Hughes, Zoe, Kern, Jeffrey C., Khawaja, Xavier, Rosenzweig-Lipson, Sharon, Moore, William J., Neal, Sarah J., Olsen, Michael, Rizzo, Stacey J. Sukoff, Springer, Dane

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Novel imidazolopyrimidines as dual PI3-Kinase/mTOR inhibitors von Venkatesan, Aranapakam M., Dehnhardt, Christoph M., Chen, Zecheng, Santos, Efren Delos, Dos Santos, Osvaldo, Bursavich, Matthew, Gilbert, Adam M., Ellingboe, John W., Ayral-Kaloustian, Semiramis, Khafizova, Gulnaz, Brooijmans, Natasja, Mallon, Robert, Hollander, Irwin, Feldberg, Larry, Lucas, Judy, Yu, Ker, Gibbons, Jay, Abraham, Robert, Mansour, Tarek S.

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A Fluorescence Polarization Displacement Assay for Aggrecanase-1 and -2 von Cunningham, Kristina M., Bursavich, Matthew, Mackie, Stuart, Krishnamurthy, Girija, Levin, Jeremy

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Novel benzofuran-3-one indole inhibitors of PI3 kinase-a and the mammalian target of rapamycin: Hit to lead studies von Bursavich, Matthew G, Brooijmans, Natasja, Feldberg, Lawrence, Hollander, Irwin, Kim, Stephen, Lombardi, Sabrina, Park, Kaapjoo, Mallon, Robert, Gilbert, Adam M

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Novel purine and pyrazolo[3,4-d]pyrimidine inhibitors of PI3 kinase-a: Hit to lead studies von Gilbert, Adam M, Nowak, Pawel, Brooijmans, Natasja, Bursavich, Matthew G, Dehnhardt, Christoph, Santos, Efren Delos, Feldberg, Larry R, Hollander, Irwin, Kim, Stephen, Lombardi, Sabrina, Park, Kaapjoo, Venkatesan, Aranapakam M, Mallon, Robert

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Hit to lead studies on (hetero)arylpyrimidines - Agonists of the canonical Wnt-b-catenin cellular messaging system von Gilbert, Adam M, Bursavich, Matthew G, Alon, Nippa, Bhat, Bheem M, Bex, Frederick J, Cain, Michael, Coleburn, Valerie, Gironda, Virginia, Green, Paula, Hauze, Diane B, Kharode, Yogendra, Krishnamurthy, Girija, Kirisits, Matthew, Lam, Ho-Sun, Liu, Yao-Bin, Lombardi, Sabrina, Matteo, Jeanne, Murrills, Richard, Robinson, John A, Selim, Sally, Sharp, Michael, Unwalla, Raymond, Varadarajan, Usha, Zhao, Weiguang, Yaworsky, Paul J

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