Direct regulation of CLOCK expression by REV-ERB von Crumbley, Christine, Burris, Thomas P

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REV-ERB agonism improves liver pathology in a mouse model of NASH von Griffett, Kristine, Bedia-Diaz, Gonzalo, Elgendy, Bahaa, Burris, Thomas P

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Nuclear Receptor Subfamily 1 Group D Member 1 Regulates Circadian Activity of NLRP3 Inflammasome to Reduce the Severity of Fulminant Hepatitis in Mice von Pourcet, Benoit, Zecchin, Mathilde, Ferri, Lise, Beauchamp, Justine, Sitaula, Sadicha, Billon, Cyrielle, Delhaye, Stéphane, Vanhoutte, Jonathan, Mayeuf-Louchart, Alicia, Thorel, Quentin, Haas, Joel T., Eeckhoute, Jérome, Dombrowicz, David, Duhem, Christian, Boulinguiez, Alexis, Lancel, Steve, Sebti, Yasmine, Burris, Thomas P., Staels, Bart, Duez, Hélène M.

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Small Molecule Modulation of Nuclear Receptor Conformational Dynamics: Implications for Function and Drug Discovery von Kojetin, Douglas J., Burris, Thomas P.

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Promiscuous activity of the LXR antagonist GSK2033 in a mouse model of fatty liver disease von Griffett, Kristine, Burris, Thomas P.

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DNA binding alters coactivator interaction surfaces of the intact VDR–RXR complex von Zhang, Jun, Chalmers, Michael J, Stayrook, Keith R, Burris, Lorri L, Wang, Yongjun, Busby, Scott A, Pascal, Bruce D, Garcia-Ordonez, Ruben D, Bruning, John B, Istrate, Monica A, Kojetin, Douglas J, Dodge, Jeffrey A, Burris, Thomas P, Griffin, Patrick R

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Broad Anti-tumor Activity of a Small Molecule that Selectively Targets the Warburg Effect and Lipogenesis von Flaveny, Colin A., Griffett, Kristine, El-Gendy, Bahaa El-Dien M., Kazantzis, Melissa, Sengupta, Monideepa, Amelio, Antonio L., Chatterjee, Arindam, Walker, John, Solt, Laura A., Kamenecka, Theodore M., Burris, Thomas P.

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International Union of Basic and Clinical Pharmacology. XC. multisite pharmacology: recommendations for the nomenclature of receptor allosterism and allosteric ligands von Christopoulos, Arthur, Changeux, Jean-Pierre, Catterall, William A, Fabbro, Doriano, Burris, Thomas P, Cidlowski, John A, Olsen, Richard W, Peters, John A, Neubig, Richard R, Pin, Jean-Philippe, Sexton, Patrick M, Kenakin, Terry P, Ehlert, Frederick J, Spedding, Michael, Langmead, Christopher J

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Structural basis of synthetic agonist activation of the nuclear receptor REV-ERB von Murray, Meghan H., Valfort, Aurore Cecile, Koelblen, Thomas, Ronin, Céline, Ciesielski, Fabrice, Chatterjee, Arindam, Veerakanellore, Giri Babu, Elgendy, Bahaa, Walker, John K., Hegazy, Lamees, Burris, Thomas P.

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Suppression of atherosclerosis by synthetic REV-ERB agonist von Sitaula, Sadichha, Billon, Cyrielle, Kamenecka, Theodore M., Solt, Laura A., Burris, Thomas P.

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Development of LXR inverse agonists to treat MAFLD, NASH, and other metabolic diseases von Griffett, Kristine, Burris, Thomas P

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Recent Advances in the Medicinal Chemistry of Liver X Receptors von El-Gendy, Bahaa El-Dien M, Goher, Shaimaa S, Hegazy, Lamees S, Arief, Mohamed M H, Burris, Thomas P

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Rev-erbα heterozygosity produces a dose-dependent phenotypic advantage in mice von Welch, Ryan D, Billon, Cyrielle, Kameric, Amina, Burris, Thomas P, Flaveny, Colin A

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Disrupting the key circadian regulator CLOCK leads to age-dependent cardiovascular disease von Alibhai, Faisal J, LaMarre, Jonathan, Reitz, Cristine J, Tsimakouridze, Elena V, Kroetsch, Jeffrey T, Bolz, Steffen-Sebastian, Shulman, Alex, Steinberg, Samantha, Burris, Thomas P, Oudit, Gavin Y, Martino, Tami A

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Distinct roles for REV-ERBα and REV-ERBβ in oxidative capacity and mitochondrial biogenesis in skeletal muscle von Amador, Ariadna, Campbell, Sean, Kazantzis, Melissa, Lan, Gary, Burris, Thomas P, Solt, Laura A

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Pharmacological and Genetic Modulation of REV-ERB Activity and Expression Affects Orexigenic Gene Expression von Amador, Ariadna, Wang, Yongjun, Banerjee, Subhashis, Kameneka, Theodore M, Solt, Laura A, Burris, Thomas P

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Regulation of p53 stability and apoptosis by a ROR agonist von Wang, Yongjun, Solt, Laura A, Kojetin, Douglas J, Burris, Thomas P

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A two-hit model of alcoholic liver disease that exhibits rapid, severe fibrosis von Sengupta, Monideepa, Abuirqeba, Suomia, Kameric, Amina, Cecile-Valfort, Aurore, Chatterjee, Arindam, Griffett, Kristine, Burris, Thomas P, Flaveny, Colin A

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Restoration of the molecular clock is tumor suppressive in neuroblastoma von Moreno-Smith, Myrthala, Milazzo, Giorgio, Tao, Ling, Fekry, Baharan, Zhu, Bokai, Mohammad, Mahmoud A., Di Giacomo, Simone, Borkar, Roshan, Reddy, Karthik Reddy Kami, Capasso, Mario, Vasudevan, Sanjeev A., Sumazin, Pavel, Hicks, John, Putluri, Nagireddy, Perini, Giovanni, Eckel-Mahan, Kristin, Burris, Thomas P., Barbieri, Eveline

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Identification of SR8278, a Synthetic Antagonist of the Nuclear Heme Receptor REV-ERB von Kojetin, Douglas, Wang, Yongjun, Kamenecka, Theodore M, Burris, Thomas P

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