The azaindole framework in the design of kinase inhibitors von Mérour, Jean-Yves, Buron, Frédéric, Plé, Karen, Bonnet, Pascal, Routier, Sylvain

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Access and Modulation of Substituted Pyrrolo[3,4- c ]pyrazole-4,6-(2 H ,5 H )-diones von Ejjoummany, Abdelaziz, Elie, Jonathan, El Hakmaoui, Ahmed, Akssira, Mohamed, Routier, Sylvain, Buron, Frédéric

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Glycosaminoglycan Mimetics Obtained by Microwave-Assisted Sulfation of Marine Bacterium Sourced Infernan Exopolysaccharide von Colliec-Jouault, Sylvia, Esposito, Fabiana, Ledru, Hélène, Sinquin, Corinne, Marchand, Laetitia, Fillaudeau, Arnaud, Routier, Sylvain, Buron, Frédéric, Lopin-Bon, Chrystel, Cuenot, Stéphane, Bedini, Emiliano, Zykwinska, Agata

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Design, Synthesis, and Biological Activity of Pyridopyrimidine Scaffolds as Novel PI3K/mTOR Dual Inhibitors von Saurat, Thibault, Buron, Frédéric, Rodrigues, Nuno, de Tauzia, Marie-Ludivine, Colliandre, Lionel, Bourg, Stéphane, Bonnet, Pascal, Guillaumet, Gérald, Akssira, Mohamed, Corlu, Anne, Guillouzo, Christiane, Berthier, Pauline, Rio, Pascale, Jourdan, Marie-Lise, Bénédetti, Hélène, Routier, Sylvain

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Synthesis of γ-carboline N-oxide under gold(I)-catalysis and C-1 amino and fluoro γ-carboline von Agnieszka, Zak, Hamid, Marzag, Nuno, Rodrigues, Johnny, Vercouillie, Sylvie, Chalon, Frédéric, Buron, Sylvain, Routier

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Numerical modeling and evaluation of solid-liquid extraction with pressurized hot water extraction applied to Robinia Pseudoacacia wood von Sangaré, Diakaridia, Caré, Flore, Buron, Frédéric, Lafite, Pierre, Bostyn, Stéphane

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Synthesis of [1,3,4]Thiadiazolo[3′,2′:1,2]imidazo[4,5‑c]quinolines including Pictet–Spengler Reaction and Exploration of Their C‑2 Reactivity through SNAr von Place, Matthieu, Copin, Chloé, Apotrosoaei, Maria, Constantin, Sandra, Vasincu, Ioana Mirela, Profire, Lenuta, Buron, Frédéric, Routier, Sylvain

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Access to Mono‐, Di‐ and Tri‐(Het)Arylated Pyrazolo[5,1‐b]oxazoles Using Cyclization, C−H Activation and Suzuki–Miyaura Palladium‐Catalyzed Reactions von Michel, Marion, Caré, Flore, Bourg, Stéphane, Bostyn, Stéphane, Lafite, Pierre, Routier, Sylvain, Buron, Frédéric

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Synthesis of novel series of 3,5-disubstituted imidazo[1,2-d] [1,2,4]thiadiazoles involving SNAr and Suzuki–Miyaura cross-coupling reactions von Pescheteau, Clémentine, Place, Matthieu, Sava, Alexandru, Nunes, Lea, Profire, Lenuta, Routier, Sylvain, Buron, Frédéric

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Palladium-Catalyzed Amination of C-5 Bromoimidazo[2,1-b]­[1,3,4]­thiadiazoles von Copin, Chloé, Buron, Frédéric, Routier, Sylvain

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Design and biological evaluation of substituted 5,7-dihydro-6H-indolo[2,3-c]quinolin-6-one as novel selective Haspin inhibitors von Avula, Sreenivas, Peng, Xudan, Lang, Xingfen, Tortorella, Micky, Josselin, Béatrice, Bach, Stéphane, Bourg, Stephane, Bonnet, Pascal, Buron, Frédéric, Ruchaud, Sandrine, Routier, Sylvain, Neagoie, Cleopatra

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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3 von Oukoloff, Killian, Coquelle, Nicolas, Bartolini, Manuela, Naldi, Marina, Le Guevel, Rémy, Bach, Stéphane, Josselin, Béatrice, Ruchaud, Sandrine, Catto, Marco, Pisani, Leonardo, Denora, Nunzio, Iacobazzi, Rosa Maria, Silman, Israel, Sussman, Joel L., Buron, Frédéric, Colletier, Jacques-Philippe, Jean, Ludovic, Routier, Sylvain, Renard, Pierre-Yves

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Stereoselective Synthesis of Iminosugar‐ C ‐Glycosides through Addition of Organometallic Reagents to N ‐ tert ‐Butanesulfinyl Glycosylamines: A Comprehensive Study von Kamzol, Daniel, Neuville, Maxime, Cocaud, Chloé, Tiger, Killian, Taffoureau, Baptiste, Lewiński, Krzysztof, Jaszczyk, Justyna, Martin, Olivier R., Baś, Sebastian, Routier, Sylvain, Gillaizeau, Isabelle, Buron, Frédéric, Nicolas, Cyril

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Pyridine-Based Lanthanide Complexes Combining MRI and NIR Luminescence Activities von Bonnet, Célia S., Buron, Frédéric, Caillé, Fabien, Shade, Chad M., Drahoš, Bohuslav, Pellegatti, Laurent, Zhang, Jian, Villette, Sandrine, Helm, Lothar, Pichon, Chantal, Suzenet, Franck, Petoud, Stéphane, Tóth, Éva

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Efficient Transposition of the Sandmeyer Reaction from Batch to Continuous Process von D’Attoma, Joseph, Camara, Titi, Brun, Pierre Louis, Robin, Yves, Bostyn, Stéphane, Buron, Frédéric, Routier, Sylvain

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Design of selective COX-2 inhibitors in the (aza)indazole series. Chemistry, in vitro studies, radiochemistry and evaluations in rats of a [18F] PET tracer von Elie, Jonathan, Vercouillie, Johnny, Arlicot, Nicolas, Lemaire, Lucas, Bidault, Rudy, Bodard, Sylvie, Hosselet, Christel, Deloye, Jean-Bernard, Chalon, Sylvie, Emond, Patrick, Guilloteau, Denis, Buron, Frédéric, Routier, Sylvain

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Selection of Bis-Indolyl Pyridines and Triphenylamines as New Inhibitors of SARS-CoV-2 Cellular Entry by Modulating the Spike Protein/ACE2 Interfaces von Lapaillerie, Delphine, Charlier, Cathy, Guyonnet-Dupérat, Véronique, Murigneux, Emilie, Fernandes, Henrique S, Martins, Fábio G, Magalhães, Rita P, Vieira, Tatiana F, Richetta, Clémence, Subra, Frédéric, Lebourgeois, Samuel, Charpentier, Charlotte, Descamps, Diane, Visseaux, Benoît, Weigel, Pierre, Favereaux, Alexandre, Beauvineau, Claire, Buron, Frédéric, Teulade-Fichou, Marie-Paule, Routier, Sylvain, Gallois-Montbrun, Sarah, Meertens, Laurent, Delelis, Olivier, Sousa, Sérgio F, Parissi, Vincent

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Aminations and arylations by direct C-O activation for the design of 7,8-dihydro-6H-5,8-ethanopyrido[3,2-d]pyrimidines von Laurent, Mazarine, Bostyn, Stephane, Marchivie, Mathieu, Robin, Yves, Routier, Sylvain, Buron, Frederic

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Isoquinoline-Based Lanthanide Complexes: Bright NIR Optical Probes and Efficient MRI Agents von Caillé, Fabien, Bonnet, Célia S, Buron, Frédéric, Villette, Sandrine, Helm, Lothar, Petoud, Stéphane, Suzenet, Franck, Tóth, Éva

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Neuroprotective effect of the alpha 7 nicotinic receptor agonist PHA 543613 in an in vivo excitotoxic adult rat model von Foucault-Fruchard, Laura, Doméné, Aurélie, Page, Guylène, Windsor, Marguerite, Emond, Patrick, Rodrigues, Nuno, Dollé, Frédéric, Damont, Annelaure, Buron, Frédéric, Routier, Sylvain, Chalon, Sylvie, Antier, Daniel

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