Enantiomers of Diastereomeric cis-N-[1-(2-Hydroxy-2-phenylethyl)-3-methyl-4-piperidyl]-N-phenylpropanamides: Synthesis, X-ray Analysis, and Biological Activities von Brine, George A, Stark, Peter A, Liu, Young, Carroll, F. Ivy, Singh, P, Xu, Heng, Rothman, Richard B

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Synthesis of N 6 -[endo-2′-(endo-5′-Hydroxy)norbornyl]-8-(N-methylisopropylamino)-9-methyladenine (WRC-0571): A Potent and Selective Adenosine A1 Receptor Antagonist von Jin, Chunyang, Burgess, Jason P., Rehder, Kenneth S., Brine, George A.

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Enantiomers of Diastereoisomeric cis-N-[1-(2-Hydroxy-2-phenylethyl)-3-methyl-4-piperidyl]-N-phenylpropanamides:  Synthesis, X-ray Analysis, and Biological Activities von Brine, George A, Stark, Peter A, Liu, Young, Carroll, F. Ivy, Singh, P, Xu, Heng, Rothman, Richard B

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Opioid Agonist Effects on Mouse Writhing After Irreversible Mu Receptor Blockade With Clocinnamox von Zernig, Gerald, Broadbear, Jillian, Lewis, John W, Brine, George A, Woods, James H

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p-hydroxymethadone : synthesis, crystal structure and CD properties von BRINE, G. A, BOLDT, K. G, PRAKASH, D, KOTCHMAR, D. J, BONDESON, V. C, BRADLEY, D. J, SINGH, P, IVY CARROLL, F

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Opioid peptide receptor studies. 7. The methylfentanyl congener RTI-4614-4 and its four enantiomers bind to different domains of the rat ? opioid receptor von Lu, Yi-Feng, Xu, Heng, Liu-Chen, Lee-Yuan, Chen, Chongguang, Partilla, John S., Brine, George A., Carroll, F. Ivy, Rice, Kenner C., Lai, Josephine, Porreca, Frank, Sadee, Wolfgang, Rothman, Richard B.

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Chemical synthesis and structural elucidation of a new serotonin metabolite: (4 R)-2-[(5′-hydroxy-1′ H-indol-3′-yl)methyl]thiazolidine-4-carboxylic acid von Jin, Chunyang, Burgess, Jason P., Gopinathan, Madathil B., Brine, George A.

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X-ray structures of the ? opioid antagonist TIPP and a protected derivative of the ? opioid antagonist ICI 174,864 von Flippen-Anderson, Judith L., George, Clifford, Deschamps, Jeffrey R., Reddy, P. Anantha, Lewin, Anita H., Brine, George A.

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Carbon-13 nuclear magnetic resonance spectra of morphine alkaloids von Carroll, Frank I, Moreland, Charles G, Brine, George A, Kepler, John A

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Opioid peptide receptor studies, 11: Involvement of Tyr148, Trp318 and His319 of the rat μ-opioid receptor in binding of μ-selective ligands von Xu, Heng, Lu, Yi-Feng, Partilla, John S., Zheng, Qiao-Xi, Wang, Jia-Bei, Brine, George A., Carroll, F. Ivy, Rice, Kenner C., Chen, Kai-Xian, Chi, Zhi-Qiang, Rothman, Richard B.

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Synthesis of Morphine-3,6-di-β-D-glucuronide von Berrang, Bertold, Brine, George A., Carroll, F. Ivy

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Receptor reserve and affinity of mu opioid agonists in mouse antinociception: correlation with receptor binding von Zernig, Gerald, Issaevitch, Tom, Broadbear, Jillian H., Burke, Timothy F., Lewis, John W., Brine, George A., Woods, James H.

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Phencyclidine metabolism: resolution, structure, and biological activity of the isomers of the hydroxymetabolite, 4-phenyl-4-(1-piperidinyl)cyclohexanol von Carroll, F. Ivy, Brine, George A, Boldt, Karl G, Cone, Edward J, Yousefnejad, David, Vaupel, D. Bruce, Buchwald, William F

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Formamidinesulfinic acid reduction of dihydrocodeinone derivatives von Brine, George A, Boldt, Karl G, Coleman, Michael L, Bradley, David J, Carroll, F. Ivy

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Isolation, structure, and biological activity of several metabolites of .DELTA.9/tetrahydrocannabinol von Wall, Monroe E, Brine, Dolores R, Brine, George A, Pitt, Colin G, Freudenthal, Ralph I, Christensen, H. Dix

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Ring C conformation of 6.beta.-naltrexol and 6.alpha.-naltrexol. Evidence from proton and carbon-13 nuclear magnetic resonance von Brine, George A, Prakash, Doriswamy, Hart, Carolyn King, Kotchmar, Dennis J, Moreland, Charles G, Carroll, Frank I

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Opioid peptide receptor studies. 7. The methylfentanyl congener RTI-4614-4 and its four enantiomers bind to different domains of the rat μ opioid receptor von Lu, Yi-Feng, Xu, Heng, Liu-Chen, Lee-Yuan, Chen, Chongguang, Partilla, John S., Brine, George A., Carroll, F. Ivy, Rice, Kenner C., Lai, Josephine, Porreca, Frank, Sadee, Wolfgang, Rothman, Richard B.

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RTI-4614-4: An analog of (+)-cis-3-methylfentanyl with a 27,000-fold binding selectivity for mu versus delta opioid binding sites von Rothman, Richard B., Heng Xu, Seggel, Mark, Jacobson, Arthur E., Rice, Kenner C., Brine, George A., Carroll, F.Ivy

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Opioid peptide receptor studies, 11: Involvement of Tyr148, Trp318 and His319 of the rat ?-opioid receptor in binding of ?-selective ligands von Xu, Heng, Lu, Yi-Feng, Partilla, John S., Zheng, Qiao-Xi, Wang, Jia-Bei, Brine, George A., Carroll, F. Ivy, Rice, Kenner C., Chen, Kai-Xian, Chi, Zhi-Qiang, Rothman, Richard B.

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AN EFFICIENT SYNTHESIS OF DAGO von Reddy, P. Anantha, Hayes, James P., Lewin, Anita H., Brine, George A.

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