Discovery, Modeling, and Human Pharmacokinetics of N-(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ETA... von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Bui, Huong, You, Tony J., Wang, Junmei, Bourgoyne, Andree R., Knowles, Vippra, Berens, Kurt L., Holland, George W., Brock, Tommy A., Dixon, Richard A. F.

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Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides:  TBC3214, an ETA Selective Endothelin Antagonist von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Li, Jian, Bourgoyne, Andree R, Bui, Huong, Keller, Karin M, Knowles, Vippra, Li, Wen, Stavros, Fiona D, Holland, George W, Brock, Tommy A, Dixon, Richard A. F

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Endothelin Antagonists:  Substituted Mesitylcarboxamides with High Potency and Selectivity for ETA Receptors von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Bui, Huong, Chen, Qi, Raju, B, Bourgoyne, Andree R, Knowles, Vippra, Biediger, Ronald J, Market, Robert V, Lin, Shuqun, Dupré, Brian, Kogan, Timothy P, Holland, George W, Brock, Tommy A, Dixon, Richard A. F

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Discovery, Modeling, and Human Pharmacokinetics of N -(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ET... von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Bui, Huong, You, Tony J., Wang, Junmei, Bourgoyne, Andree R., Knowles, Vippra, Berens, Kurt L., Holland, George W., Brock, Tommy A., Dixon, Richard A. F.

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Discovery, modeling, and human pharmacokinetics of N-(2-acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)-thiophene -2-carboxamide (TBC3711), a second generation, E... von WU, Chengde, DECKER, E. Radford, BROCK, Tommy A, DIXON, Richard A. F, BLOK, Natalie, HUONG BUI, YOU, Tony J, JUNMEI WANG, BOURGOYNE, Andree R, KNOWLES, Vippra, BERENS, Kurt L, HOLLAND, George W

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Endothelin antagonists: substituted mesitylcarboxamides with high potency and selectivity for ET(A) receptors von Wu, C, Decker, E R, Blok, N, Bui, H, Chen, Q, Raju, B, Bourgoyne, A R, Knowles, V, Biediger, R J, Market, R V, Lin, S, Dupré, B, Kogan, T P, Holland, G W, Brock, T A, Dixon, R A

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Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides:  TBC3214, an ET A Selective Endothelin Antagonist von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Li, Jian, Bourgoyne, Andree R., Bui, Huong, Keller, Karin M., Knowles, Vippra, Li, Wen, Stavros, Fiona D., Holland, George W., Brock, Tommy A., Dixon, Richard A. F.

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