Cobalt–Chromium Dental Alloys: Metal Exposures, Toxicological Risks, CMR Classification, and EU Regulatory Framework von Vaicelyte, Alina, Janssen, Christine, Le Borgne, Marc, Grosgogeat, Brigitte

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Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles von Kita, Diogo Henrique, Guragossian, Nathalie, Zattoni, Ingrid Fatima, Moure, Vivian Rotuno, Rego, Fabiane Gomes de Moraes, Lusvarghi, Sabrina, Moulenat, Thomas, Belhani, Billel, Picheth, Geraldo, Bouacida, Sofiane, Bouaziz, Zouhair, Marminon, Christelle, Berredjem, Malika, Jose, Joachim, Gonçalves, Marcos Brown, Ambudkar, Suresh V., Valdameri, Glaucio, Le Borgne, Marc

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Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors von Kufareva, Irina, Bestgen, Benoit, Brear, Paul, Prudent, Renaud, Laudet, Béatrice, Moucadel, Virginie, Ettaoussi, Mohamed, Sautel, Celine F., Krimm, Isabelle, Engel, Matthias, Filhol, Odile, Borgne, Marc Le, Lomberget, Thierry, Cochet, Claude, Abagyan, Ruben

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Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production von Bayart, Caroline, Mularoni, Angélique, Hemmani, Nada, Kerachni, Soumeya, Jose, Joachim, Gouet, Patrice, Paladino, Joseph, Le Borgne, Marc

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QSAR Model of Indeno[1,2- b ]indole Derivatives and Identification of N -isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3- b ]furan-3-carboxamide as a Potent CK2 Inhibitor von Haidar, Samer, Marminon, Christelle, Aichele, Dagmar, Nacereddine, Abdelhamid, Zeinyeh, Wael, Bouzina, Abdeslem, Berredjem, Malika, Ettouati, Laurent, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim

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Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols von Lebouvier, Nicolas, Pagniez, Fabrice, Na, Young Min, Shi, Da, Pinson, Patricia, Marchivie, Mathieu, Guillon, Jean, Hakki, Tarek, Bernhardt, Rita, Yee, Sook Wah, Simons, Claire, Lézé, Marie-Pierre, Hartmann, Rolf W, Mularoni, Angélique, Le Baut, Guillaume, Krimm, Isabelle, Abagyan, Ruben, Le Pape, Patrice, Le Borgne, Marc

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Occurrence of the Synthetic Analgesic Tramadol in an African Medicinal Plant von Boumendjel, Ahcène, Sotoing Taïwe, Germain, Ngo Bum, Elisabeth, Chabrol, Tanguy, Beney, Chantal, Sinniger, Valérie, Haudecoeur, Romain, Marcourt, Laurence, Challal, Soura, Ferreira Queiroz, Emerson, Souard, Florence, Le Borgne, Marc, Lomberget, Thierry, Depaulis, Antoine, Lavaud, Catherine, Robins, Richard, Wolfender, Jean-Luc, Bonaz, Bruno, De Waard, Michel

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Toxicological Risks of the Cobalt–Chromium Alloys in Dentistry: A Systematic Review von Grosgogeat, Brigitte, Vaicelyte, Alina, Gauthier, Rémy, Janssen, Christine, Le Borgne, Marc

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4-Pyridinio-1,4-Dihydropyridines as Calcium Ion Transport Modulators: Antagonist, Agonist, and Dual Action von Duburs, Gunars, Velena, Astrida, Bisenieks, Egils, Bruvere, Imanta, Vilskersts, Reinis, Kanepe-Lapsa, Iveta, Domracheva, Ilona, Turovska, Baiba

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Carbazole scaffolds in cancer therapy: a review from 2012 to 2018 von Issa, Samar, Prandina, Anthony, Bedel, Nicolas, Rongved, Pål, Yous, Saïd, Le Borgne, Marc, Bouaziz, Zouhair

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Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2 von Alchab, Faten, Ettouati, Laurent, Bouaziz, Zouhair, Bollacke, Andre, Delcros, Jean-Guy, Gertzen, Christoph G W, Gohlke, Holger, Pinaud, Noël, Marchivie, Mathieu, Guillon, Jean, Fenet, Bernard, Jose, Joachim, Borgne, Marc Le

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Behaviour of Tetrabenazine in Acid Medium: Reassessment and Impact on Formulation von Ettouati, Laurent, Senta-Loys, Zoé, Bourgeois, Sandrine, Fenet, Bernard, Borgne, Marc Le, Fessi, Hatem

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Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity von Gozzi, Gustavo Jabor, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Honorat, Mylène, Guragossian, Nathalie, Marminon, Christelle, Valdameri, Glaucio, Bollacke, Andre, Guillon, Jean, Pinaud, Noël, Marchivie, Mathieu, Cadena, Silvia M, Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio

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Biological exploration of a novel 1,2,4-triazole-indole hybrid molecule as antifungal agent von Pagniez, Fabrice, Lebouvier, Nicolas, Na, Young Min, Ourliac-Garnier, Isabelle, Picot, Carine, Le Borgne, Marc, Le Pape, Patrice

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Solubility enhancement of mefenamic acid by inclusion complex with β-cyclodextrin: in silico modelling, formulation, characterisation, and in vitro studies von Sid, Dounia, Baitiche, Milad, Elbahri, Zineb, Djerboua, Ferhat, Boutahala, Mokhtar, Bouaziz, Zouhair, Le Borgne, Marc

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1st Joint European Conference on Therapeutic Targets and Medicinal Chemistry (TTMC 2015) von Le Borgne, Marc, Haidar, Samer, Duval, Olivier, Wünsch, Bernhard, Jose, Joachim

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Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2 von Bouzina, Abdeslem, Berredjem, Malika, Bouacida, Sofiane, Bachari, Khaldoun, Marminon, Christelle, Borgne, Marc Le, Bouaziz, Zouhair, Bouone, Yousra Ouafa

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The combined use of analytical tools for exploring tetanus toxin and tetanus toxoid structures von Bayart, Caroline, Peronin, Sébastien, Jean, Elisa, Paladino, Joseph, Talaga, Philippe, Borgne, Marc Le

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Toward selective CK2alpha and CK2alpha’ inhibitors: Development of a novel whole-cell kinase assay by Autodisplay of catalytic CK2alpha von Bollacke, Andre, Nienberg, Christian, Borgne, Marc Le, Jose, Joachim

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1D NMR WaterLOGSY as an efficient method for fragment-based lead discovery von Raingeval, Claire, Cala, Olivier, Brion, Béatrice, Le Borgne, Marc, Hubbard, Roderick Eliot, Krimm, Isabelle

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