Discovery and Pharmacokinetic and Pharmacological Properties of the Potent and Selective MET Kinase Inhibitor 1‑{6-[6-(4-Fluorophenyl)-[1,2,4]triazolo[4,3‑b]pyridazin-3-ylsulfanyl]... von Ugolini, Antonio, Kenigsberg, Mireille, Rak, Alexey, Vallée, Francois, Houtmann, Jacques, Lowinski, Maryse, Capdevila, Cécile, Khider, Jean, Albert, Eva, Martinet, Nathalie, Nemecek, Conception, Grapinet, Sandrine, Bacqué, Eric, Roesner, Manfred, Delaisi, Christine, Calvet, Loreley, Bonche, Fabrice, Semiond, Dorothée, Egile, Coumaran, Goulaouic, Hélène, Schio, Laurent

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Fatty acid acylated peptide therapeutics: discovery of omega-n oxidation of the lipid chain as a novel metabolic pathway in preclinical species von Esposito, Simone, Krick, Alain, Pasquier, Olivier, Bonche, Fabrice, Ingenito, Raffaele, Magotti, Paola, Bianchi, Elisabetta, Monteagudo, Edith, Gallo, Mariana, Cicero, Daniel Oscar, Orsatti, Laura, Veneziano, Maria, Caretti, Fulvia, Mele, Riccardo, Roversi, Daniela, Gennari, Nadia, Brasseur, Denis, Gauzy-Lazo, Laurence, Duclos, Olivier, Mauriac, Christine, Illiano, Stephane, Mallart, Sergio

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Mobilise-D insights to estimate real-world walking speed in multiple conditions with a wearable device von Kirk, Cameron, Küderle, Arne, Micó-Amigo, M. Encarna, Bonci, Tecla, Paraschiv-Ionescu, Anisoara, Ullrich, Martin, Soltani, Abolfazl, Gazit, Eran, Salis, Francesca, Alcock, Lisa, Aminian, Kamiar, Becker, Clemens, Bertuletti, Stefano, Brown, Philip, Buckley, Ellen, Cantu, Alma, Carsin, Anne-Elie, Caruso, Marco, Caulfield, Brian, Cereatti, Andrea, Chiari, Lorenzo, D’Ascanio, Ilaria, Garcia-Aymerich, Judith, Hansen, Clint, Hausdorff, Jeffrey M., Hiden, Hugo, Hume, Emily, Keogh, Alison, Kluge, Felix, Koch, Sarah, Maetzler, Walter, Megaritis, Dimitrios, Mueller, Arne, Niessen, Martijn, Palmerini, Luca, Schwickert, Lars, Scott, Kirsty, Sharrack, Basil, Sillén, Henrik, Singleton, David, Vereijken, Beatrix, Vogiatzis, Ioannis, Yarnall, Alison J., Rochester, Lynn, Mazzà, Claudia, Eskofier, Bjoern M., Del Din, Silvia

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Author Correction: Mobilise-D insights to estimate real-world walking speed in multiple conditions with a wearable device von Kirk, Cameron, Küderle, Arne, Micó-Amigo, M. Encarna, Bonci, Tecla, Paraschiv-Ionescu, Anisoara, Ullrich, Martin, Soltani, Abolfazl, Gazit, Eran, Salis, Francesca, Alcock, Lisa, Aminian, Kamiar, Becker, Clemens, Bertuletti, Stefano, Brown, Philip, Buckley, Ellen, Cantu, Alma, Carsin, Anne-Elie, Caruso, Marco, Caulfield, Brian, Cereatti, Andrea, Chiari, Lorenzo, D’Ascanio, Ilaria, Garcia-Aymerich, Judith, Hansen, Clint, Hausdorff, Jeffrey M., Hiden, Hugo, Hume, Emily, Keogh, Alison, Kluge, Felix, Koch, Sarah, Maetzler, Walter, Megaritis, Dimitrios, Mueller, Arne, Niessen, Martijn, Palmerini, Luca, Schwickert, Lars, Scott, Kirsty, Sharrack, Basil, Sillén, Henrik, Singleton, David, Vereijken, Beatrix, Vogiatzis, Ioannis, Yarnall, Alison J., Rochester, Lynn, Mazzà, Claudia, Eskofier, Bjoern M., Del Din, Silvia

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The selective intravenous inhibitor of the MET tyrosine kinase SAR125844 inhibits tumor growth in MET-amplified cancer von Egile, Coumaran, Kenigsberg, Mireille, Delaisi, Christine, Bégassat, Françoise, Do-Vale, Véronique, Mestadier, Jessica, Bonche, Fabrice, Bénard, Tsiala, Nicolas, Jean-Paul, Valence, Sandrine, Lefranc, Céline, Francesconi, Elisa, Castell, Christelle, Lefebvre, Anne-Marie, Nemecek, Conception, Calvet, Loreley, Goulaouic, Hélène

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Abstract 845: In vitro and in vivo pharmacology of SAR125844, a potent and selective intravenous MET kinase inhibitor undergoing Phase I clinical trial von Goulaouic, Hélène, Kenigsberg, Mireille, Delaisi, Christine, Begassat, Françoise, Do-Vale, Véronique, Mestadier, Jessica, Bonche, Fabrice, Bénard, Tsiala, Nicolas, Jean-Paul, Calvet, Loreley, Egile, Coumaran, Nemecek, Conception, Lengauer, Christoph

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Abstract 2911: SAR125844: a potent and selective ATP-competitive inhibitor of MET kinase von Schio, Laurent, Nemecek, Conception, Ugolini, Antonio, Wentzler, Sylvie, Grapinet, Sandrine, Khider, Jean, Albert, Eva, Dischamps, Nathalie, Gay, Frédéric, Sonnefraud, Véronique, Bacqué, Eric, Kenigsberg, Mireille, Goulaouic, Hélène, Dagallier, Anne, Vallée, François, Bonche, Fabrice, Lengauer, Christoph

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