Synthesis, Identification, and Structure–Activity Relationship Analysis of GATA4 and NKX2‑5 Protein–Protein Interaction Modulators von Jumppanen, Mikael, Kinnunen, Sini M, Välimäki, Mika J, Talman, Virpi, Auno, Samuli, Bruun, Tanja, Boije af Gennäs, Gustav, Xhaard, Henri, Aumüller, Ingo B, Ruskoaho, Heikki, Yli-Kauhaluoma, Jari

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Total Synthesis of Bistramide A and Its 36(Z) Isomers: Differential Effect on Cell Division, Differentiation, and Apoptosis von Tomas, Loïc, Boije af Gennäs, Gustav, Hiebel, Marie Aude, Hampson, Peter, Gueyrard, David, Pelotier, Béatrice, Yli-Kauhaluoma, Jari, Piva, Olivier, Lord, Janet M., Goekjian, Peter G.

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Acetylcholinesterase inhibitory guided fractionation of Melissa officinalis L von Dastmalchi, Keyvan, Ollilainen, Velimatti, Lackman, Petri, Gennäs, Gustav Boije af, Dorman, H.J. Damien, Järvinen, Päivi P., Yli-Kauhaluoma, Jari, Hiltunen, Raimo

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Chemical analysis using 3D printed glass microfluidics von Gal-Or, Eran, Gershoni, Yaniv, Scotti, Gianmario, Nilsson, Sofia M. E, Saarinen, Jukka, Jokinen, Ville, Strachan, Clare J, Boije af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Kotiaho, Tapio

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Structural Isosteres of Phosphate Groups in the Protein Data Bank von Zhang, Yuezhou, Borrel, Alexandre, Ghemtio, Leo, Regad, Leslie, Boije af Gennäs, Gustav, Camproux, Anne-Claude, Yli-Kauhaluoma, Jari, Xhaard, Henri

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Scaffold hopping from (5-hydroxymethyl) isophthalates to multisubstituted pyrimidines diminishes binding affinity to the C1 domain of protein kinase C von Provenzani, Riccardo, Tarvainen, Ilari, Brandoli, Giulia, Lempinen, Antti, Artes, Sanna, Turku, Ainoleena, Jäntti, Maria Helena, Talman, Virpi, Yli-Kauhaluoma, Jari, Tuominen, Raimo K, Boije Af Gennäs, Gustav

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Separation of steroid isomers by ion mobility mass spectrometry von Ahonen, Linda, Fasciotti, Maíra, Gennäs, Gustav Boije af, Kotiaho, Tapio, Daroda, Romeu J., Eberlin, Marcos, Kostiainen, Risto

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Mechanism of the Oxidation of Heptafulvenes to Tropones Studied by Online Mass Spectrometry and Density Functional Theory Calculations von Nilsson, Sofia M. E, Henschel, Henning, Scotti, Gianmario, Haapala, Markus, Kiriazis, Alexandros, Boije af Gennäs, Gustav, Kotiaho, Tapio, Yli-Kauhaluoma, Jari

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Design, Synthesis, and Biological Activity of Isophthalic Acid Derivatives Targeted to the C1 Domain of Protein Kinase C von af Gennäs, Gustav Boije, Talman, Virpi, Aitio, Olli, Ekokoski, Elina, Finel, Moshe, Tuominen, Raimo K, Yli-Kauhaluoma, Jari

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Interaction between retinoid acid receptor-related orphan receptor alpha (RORA) and neuropeptide S receptor 1 (NPSR1) in asthma von Acevedo, Nathalie, Sääf, Annika, Söderhäll, Cilla, Melén, Erik, Mandelin, Jami, Pietras, Christina Orsmark, Ezer, Sini, Karisola, Piia, Vendelin, Johanna, Gennäs, Gustav Boije af, Yli-Kauhaluoma, Jari, Alenius, Harri, von Mutius, Erika, Doekes, Gert, Braun-Fahrländer, Charlotte, Riedler, Josef, van Hage, Marianne, D'Amato, Mauro, Scheynius, Annika, Pershagen, Göran, Kere, Juha, Pulkkinen, Ville

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C1 Domain-targeted isophthalate derivatives induce cell elongation and cell cycle arrest in HeLa cells von Talman, Virpi, Tuominen, Raimo K, Boije af Gennäs, Gustav, Gennäs, Gustav Boije Af, Yli-Kauhaluoma, Jari, Ekokoski, Elina

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Affinity chromatography reveals direct binding of the GATA4–NKX2-5 interaction inhibitor (3i-1000) with GATA4 von Jumppanen, Mikael, Kinnunen, Sini M., Zore, Matej, Välimäki, Mika J., Talman, Virpi, Gennäs, Gustav Boije af, Ruskoaho, Heikki J., Yli-Kauhaluoma, Jari

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Orexin receptor agonist Yan 7874 is a weak agonist of orexin/hypocretin receptors and shows orexin receptor-independent cytotoxicity von Turku, Ainoleena, Rinne, Maiju K, Boije Af Gennäs, Gustav, Xhaard, Henri, Lindholm, Dan, Kukkonen, Jyrki P

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Stem cells are the most sensitive screening tool to identify toxicity of GATA4-targeted novel small-molecule compounds von Karhu, S. Tuuli, Välimäki, Mika J., Jumppanen, Mikael, Kinnunen, Sini M., Pohjolainen, Lotta, Leigh, Robert S., Auno, Samuli, Földes, Gábor, Boije af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Ruskoaho, Heikki, Talman, Virpi

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Screening for Thermotoga maritima Membrane-Bound Pyrophosphatase Inhibitors von Vidilaseris, Keni, Johansson, Niklas G, Turku, Ainoleena, Kiriazis, Alexandros, Boije Af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Xhaard, Henri, Goldman, Adrian

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Discovery of Membrane-Bound Pyrophosphatase Inhibitors Derived from an Isoxazole Fragment von Johansson, Niklas G, Turku, Ainoleena, Vidilaseris, Keni, Dreano, Loïc, Khattab, Ayman, Ayuso Pérez, Daniel, Wilkinson, Aaron, Zhang, Yuezhou, Tamminen, Matti, Grazhdankin, Evgeni, Kiriazis, Alexandros, Fishwick, Colin W. G, Meri, Seppo, Yli-Kauhaluoma, Jari, Goldman, Adrian, Boije af Gennäs, Gustav, Xhaard, Henri

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A miniaturised 3D printed polypropylene reactor for online reaction analysis by mass spectrometry von Scotti, Gianmario, Nilsson, Sofia M. E., Haapala, Markus, Pöhö, Päivi, Boije af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Kotiaho, Tapio

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Asymmetry in catalysis by Thermotoga maritima membrane-bound pyrophosphatase demonstrated by a nonphosphorus allosteric inhibitor von Vidilaseris, Keni, Kiriazis, Alexandros, Turku, Ainoleena, Khattab, Ayman, Johansson, Niklas G, Leino, Teppo O, Kiuru, Paula S, Boije Af Gennäs, Gustav, Meri, Seppo, Yli-Kauhaluoma, Jari, Xhaard, Henri, Goldman, Adrian

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Simple 3D printed stainless steel microreactors for online mass spectrometric analysis von Scotti, Gianmario, Nilsson, Sofia M.E., Matilainen, Ville-Pekka, Haapala, Markus, Boije af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Salminen, Antti, Kotiaho, Tapio

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Design, Synthesis, and Biological Activity of Urea Derivatives as Anaplastic Lymphoma Kinase Inhibitors von Boije af Gennäs, Gustav, Mologni, Luca, Ahmed, Shaheen, Rajaratnam, Mohanathas, Marin, Oriano, Lindholm, Niko, Viltadi, Michela, Gambacorti-Passerini, Carlo, Scapozza, Leonardo, Yli-Kauhaluoma, Jari

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