Evaluation of 1H‑Triazole-1‑[N,N′‑Bis(tert-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation von Wester, Anita, Björkling, Fredrik, Franzyk, Henrik

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Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment von Wróbel, Tomasz M., Jørgensen, Flemming Steen, Pandey, Amit V., Grudzińska, Angelika, Sharma, Katyayani, Yakubu, Jibira, Björkling, Fredrik

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Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids von Jørgensen, Johan Storm, Mood, Elnaz Harifi, Knap, Anne Sofie Holst, Nielsen, Simone Eidnes, Nielsen, Peter E., Żabicka, Dorota, Matias, Carina, Domraceva, Ilona, Björkling, Fredrik, Franzyk, Henrik

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Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity von Frederiksen, Nicki, Hansen, Paul R, Björkling, Fredrik, Franzyk, Henrik

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Selected strategies to fight pathogenic bacteria von Plotniece, Aiva, Sobolev, Arkadij, Supuran, Claudiu T., Carta, Fabrizio, Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, Jari, Augustyns, Koen, Cos, Paul, De Vooght, Linda, Govaerts, Matthias, Aizawa, Juliana, Tammela, Päivi, Žalubovskis, Raivis

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Optimized Synthesis of Fmoc/Boc‐Protected PNA Monomers and their Assembly into PNA Oligomers von Shaikh, Ashif Y., Björkling, Fredrik, Nielsen, Peter E., Franzyk, Henrik

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Alternating Cationic‐Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity von Frederiksen, Nicki, Hansen, Paul R., Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Domraceva, Ilona, Björkling, Fredrik, Franzyk, Henrik

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Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors von Brem, Jürgen, Panduwawala, Tharindi, Hansen, Jon Ulf, Hewitt, Joanne, Liepins, Edgars, Donets, Pawel, Espina, Laura, Farley, Alistair J. M., Shubin, Kirill, Campillos, Gonzalo Gomez, Kiuru, Paula, Shishodia, Shifali, Krahn, Daniel, Leśniak, Robert K., Schmidt (Adrian), Juliane, Calvopiña, Karina, Turrientes, María-Carmen, Kavanagh, Madeline E., Lubriks, Dmitrijs, Hinchliffe, Philip, Langley, Gareth W., Aboklaish, Ali F., Eneroth, Anders, Backlund, Maria, Baran, Andrei G., Nielsen, Elisabet I., Speake, Michael, Kuka, Janis, Robinson, John, Grinberga, Solveiga, Robinson, Lindsay, McDonough, Michael A., Rydzik, Anna M., Leissing, Thomas M., Jimenez-Castellanos, Juan Carlos, Avison, Matthew B., Da Silva Pinto, Solange, Pannifer, Andrew D., Martjuga, Marina, Widlake, Emma, Priede, Martins, Hopkins Navratilova, Iva, Gniadkowski, Marek, Belfrage, Anna Karin, Brandt, Peter, Yli-Kauhaluoma, Jari, Bacque, Eric, Page, Malcolm G. P., Björkling, Fredrik, Tyrrell, Jonathan M., Spencer, James, Lang, Pauline A., Baranczewski, Pawel, Cantón, Rafael, McElroy, Stuart P., Jones, Philip S., Baquero, Fernando, Suna, Edgars, Morrison, Angus, Walsh, Timothy R., Schofield, Christopher J.

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Silver carbene complexes: An emerging class of anticancer agents von Kankala, Shravankumar, Thota, Niranjan, Björkling, Fredrik, Taylor, Myles K., Vadde, Ravinder, Balusu, Ramesh

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Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues von Shaikh, Ashif Y., Björkling, Fredrik, Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Domraceva, Ilona, Kreicberga, Agrita, Franzyk, Henrik

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Synthesis and Antitumor Effect in Vitro and in Vivo of Substituted 1,3-Dihydroindole-2-ones von Christensen, Mette K, Erichsen, Kamille D, Trojel-Hansen, Christina, Tjørnelund, Jette, Nielsen, Søren J, Frydenvang, Karla, Johansen, Tommy N, Nielsen, Birgitte, Sehested, Maxwell, Jensen, Peter B, Ikaunieks, Martins, Zaichenko, Andrei, Loza, Einars, Kalvinsh, Ivars, Björkling, Fredrik

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Structural Basis of Metallo-β-lactamase Inhibition by N‑Sulfamoylpyrrole-2-carboxylates von Farley, Alistair J. M, Ermolovich, Yuri, Calvopiña, Karina, Rabe, Patrick, Panduwawala, Tharindi, Brem, Jürgen, Björkling, Fredrik, Schofield, Christopher J

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Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties von Frederiksen, Nicki, Louka, Stavroula, Mudaliar, Chirag, Domraceva, Ilona, Kreicberga, Agrita, Pugovics, Osvalds, Żabicka, Dorota, Tomczak, Magdalena, Wygoda, Weronika, Björkling, Fredrik, Franzyk, Henrik

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Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae von Hansen, Anna Mette, Bonke, Gitte, Hogendorf, Wouter Frederik Johan, Björkling, Fredrik, Nielsen, John, Kongstad, Kenneth T., Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Nielsen, Peter E., Franzyk, Henrik

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Nicotinamide Phosphoribosyltransferase Inhibitors, Design, Preparation, and Structure–Activity Relationship von Christensen, Mette K, Erichsen, Kamille D, Olesen, Uffe H, Tjørnelund, Jette, Fristrup, Peter, Thougaard, Annemette, Nielsen, Søren Jensby, Sehested, Maxwell, Jensen, Peter B, Loza, Einars, Kalvinsh, Ivars, Garten, Antje, Kiess, Wieland, Björkling, Fredrik

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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET von Munk Jensen, Mette, Erichsen, Kamille Dumong, Björkling, Fredrik, Madsen, Jacob, Jensen, Peter Buhl, Sehested, Maxwell, Højgaard, Liselotte, Kjær, Andreas

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Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents von Craig, Alexander J., Ermolovich, Yuri, Cameron, Alan, Rodler, Agnes, Wang, Helen, Hawkes, Jeffrey A., Hubert, Madlen, Björkling, Fredrik, Molchanova, Natalia, Brimble, Margaret A., Moodie, Lindon W. K., Svenson, Johan

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Anticancer agent CHS-828 inhibits cellular synthesis of NAD von Olesen, Uffe Høgh, Christensen, Mette Knak, Björkling, Fredrik, Jäättelä, Marja, Jensen, Peter Buhl, Sehested, Maxwell, Nielsen, Søren Jensby

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Rapid Synthesis of Aryl Azides from Aryl Halides under Mild Conditions von Andersen, Jacob, Madsen, Ulf, Björkling, Fredrik, Liang, Xifu

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Synthesis and Structure-Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents von Wróbel, Tomasz M, Rogova, Oksana, Sharma, Katyayani, Rojas Velazquez, Maria Natalia, Pandey, Amit V, Jørgensen, Flemming Steen, Arendrup, Frederic S, Andersen, Kasper L, Björkling, Fredrik

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