Plasmin‐activated doxorubicin prodrugs containing a spacer reduce tumor growth and angiogenesis without systemic toxicity von Devy, Laetitia, Groot, Franciscus M. H., Blacher, Silvia, Hajitou, Amin, Beusker, Patrick H., Scheeren, Hans W., Foidart, Jean‐Michel, Noël, Agnès

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Rearrangement of O-Cinnamoyltaxicin I to a Novel C-13 Spiro-Taxane von van Rozendaal, Erik L. M, Veldhuis, Harald, van Veldhuizen, Beb, van Beek, Teris A, de Groot, Aede, Beusker, Patrick H, Scheeren, Hans W

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"Cascade-Release Dendrimers" Liberate All End Groups upon a Single Triggering Event in the Dendritic Core von de Groot, Franciscus M. H., Albrecht, Carsten, Koekkoek, Ralph, Beusker, Patrick H., Scheeren, Hans W.

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FASEB Journal von Devy, L, de Groot, F. M, Blacher, Silvia, Hajitou, A, Beusker, P. H, Scheeren, H. W, Foidart, Jean-Michel, Noël, Agnès

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Semisynthesis of 7-Deoxypaclitaxel Derivatives Devoid of an Oxetane D-Ring, Starting from Taxine B von Beusker, Patrick H., Veldhuis, Harald, Brinkhorst, Johan, Hetterscheid, Dennis G. H., Feichter, Nicolas, Bugaut, Anthony, Scheeren, Hans W.

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Semisynthesis of Flexible 5,7-Dideoxypaclitaxel Derivatives from Taxine B von Beusker, Patrick H., Veldhuis, Harald, van den Bossche, Bianca A.C., Scheeren, Hans W.

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Exploration of High-Pressure Cycloadducts of Furans and Citraconic Anhydride as Precursors for CD-Ring Fragments of Paclitaxel and Its Analogues von Beusker, Patrick H., M. Aben, René W., Seerden, Jean-Paul G., Smits, Jan M. M., Scheeren, Hans W.

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ChemInform Abstract: Exploration of High-Pressure Cycloadducts of Furans and Citraconic Anhydride as Precursors for CD-Ring Fragments of Paclitaxel and Its Analogues von BEUSKER, P. H., ABEN, R. W. M., SEERDEN, J.-P. G., SMITS, J. M. M., SCHEEREN, H. W.

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Design, Synthesis, and Evaluation of Linker-Duocarmycin Payloads: Toward Selection of HER2-Targeting Antibody–Drug Conjugate SYD985 von Elgersma, Ronald C, Coumans, Ruud G. E, Huijbregts, Tijl, Menge, Wiro M. P. B, Joosten, John A. F, Spijker, Henri J, de Groot, Franciscus M. H, van der Lee, Miranda M. C, Ubink, Ruud, van den Dobbelsteen, Diels J, Egging, David F, Dokter, Wim H. A, Verheijden, Gijs F. M, Lemmens, Jacques M, Timmers, C. Marco, Beusker, Patrick H

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Preclinical profile of the HER2-targeting ADC SYD983/SYD985: introduction of a new duocarmycin-based linker-drug platform von Dokter, Wim, Ubink, Ruud, van der Lee, Miranda, van der Vleuten, Monique, van Achterberg, Tanja, Jacobs, Danielle, Loosveld, Eline, van den Dobbelsteen, Diels, Egging, David, Mattaar, Ellen, Groothuis, Patrick, Beusker, Patrick, Coumans, Ruud, Elgersma, Ronald, Menge, Wiro, Joosten, John, Spijker, Henri, Huijbregts, Tijl, de Groot, Vincent, Eppink, Michel, de Roo, Guy, Verheijden, Gijs, Timmers, Marco

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P10.30.B COMBINATION TREATMENT WITH ERIBULIN AND TTFIELDS INDUCES APOPTOSIS AND G2/M CELL CYCLE ARREST IN HUMAN GLIOBLASTOMA CELLS von Goett, H, Schön, C, Beusker, P, Uhl, E, Stein, M

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A Platform for the Generation of Site-Specific Antibody–Drug Conjugates That Allows for Selective Reduction of Engineered Cysteines von Coumans, Ruud G. E, Ariaans, Gerry J. A, Spijker, Henri J, Renart Verkerk, Pascal, Beusker, Patrick H, Kokke, Bas P. A, Schouten, Jan, Blomenröhr, Marion, van der Lee, Miranda M. C, Groothuis, Patrick G, Ubink, Ruud, Dokter, Wim H. A, Timmers, C. Marco

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Tumor treating fields with the TERT-inhibitor eribulin have synergistic antiproliferative effects on human glioblastoma cells von Beusker, P., Gött, H., Kolodziej, M., Uhl, E., Stein, M.

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