Structure-based Discovery of Antagonists of Nuclear Receptor LRH-1 von Benod, Cindy, Carlsson, Jens, Uthayaruban, Rubatharshini, Hwang, Peter, Irwin, John J., Doak, Allison K., Shoichet, Brian K., Sablin, Elena P., Fletterick, Robert J.

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Nuclear receptor liver receptor homologue 1 (LRH-1) regulates pancreatic cancer cell growth and proliferation von Benod, Cindy, Vinogradova, Maia V., Jouravel, Natalia, Kim, Grace E., Fletterick, Robert J., Sablin, Elena P.

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The human orphan nuclear receptor tailless (TLX, NR2E1) is druggable von Benod, Cindy, Villagomez, Rosa, Filgueira, Carly S, Hwang, Peter K, Leonard, Paul G, Poncet-Montange, Guillaume, Rajagopalan, Senapathy, Fletterick, Robert J, Gustafsson, Jan-Åke, Webb, Paul

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TLX: An elusive receptor von Benod, Cindy, Villagomez, Rosa, Webb, Paul

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Abstract 2452: Deorphanizing TLX: Implications for treatment of glioblastomas von Benod, Cindy C., Villagomez, Rosa, Webb, Paul

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Structure of the retinoid X receptor α–liver X receptor β (RXRα–LXRβ) heterodimer on DNA von Lou, Xiaohua, Toresson, Gudrun, Benod, Cindy, Suh, Ji Ho, Philips, Kevin J, Webb, Paul, Gustafsson, Jan-Ake

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Abstract A06: Biophysical and biochemical characterization of KRAS G12C inhibition through the SMARTTM platform von Zhou, Minyun, Yuzhakov, Alexander, Benod, Cindy C, Xue, Linlong, Silver, Alec D, Iyer, Ganesh, Townson, Sharon A., Jin, Meizhong, Perl, Nicholas R., Kohlmann, Anna, Mann, Alan S., Akcay, Gizem, May, Earl W.

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Abstract 1858: Estrogen receptor beta as a tractable therapeutic target von Filgueira, Carly S., Benod, Cindy, Lou, Xiaohua, Strom, Anders, Gustafsson, Jan-Åke, Berkenstam, Anders, Webb, Paul

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Abstract B37: Development of inhibitors of the activated form of KRAS G12C von Stewart, Michelle L., Perl, Nicholas R., Lee, Seung-Joo, Xue, Linlong, Zhou, Minyun, Simon, Jonah, Luly, Kathryn M., Grigoriu, Siminia, Yuzhakov, Alex, Silver, Alec, Lowe, Jason T., Benod, Cindy C., Mann, Alan S., Verdine, Gregory L., Rigby, Alan C., Mulvihill, Mark J., May, Earl W., Kohlmann, Anna, Townson, Sharon A., Pollock, Roy M., Jin, Meizhong

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Structure of the retinoid X receptor [alpha]-liver X receptor [beta] (RXR[alpha]-LXR[beta]) heterodimer on DNA von Lou, Xiaohua, Toresson, Gudrun, Benod, Cindy, Suh, Ji Ho, Philips, Kevin J, Webb, Paul, Gustafsson, Jan-ake

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Discovery of a highly active ligand of human pregnane x receptor: a case study from pharmacophore modeling and virtual screening to "in vivo" biological activity von Lemaire, Géraldine, Benod, Cindy, Nahoum, Virginie, Pillon, Arnaud, Boussioux, Anne-Marie, Guichou, Jean-François, Subra, Guy, Pascussi, Jean-Marc, Bourguet, William, Chavanieu, Alain, Balaguer, Patrick

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A screening cascade to identify ERβ ligands von Filgueira, Carly S, Benod, Cindy, Lou, Xiaohua, Gunamalai, Prem S, Villagomez, Rosa A, Strom, Anders, Gustafsson, Jan-Åke, Berkenstam, Anders L, Webb, Paul

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N-1H-Benzimidazol-5-ylbenzenesulfonamide derivatives as potent hPXR agonists von BENOD, Cindy, SUBRA, Guy, CHAVANIEU, Alain, NAHOUM, Virginie, MALLAVIALLE, Aude, GUICHOU, Jean-Francois, MILHAU, Julien, ROBLES, Samuel, BOURGUET, William, PASCUSSI, Jean-Marc, BALAGUER, Patrick

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CRAACK:  Consensus Program for NMR Amino Acid Type Assignment von Benod, Cindy, Delsuc, Marc-André, Pons, Jean-Luc

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N-1 H-Benzimidazol-5-ylbenzenesulfonamide derivatives as potent hPXR agonists von Benod, Cindy, Subra, Guy, Nahoum, Virginie, Mallavialle, Aude, Guichou, Jean-François, Milhau, Julien, Roblés, Samuel, Bourguet, William, Pascussi, Jean-Marc, Balaguer, Patrick, Chavanieu, Alain

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Discovery of a Highly Active Ligand of Human Pregnane X Receptor: A Case Study from Pharmacophore Modeling and Virtual Screening to “In Vivo” Biological Activity von Géraldine Lemaire, Cindy Benod, Virginie Nahoum, Arnaud Pillon, Anne-Marie Boussioux, Jean-François Guichou, Guy Subra, Jean-Marc Pascussi, William Bourguet, Alain Chavanieu, Patrick Balaguer

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