6-LB: GPR119 Agonist PRM A Increases Glucagon Response to Hypoglycemia in Rats von KWOK, DAVID W.K., ALEXANDER, DIANE, BEELEY, NIGEL R.A., KELLEY, DAVID

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Discovery and Structure−Activity Relationship of (1R)-8-Chloro-2,3,4,5-tetrahydro-1-methyl-1H-3-benzazepine (Lorcaserin), a Selective Serotonin 5-HT2C Receptor Agonist for the Trea... von Smith, Brian M, Smith, Jeffrey M, Tsai, James H, Schultz, Jeffrey A, Gilson, Charles A, Estrada, Scott A, Chen, Rita R, Park, Douglas M, Prieto, Emily B, Gallardo, Charlemagne S, Sengupta, Dipanjan, Dosa, Peter I, Covel, Jon A, Ren, Albert, Webb, Robert R, Beeley, Nigel R. A, Martin, Michael, Morgan, Michael, Espitia, Stephen, Saldana, Hazel R, Bjenning, Christina, Whelan, Kevin T, Grottick, Andrew J, Menzaghi, Frederique, Thomsen, William J

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Discovery and SAR of new benzazepines as potent and selective 5-HT2C receptor agonists for the treatment of obesity von SMITH, Brian M, SMITH, Jeffrey M, DIPANJAN SENGUPTA, THOMSEN, William J, SALDANA, Hazel R, WHELAN, Kevin T, MENZAGHI, Frederique, WEBB, Robert R, BEELEY, Nigel R. A, TSAI, James H, SCHULTZ, Jeffrey A, GILSON, Charles A, ESTRADA, Scott A, CHEN, Rita R, PARK, Douglas M, PRIETO, Emily B, GALLARDO, Charlemagne S

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Discovery of 1-[3-(4-Bromo-2-methyl-2 H -pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine 2A Inverse Agonists for the Treatm... von Teegarden, Bradley R., Li, Hongmei, Jayakumar, Honnappa, Strah-Pleynet, Sonja, Dosa, Peter I., Selaya, Susan D., Kato, Naomi, Elwell, Katie H., Davidson, Jarrod, Cheng, Karen, Saldana, Hazel, Frazer, John M., Whelan, Kevin, Foster, Jonathan, Espitia, Stephan, Webb, Robert R., Beeley, Nigel R. A., Thomsen, William, Morairty, Stephen R., Kilduff, Thomas S., Al-Shamma, Hussien A.

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Can peptides be mimicked? von Beeley, Nigel R.A

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Discovery of 1-[3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (Nelotanserin) and Related 5-Hydroxytryptamine2A Inverse Agonists for the Treatment... von Teegarden, Bradley R, Li, Hongmei, Jayakumar, Honnappa, Strah-Pleynet, Sonja, Dosa, Peter I, Selaya, Susan D, Kato, Naomi, Elwell, Katie H, Davidson, Jarrod, Cheng, Karen, Saldana, Hazel, Frazer, John M, Whelan, Kevin, Foster, Jonathan, Espitia, Stephan, Webb, Robert R, Beeley, Nigel R. A, Thomsen, William, Morairty, Stephen R, Kilduff, Thomas S, Al-Shamma, Hussien A

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Improved tumor targeting with chemically cross-linked recombinant antibody fragments von KING, D. J, TURNER, A, MILLAR, K, MILLICAN, T. A, BOYCE, B. A, ANTONIW, P, MOUNTAIN, A, BEGENT, R. H. J, SHOCHAT, D, YARRANTON, G. T, FARNSWORTH, A. P. H, ADAIR, J. R, OWENS, R. J, PEDLEY, R. B, BALDOCK, D, PROUDFOOT, K. A, LAWSON, A. D. G, BEELEY, N. R. A

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Discovery and SAR of new benzazepines as potent and selective 5-HT 2C receptor agonists for the treatment of obesity von Smith, Brian M., Smith, Jeffrey M., Tsai, James H., Schultz, Jeffrey A., Gilson, Charles A., Estrada, Scott A., Chen, Rita R., Park, Douglas M., Prieto, Emily B., Gallardo, Charlemagne S., Sengupta, Dipanjan, Thomsen, William J., Saldana, Hazel R., Whelan, Kevin T., Menzaghi, Frederique, Webb, Robert R., Beeley, Nigel R.A.

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An in Vivo Model for Screening Peptidomimetic Inhibitors of Gelatinase A von Chander, Surinder K., Antoniw, Pari, Beeley, Nigel R.A., Boyce, Byron, Crabbe, Thomas, Docherty, Andrew J.P., Leonard, Joanna, Mason, Barbara, Millar, Kenneth, Millican, Andrew T., Morphy, Richard, Mountain, Andrew, O'Connell, James, Porter, John R., Willmott, Neville

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Section Review Oncologic, Endocrine & Metabolic: The amylin, CGRP and calcitonin family of peptides von RA Beeley, Nigel, Prickett, Kathryn S

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Medicinal Chemistry – An Introduction von Beeley, Nigel R.A

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Discovery of 4-(dimethylamino)quinazolines as potent and selective antagonists for the melanin-concentrating hormone receptor 1 von Kanuma, Kosuke, Omodera, Katsunori, Nishiguchi, Mariko, Funakoshi, Takeo, Chaki, Shigeyuki, Semple, Graeme, Tran, Thuy-Anh, Kramer, Bryan, Hsu, Debbie, Casper, Martin, Thomsen, Bill, Beeley, Nigel, Sekiguchi, Yoshinori

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Corrigendum von Beeley, Nigel R.A.

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Peptidomimetics and small-molecule drug design: Towards improved bioavailability and in vivo stability von Beeley, Nigel

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Compositions and methods for treating metabolic disorders von Beeley, Nigel R. A, Fineman, Mark S, Baron, Alain D

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GPCRs: an update on structural approaches to drug discovery von Beeley, Nigel R.A., Sage, Carleton

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Biguanide compositions and methods of treating metabolic disorders von Beeley, Nigel R. A, Fineman, Mark S, Baron, Alain D

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COMPOSITIONS AND METHODS FOR TREATING METABOLIC DISORDERS von BEELEY, Nigel R.A, FINEMAN, Mark S, BARON, Alain D

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Overview: Macrocyclic Chelators as Anticancer Agents in Radioimmunotherapy von Beeley, Nigel R A, Ansell, Phillip R J

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METHODS FOR TREATING A PULMONARY DISEASE WITH AN ALK-5 (TGF BETA R1) INHIBITOR von Beeley, Nigel R.A, FOULKES, John Gordon, Crystal, Roger, BULLOUGH, David A

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