New approaches for the treatment of Alzheimer’s disease von Fish, Paul V., Steadman, David, Bayle, Elliott D., Whiting, Paul

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Copper-Catalyzed Electrophilic Carbofunctionalization of Alkynes to Highly Functionalized Tetrasubstituted Alkenes von Suero, Marcos G, Bayle, Elliott D, Collins, Beatrice S. L, Gaunt, Matthew J

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Systematic Investigation of the Permeability of Androgen Receptor PROTACs von Scott, Duncan E, Rooney, Timothy P. C, Bayle, Elliott D, Mirza, Tashfina, Willems, Henriette M. G, Clarke, Jonathan H, Andrews, Stephen P, Skidmore, John

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Design of a Chemical Probe for the Bromodomain and Plant Homeodomain Finger-Containing (BRPF) Family of Proteins von Igoe, Niall, Bayle, Elliott D, Tallant, Cynthia, Fedorov, Oleg, Meier, Julia C, Savitsky, Pavel, Rogers, Catherine, Morias, Yannick, Scholze, Sarah, Boyd, Helen, Cunoosamy, Danen, Andrews, David M, Cheasty, Anne, Brennan, Paul E, Müller, Susanne, Knapp, Stefan, Fish, Paul V

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An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent von Willis, Nicky J, Bayle, Elliott D, Papageorgiou, George, Steadman, David, Atkinson, Benjamin N, Mahy, William, Fish, Paul V

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Carboxylesterase Notum Is a Druggable Target to Modulate Wnt Signaling von Bayle, Elliott D, Svensson, Fredrik, Atkinson, Benjamin N, Steadman, David, Willis, Nicky J, Woodward, Hannah L, Whiting, Paul, Vincent, Jean-Paul, Fish, Paul V

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What Value Can Operational Feasibility Studies Bring to Post Marketing Observational Studies (PMOS)? Example of Feasibility Study Performed in Eastern Europe to Assess Hepatitis C... von El Kebir, S, Bayle, D, Gauchoux, R

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New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atoms von Spurr, Sophie S., Bayle, Elliott D., Yu, Wenyu, Li, Fengling, Tempel, Wolfram, Vedadi, Masoud, Schapira, Matthieu, Fish, Paul V.

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Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit von Willis, Nicky J., Mahy, William, Sipthorp, James, Zhao, Yuguang, Woodward, Hannah L., Atkinson, Benjamin N., Bayle, Elliott D., Svensson, Fredrik, Frew, Sarah, Jeganathan, Fiona, Monaghan, Amy, Benvegnù, Stefano, Jolly, Sarah, Vecchia, Luca, Ruza, Reinis R., Kjær, Svend, Howell, Steven, Snijders, Ambrosius P., Bictash, Magda, Salinas, Patricia C., Vincent, Jean-Paul, Jones, E. Yvonne, Whiting, Paul, Fish, Paul V.

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Physical exercise influences attentional orientation towards emotional stimuli von Mansouri, N., Coutté, A., Dru, V., Bayle, D.

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Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors von Atkinson, Benjamin N., Steadman, David, Mahy, William, Zhao, Yuguang, Sipthorp, James, Bayle, Elliott D., Svensson, Fredrik, Papageorgiou, George, Jeganathan, Fiona, Frew, Sarah, Monaghan, Amy, Bictash, Magda, Jones, E. Yvonne, Fish, Paul V.

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Design of a Biased Potent Small Molecule Inhibitor of the Bromodomain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies von Igoe, Niall, Bayle, Elliott D, Fedorov, Oleg, Tallant, Cynthia, Savitsky, Pavel, Rogers, Catherine, Owen, Dafydd R, Deb, Gauri, Somervaille, Tim C. P, Andrews, David M, Jones, Neil, Cheasty, Anne, Ryder, Hamish, Brennan, Paul E, Müller, Susanne, Knapp, Stefan, Fish, Paul V

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Cortical dynamics of externally and self-directed attention: a MEG study of a card sorting task von Fonlupt, P., Henaff, M.A., Bayle, D., Krolak-Salmon, P.

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Structural Analysis and Development of Notum Fragment Screening Hits von Zhao, Yuguang, Mahy, William, Willis, Nicky J, Woodward, Hannah L, Steadman, David, Bayle, Elliott D, Atkinson, Benjamin N, Sipthorp, James, Vecchia, Luca, Ruza, Reinis R, Harlos, Karl, Jeganathan, Fiona, Constantinou, Stefan, Costa, Artur, Kjær, Svend, Bictash, Magda, Salinas, Patricia C, Whiting, Paul, Vincent, Jean-Paul, Fish, Paul V, Jones, E Yvonne

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Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation von Meier, Julia C, Tallant, Cynthia, Fedorov, Oleg, Witwicka, Hanna, Hwang, Sung-Yong, van Stiphout, Ruud G, Lambert, Jean-Philippe, Rogers, Catherine, Yapp, Clarence, Gerstenberger, Brian S, Fedele, Vita, Savitsky, Pavel, Heidenreich, David, Daniels, Danette L, Owen, Dafydd R, Fish, Paul V, Igoe, Niall M, Bayle, Elliott D, Haendler, Bernard, Oppermann, Udo C.T, Buffa, Francesca, Brennan, Paul E, Müller, Susanne, Gingras, Anne Claude, Odgren, Paul R, Birnbaum, Mark J, Knapp, Stefan

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Inhibitory effect of procyanidin-rich extracts on LDL oxidation in vitro von Mazur, A, Bayle, D, Lab, C, Rock, E, Rayssiguier, Y

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Morphological and immune response alterations in the intestinal mucosa of the mouse after short periods on a low-magnesium diet von Zimowska, W., Girardeau, J. P., Kuryszko, J., Bayle, D., Rayssiguier, Y., Mazur, A.

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PRM216 - What Value Can Operational Feasibility Studies Bring to Post Marketing Observational Studies (PMOS)? Example of Feasibility Study Performed in Eastern Europe to Assess Hep... von El Kebir, S., Bayle, D., Gauchoux, R.

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Migraine headaches and pain with neuropathic characteristics: Comorbid conditions in patients with multiple sclerosis von Moisset, Xavier, Ouchchane, Lemlih, Guy, Nathalie, Bayle, Dimitri J., Dallel, Radhouane, Clavelou, Pierre

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Hiva Oa (1901-1903): Gauguin aux îles Marquises von Bayle-Ottenheim, Jacques

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