A bitopic agonist bound to the dopamine 3 receptor reveals a selectivity site von Arroyo-Urea, Sandra, Nazarova, Antonina L., Carrión-Antolí, Ángela, Bonifazi, Alessandro, Battiti, Francisco O., Lam, Jordy Homing, Newman, Amy Hauck, Katritch, Vsevolod, García-Nafría, Javier

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2016 Philip S. Portoghese Medicinal Chemistry Lectureship: Designing Bivalent or Bitopic Molecules for G‑Protein Coupled Receptors. The Whole Is Greater Than the Sum of Its Parts von Newman, Amy Hauck, Battiti, Francisco O, Bonifazi, Alessandro

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Chirality of Novel Bitopic Agonists Determines Unique Pharmacology at the Dopamine D3 Receptor von Adhikari, Pramisha, Xie, Bing, Semeano, Ana, Bonifazi, Alessandro, Battiti, Francisco O., Newman, Amy H., Yano, Hideaki, Shi, Lei

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Chiral Cyclic Aliphatic Linkers as Building Blocks for Selective Dopamine D-2 or D-3 Receptor Agonists von Battiti, Francisco O., Zaidi, Saheem A., Katritch, Vsevolod, Newman, Amy Hauck, Bonifazi, Alessandro

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Chiral Cyclic Aliphatic Linkers as Building Blocks for Selective Dopamine D2 or D3 Receptor Agonists von Battiti, Francisco O, Zaidi, Saheem A, Katritch, Vsevolod, Newman, Amy Hauck, Bonifazi, Alessandro

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Involvement of dopamine D3 receptor in impulsive choice decision-making in male rats von Shen, Hui, Ma, Zilu, Hans, Emma, Duan, Ying, Bi, Guo-Hua, Chae, Yurim C., Bonifazi, Alessandro, Battiti, Francisco O., Newman, Amy Hauck, Xi, Zheng-Xiong, Yang, Yihong

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Structure Activity Relationships for a Series of Eticlopride-Based Dopamine D-2/D-3 Receptor Bitopic Ligands von Shaik, Anver Basha, Boateng, Comfort A., Battiti, Francisco O., Bonifazi, Alessandro, Cao, Jianjing, Chen, Li, Chitsazi, Rezvan, Ravi, Saiprasad, Lee, Kuo Hao, Shi, Lei, Newman, Amy Hauck

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Exception That Proves the Rule: Investigation of Privileged Stereochemistry in Designing Dopamine D3R Bitopic Agonists von Battiti, Francisco O, Newman, Amy Hauck, Bonifazi, Alessandro

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Chemical manipulations on the 1,4-dioxane ring of 5-HT1A receptor agonists lead to antagonists endowed with antitumor activity in prostate cancer cells von Del Bello, Fabio, Bonifazi, Alessandro, Giorgioni, Gianfabio, Quaglia, Wilma, Amantini, Consuelo, Morelli, Maria Beatrice, Santoni, Giorgio, Battiti, Francisco O., Vistoli, Giulio, Cilia, Antonio, Piergentili, Alessandro

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Novel Dual-Target mu-Opioid Receptor and Dopamine D-3 Receptor Ligands as Potential Nonaddictive Pharmacotherapeutics for Pain Management von Bonifazi, Alessandro, Battiti, Francisco O., Sanchez, Julie, Zaidi, Saheem A., Bow, Eric, Makarova, Mariia, Cao, Jianjing, Shaik, Anver Basha, Sulima, Agnieszka, Rice, Kenner C., Katritch, Vsevolod, Canals, Meritxell, Lane, J. Robert, Newman, Amy Hauck

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The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D 3 Receptor (D 3 R) Selective Agonists von Battiti, Francisco O, Cemaj, Sophie L, Guerrero, Adrian M, Shaik, Anver Basha, Lam, Jenny, Rais, Rana, Slusher, Barbara S, Deschamps, Jeffery R, Imler, Greg H, Newman, Amy Hauck, Bonifazi, Alessandro

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The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D3 Receptor (D3R) Selective Agonists von Battiti, Francisco O, Cemaj, Sophie L, Guerrero, Adrian M, Shaik, Anver Basha, Lam, Jenny, Rais, Rana, Slusher, Barbara S, Deschamps, Jeffery R, Imler, Greg H, Newman, Amy Hauck, Bonifazi, Alessandro

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Structure Activity Relationships for a Series of Eticlopride-Based Dopamine D2/D3 Receptor Bitopic Ligands von Shaik, Anver Basha, Boateng, Comfort A, Battiti, Francisco O, Bonifazi, Alessandro, Cao, Jianjing, Chen, Li, Chitsazi, Rezvan, Ravi, Saiprasad, Lee, Kuo Hao, Shi, Lei, Newman, Amy Hauck

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Linkers in Bitopic Agonists Shape Bias Profile among Transducers for the Dopamine D2 and D3 Receptors von Semeano, Ana, Garland, Rian, Bonifazi, Alessandro, Lee, Kuo Hao, Famiglietti, John, Zhang, Wenqi, Jo, Yoon Jae, Battiti, Francisco O., Shi, Lei, Newman, Amy Hauck, Yano, Hideaki

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Chirality of novel bitopic agonists determine unique pharmacology at the dopamine 2 and 3 receptors von Adhikari, Pramisha, Yano, Hideaki, Bonifazi, Alessandro, Battiti, Francisco O., Newman, Amy Hauck, Shi, Lei

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Exception That Proves the Rule: Investigation of Privileged Stereochemistry in Designing Dopamine D 3 R Bitopic Agonists von Battiti, Francisco O., Newman, Amy Hauck, Bonifazi, Alessandro

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Novel Dual-Target μ‑Opioid Receptor and Dopamine D3 Receptor Ligands as Potential Nonaddictive Pharmacotherapeutics for Pain Management von Bonifazi, Alessandro, Battiti, Francisco O, Sanchez, Julie, Zaidi, Saheem A, Bow, Eric, Makarova, Mariia, Cao, Jianjing, Shaik, Anver Basha, Sulima, Agnieszka, Rice, Kenner C, Katritch, Vsevolod, Canals, Meritxell, Lane, J. Robert, Newman, Amy Hauck

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Novel Dual-Target Mu Opioid (MOR) and Dopamine D3 Receptors (D3R) Ligands as Potential Non-Addictive Pharmacotherapeutics for Pain Management von Bonifazi, Alessandro, Battiti, Francisco O., Sanchez, Julie, Zaidi, Saheem A., Bow, Eric, Makarova, Mariia, Cao, Jianjing, Shaik, Anver Basha, Sulima, Agnieszka, Rice, Kenner C., Katritch, Vsevolod, Canals, Meritxell, Lane, J. Robert, Newman, Amy Hauck

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Chemical manipulations on the 1,4-dioxane ring of 5-HT 1A receptor agonists lead to antagonists endowed with antitumor activity in prostate cancer cells von Del Bello, Fabio, Bonifazi, Alessandro, Giorgioni, Gianfabio, Quaglia, Wilma, Amantini, Consuelo, Morelli, Maria Beatrice, Santoni, Giorgio, Battiti, Francisco O, Vistoli, Giulio, Cilia, Antonio, Piergentili, Alessandro

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DUAL-TARGET MU OPIOID AND DOPAMINE D3 RECEPTORS LIGANDS; PREPARATION AND USE THEREOF von BONIFAZI, Alessandro, BATTITI, Francisco O, NEWMAN, Amy Hauck

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