Identification of a Series of Tricyclic Natural Products as Potent Broad-Spectrum Inhibitors of Metallo-β-Lactamases von PAYNE, David J, HUESO-RODRIGUEZ, Juan Antonio, RITTENHOUSE, Stephen, TEW, David, DIEZ, Emilio, PEREZ, Paloma, DE LA FUENTE, Jesus, REES, Michael, RIVERA-SAGREDO, Alfonso, BODY, Helen, CONCHA, Néstor O, JANSON, Cheryl A, GILPIN, Martin, BATESON, John H, CHEEVER, Christy, NICONOVICH, Nancy L, PEARSON, Stewart

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Crystal Structure of the IMP-1 Metallo β-Lactamase from Pseudomonas aeruginosa and Its Complex with a Mercaptocarboxylate Inhibitor:  Binding Determinants of a Potent, Broad-Spectr... von Concha, Néstor O, Janson, Cheryl A, Rowling, Pam, Pearson, Stewart, Cheever, Christy A, Clarke, Brian P, Lewis, Ceri, Galleni, Moreno, Frère, Jean-Marie, Payne, David J, Bateson, John H, Abdel-Meguid, Sherin S

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Crystal Structure of the Zinc-Dependent β-Lactamase from Bacillus cereus at 1.9 Å Resolution:  Binuclear Active Site with Features of a Mononuclear Enzyme von Fabiane, Stella Maris, Sohi, Maninder K, Wan, Tommy, Payne, David J, Bateson, John H, Mitchell, Tim, Sutton, Brian J

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SAR of biphenyl carboxamide ligands of the human melanin-concentrating hormone receptor 1 (MCH R1): Discovery of antagonist SB-568849 von Witty, David R., Bateson, John H., Hervieu, Guillaume J., Jeffrey, Phillip, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin M., Wilson, Shelagh, Winborn, Kim Y.

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Thiocarbonyl-based 1,3-dipolarophiles for the synthesis of C(2)-unsubstituted penems von Gallagher, Timothy, Sanchez, Sylvie, Bateson, John H., O'Hanlon, Peter J.

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S-Alkyl Dithioformates as 1,3-Dipolarophiles. Generation of C(2)-Unsubstituted Penems von Sanchez, Sylvie, Bateson, John H, O'Hanlon, Peter J, Gallagher, Timothy

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beta-lactamase epidemiology and the utility of established and novel beta-lactamase inhibitors von Payne, David J, Du, Wensheng, Bateson, John H

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Characterization of Monomeric L1 Metallo-β-lactamase and the Role of the N-terminal Extension in Negative Cooperativity and Antibiotic Hydrolysis von Simm, Alan M., Higgins, Catherine S., Carenbauer, Anne L., Crowder, Michael W., Bateson, John H., Bennett, Peter M., Clarke, Anthony R., Halford, Stephen E., Walsh, Timothy R.

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Inhibition of metallo-β-lactamases by a series of thiol ester derivatives of mercaptophenylacetic acid von Payne, David J., Bateson, John H., Gasson, Brian C., Khushi, Teresa, Proctor, David, Pearson, Stewart C., Reid, Robert

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NOVEL C-3 CYCLIC ETHER CEPHALOSPORINS AND THEIR ORALLY ABSORBED PRODRUG ESTERS von BATESON, JOHN H., BURTON, GEORGE, FELL, STEPHEN C.M., SMULDERS, HAZEL C.

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Inhibition of metallo-β-lactamases by a series of thiol ester derivatives of mercaptophenylacetic acid von Payne, David J., Bateson, John H., Gasson, Brian C., Khushi, Teresa, Proctor, David, Pearson, Stewart C., Reid, Robert

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Olivanic acid analogues. Part 9. Allylic oxidative functionalisation of substituted azetidinones: synthesis of some 4-acyloxy-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylates von Bateson, John H., Robins, Alison M., Southgate, Robert

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Olivanic acid analogues. Part 11. Ozonolysis of α-ethylideneazetidinones: ozonide fragmentation to α-amino acid-N-carboxyanhydrides von Bateson, John H., Fell, Stephen C. M., Kaura, Arun C., Southgate, Robert

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Perkin communications. Stereochemistry of substituted 1-alkoxybicyclo[2.2.2]octenes; Diels–Alder synthesis versus Tandem-Michael strategy von Bateson, John H., Smith, Carol F., Wilkinson, J. Bruce

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Olivanic acid analogues. Part 8. Halogenation and sulphenylation reactions leading selectively to cis-carbapenem precursors; stereospecific synthesis of (±)-6-epithienamycin von Bateson, John H., Robins, Alison M., Southgate, Robert

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Synthesis of the 3-acetoxy-7-oxo-1-azabicyclo [3.2.0] hept-2-ene-2-carboxylate system von Bateson, John H, Fell, Stephen C.M, Southgate, Robert

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Olivanic acid analogues. Part 6. Biomimetic synthesis of (±)-PS-5, (±)-6-Epi-PS-5, and (±)-benzyl MM22381 von Bateson, John H., Hickling, Roger I., Smale, Terence C., Southgate, Robert

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Characterization of Monomeric L1 Metallo-β-lactamase and the Role of the N-terminal Extension in Negative Cooperativity and Antibiotic Hydrolysis von Alan M. Simm, Catherine S. Higgins, Anne L. Carenbauer, Michael W. Crowder, John H. Bateson, Peter M. Bennett, Anthony R. Clarke, Stephen E. Halford, Timothy R. Walsh

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The regioselectivity of cycloaddition reactions between diazomethane and 3-vinylcephalosporins von FELL, S. C. M, PEARSON, M. J, BURTON, G, BATESON, J. H

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Olivanic acid analogues. Part 5. Synthesis of 3-alkylthio and 3-alkylsulphinyl analogues via Michael addition of thiols to 3-unsubstituted 1-azabicyclo[3.2.0]hept-2-ene-2-carboxyla... von Bateson, John H., Roberts, Patricia M., Smale, Terence C., Southgate, Robert

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