Crystal structures of the M1 and M4 muscarinic acetylcholine receptors von Thal, David M., Sun, Bingfa, Feng, Dan, Nawaratne, Vindhya, Leach, Katie, Felder, Christian C., Bures, Mark G., Evans, David A., Weis, William I., Bachhawat, Priti, Kobilka, Tong Sun, Sexton, Patrick M., Kobilka, Brian K., Christopoulos, Arthur

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PL-PatchSurfer: a novel molecular local surface-based method for exploring protein-ligand interactions von Hu, Bingjie, Zhu, Xiaolei, Monroe, Lyman, Bures, Mark G, Kihara, Daisuke

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Discovery of (1S,2R,3S,4S,5R,6R)‑2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Metabo... von Chappell, Mark D, Li, Renhua, Smith, Stephon C, Dressman, Bruce A, Tromiczak, Eric G, Tripp, Allie E, Blanco, Maria-Jesus, Vetman, Tatiana, Quimby, Steven J, Matt, James, Britton, Thomas C, Fivush, Adam M, Schkeryantz, Jeffrey M, Mayhugh, Daniel, Erickson, Jon A, Bures, Mark G, Jaramillo, Carlos, Carpintero, Mercedes, Diego, José Eugenio de, Barberis, Mario, Garcia-Cerrada, Susana, Soriano, José F, Antonysamy, Stephen, Atwell, Shane, MacEwan, Iain, Condon, Bradley, Sougias, Christine, Wang, Jing, Zhang, Aiping, Conners, Kris, Groshong, Chris, Wasserman, Stephen R, Koss, John W, Witkin, Jeffrey M, Li, Xia, Overshiner, Carl, Wafford, Keith A, Seidel, Wesley, Wang, Xu-Shan, Heinz, Beverly A, Swanson, Steven, Catlow, John T, Bedwell, David W, Monn, James A, Mitch, Charles H, Ornstein, Paul L

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Synthesis and Pharmacological Characterization of 4‑Substituted-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylates: Identification of New Potent and Selective Metabotropic Glutamate 2/... von Monn, James A, Valli, Matthew J, Massey, Steven M, Hao, Junliang, Reinhard, Matthew R, Bures, Mark G, Heinz, Beverly A, Wang, Xushan, Carter, Joan H, Getman, Brian G, Stephenson, Gregory A, Herin, Marc, Catlow, John T, Swanson, Steven, Johnson, Bryan G, McKinzie, David L, Henry, Steven S

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Design and synthesis of N-[6-(Substituted Aminoethylideneamino)-2-Hydroxyindan-1-yl]arylamides as selective and potent muscarinic M1 agonists von Liu, Bin, Croy, Carrie H., Hitchcock, Stephen A., Allen, Jennifer R., Rao, Zhigang, Evans, David, Bures, Mark G., McKinzie, David L., Watt, Marla Leigh, Stuart Gregory, G., Hansen, Marvin M., Hoogestraat, Paul J., Jamison, James A., Okha-Mokube, Fese M., Stratford, Robert E., Turner, William, Bymaster, Frank, Felder, Christian C.

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Discovery of a Potent Inhibitor of the Antiapoptotic Protein Bcl-xL from NMR and Parallel Synthesis von Petros, Andrew M, Dinges, Jurgen, Augeri, David J, Baumeister, Steven A, Betebenner, David A, Bures, Mark G, Elmore, Steven W, Hajduk, Philip J, Joseph, Mary K, Landis, Shelley K, Nettesheim, David G, Rosenberg, Saul H, Shen, Wang, Thomas, Sheela, Wang, Xilu, Zanze, Irini, Zhang, Haichao, Fesik, Stephen W

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Computational methods in molecular diversity and combinatorial chemistry von Bures, Mark G, Martin, Yvonne C

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A fast new approach to pharmacophore mapping and its application to dopaminergic and benzodiazepine agonists von Martin, Y C, Bures, M G, Danaher, E A, DeLazzer, J, Lico, I, Pavlik, P A

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Discovery of a Potent Inhibitor of the Antiapoptotic Protein Bcl-x L from NMR and Parallel Synthesis von Petros, Andrew M., Dinges, Jurgen, Augeri, David J., Baumeister, Steven A., Betebenner, David A., Bures, Mark G., Elmore, Steven W., Hajduk, Philip J., Joseph, Mary K., Landis, Shelley K., Nettesheim, David G., Rosenberg, Saul H., Shen, Wang, Thomas, Sheela, Wang, Xilu, Zanze, Irini, Zhang, Haichao, Fesik, Stephen W.

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3-(2-(3-Pyridinyl)thiazolidin-4-oyl)indoles, a Novel Series of Platelet Activating Factor Antagonists von Sheppard, George S, Pireh, Daisy, Carrera, George M, Bures, Mark G, Heyman, H. Robin, Steinman, Douglas H, Davidsen, Steven K, Phillips, James G, Guinn, Denise E, May, Paul D, Conway, Richard D, Rhein, David A, Calhoun, William C, Albert, Daniel H, Magoc, Terrance J, Carter, George W, Summers, James B

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Mechanism of differential activities of ofloxacin enantiomers von MORRISSEY, I, HOSHINO, K, SATO, K, YOSHIDA, A, HAYAKAWA, I, BURES, M. G, SHEN, L. L

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The discovery of novel auxin transport inhibitors by molecular modeling and three-dimensional pattern analysis von Bures, M G, Black-Schaefer, C, Gardner, G

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Computer-assisted mechanistic evaluation of organic reactions. 15. Heterocycle synthesis von Bures, Mark G, Jorgensen, William L

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Computer-assisted mechanistic evaluation of organic reactions. 11. Electrophilic aromatic substitution von Bures, Mark G, Roos-Kozel, Barbara L, Jorgensen, William L

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5-membered heteroaryl carboxamide compounds for treatment of HBV von Rai, Roopa, Bannen, Lynne, Li, Leping, Haydar, Simon Nicolas, Bures, Mark G, Walker, Michael

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5-Membered Heteroaryl Carboxamide Compounds for Treatment of HBV von BANNEN, Lynne, HAYDAR, Simon Nicolas, LI, Leping, BURES, Mark G, WALKER, Michael, RAI, Roopa

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HEPATITIS B CORE PROTEIN MODULATORS von ARNOLD, Lee D, TURNER, William W, LI, Leping, BURES, Mark G, HAYDAR, Simon Nicolas, MAAG, Hans, FRANCIS, Samson

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5-membered heteroaryl carboxamide compounds for treatment of HBV von Rai, Roopa, Bannen, Lynne, Li, Leping, Haydar, Simon Nicolas, Bures, Mark G, Walker, Michael

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Hepatitis b core protein modulators von Maag, Hans, Li, Leping, Haydar, Simon Nicolas, Francis, Samson, Bures, Mark G, Arnold, Lee D, Turner, Jr., William W

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5-MEMBERED HETEROARYL CARBOXAMIDE COMPOUNDS FOR TREATMENT OF HBV von BANNEN, Lynne, LI, Leping, BURES, Mark G, WALKER, Michael, HAYDAR, Simon, Nicolas, RAI, Roopa

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