Novel chemical entities inhibiting Mycobacterium tuberculosis growth identified by phenotypic high-throughput screening von Kumar, Anuradha, Chettiar, Somsundaram, Brown, Brian S., Early, Julie, Ollinger, Juliane, Files, Megan, Bailey, Mai A., Korkegian, Aaron, Dennison, Devon, McNeil, Matthew, Metz, James, Osuma, Augustine, Curtin, Michael, Kunzer, Aaron, Freiberg, Gail, Bruncko, Milan, Kempf, Dale, Parish, Tanya

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Discovery of ABBV-4083, a novel analog of Tylosin A that has potent anti-Wolbachia and anti-filarial activity von von Geldern, Thomas W, Morton, Howard E, Clark, Rick F, Brown, Brian S, Johnston, Kelly L, Ford, Louise, Specht, Sabine, Carr, Robert A, Stolarik, Deanne F, Ma, Junli, Rieser, Matthew J, Struever, Dominique, Frohberger, Stefan J, Koschel, Marianne, Ehrens, Alexandra, Turner, Joseph D, Hübner, Marc P, Hoerauf, Achim, Taylor, Mark J, Ward, Stephen A, Marsh, Kennan, Kempf, Dale J

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TRPV1 antagonist, A-889425, inhibits mechanotransmission in a subclass of rat primary afferent neurons following peripheral inflammation von Brederson, Jill-Desiree, Chu, Katharine L., Reilly, Regina M., Brown, Brian S., Kym, Philip R., Jarvis, Michael F., McGaraughty, Steve

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Antagonism of TRPV1 receptors indirectly modulates activity of thermoregulatory neurons in the medial preoptic area of rats von McGaraughty, Steve, Segreti, Jason A, Fryer, Ryan M, Brown, Brian S, Faltynek, Connie R, Kym, Philip R

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Asymmetric Synthesis of Oxygen Heterocycles via Pd-Catalyzed Dynamic Kinetic Asymmetric Transformations: Application to Nucleosides von Trost, Barry M., Brown, Brian S., McEachern, Ernest J., Kuhn, Oliver

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Targeting IRAK3 for Degradation to Enhance IL-12 Pro-inflammatory Cytokine Production von Rowley, Ann, Brown, Brian S., Stofega, Mary, Hoh, Hana, Mathew, Rebecca, Marin, Violeta, Ding, Rong-Xian, McClure, Ryan A., Bittencourt, Fabiola M., Chen, Jun, Gururaja, Tarikere, Kinoshita, Taisei, Wang, Xueqing, Rivkin, Alexey, Woller, Kevin R.

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Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure-Based Drug Design von Hobson, Adrian D, Judge, Russell A, Aguirre, Ana L, Brown, Brian S, Cui, Yifang, Ding, Ping, Dominguez, Eric, DiGiammarino, Enrico, Egan, David A, Freiberg, Gail M, Gopalakrishnan, Sujatha M, Harris, Christopher M, Honore, Marie P, Kage, Karen L, Kapecki, Nicolas J, Ling, Christopher, Ma, Junli, Mack, Helmut, Mamo, Mulugeta, Maurus, Stefan, McRae, Bradford, Moore, Nigel S, Mueller, Bernhard K, Mueller, Reinhold, Namovic, Marian T, Patel, Kaushal, Pratt, Steve D, Putman, C. Brent, Queeney, Kara L, Sarris, Kathy K, Schaffter, Lisa M, Stoll, Vincent, Vasudevan, Anil, Wang, Lei, Wang, Lu, Wirthl, William, Yach, Kimberly

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Synthesis of ABBV-168, a 2′-Bromouridine for the Treatment of Hepatitis C von Voight, Eric A, Brown, Brian S, Greszler, Stephen N, Halvorsen, Geoff T, Zhao, Gang, Kruger, Albert W, Hartung, John, Lukin, Kirill A, Martinez, Steven R, Moschetta, Eric G, Tudesco, Michael T, Ide, Nathan D

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Synthesis and evaluation of 2′-dihalo ribonucleotide prodrugs with activity against hepatitis C virus von Chris Krueger, A., Chen, Hui-Ju, Randolph, John T., Brown, Brian S., Halvorsen, Geoff T., Heyman, Howard R., Li, Tongmei, Marvin, Christopher C., Shanley, Jason P., Voight, Eric A., Bow, Daniel A.J., Van Handel, Cecilia, Peterkin, Vincent, Carr, Robert A., Stolarik, DeAnne, Dekhtyar, Tatyana, Irvin, Michelle L., Krishnan, Preethi, Henry, Rodger F., Wagner, Rolf, DeGoey, David A.

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Fructose-1,6-bisphosphatase Inhibitors. 1. Purine Phosphonic Acids as Novel AMP Mimics von Dang, Qun, Brown, Brian S, Liu, Yan, Rydzewski, Robert M, Robinson, Edward D, Poelje, Paul D. van, Reddy, M. Rami, Erion, Mark D

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Contributions of Central and Peripheral TRPV1 Receptors to Mechanically Evoked and Spontaneous Firing of Spinal Neurons in Inflamed Rats von McGaraughty, Steve, Chu, Katharine L, Brown, Brian S, Zhu, Chang Z, Zhong, Chengmin, Joshi, Shailen K, Honore, Prisca, Faltynek, Connie R, Jarvis, Michael F

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Tetrahydropyridine-4-carboxamides as novel, potent transient receptor potential vanilloid 1 (TRPV1) antagonists von Brown, Brian S., Keddy, Ryan, Zheng, Guo Zhu, Schmidt, Robert G., Koenig, John R., McDonald, Heath A., Bianchi, Bruce R., Honore, Prisca, Jarvis, Michael F., Surowy, Carol S., Polakowski, James S., Marsh, Kennan C., Faltynek, Connie R., Lee, Chih-Hung

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Anti-inflammatory microRNA-146a protects mice from diet-induced metabolic disease von Runtsch, Marah C, Nelson, Morgan C, Lee, Soh-Hyun, Voth, Warren, Alexander, Margaret, Hu, Ruozhen, Wallace, Jared, Petersen, Charisse, Panic, Vanja, Villanueva, Claudio J, Evason, Kimberley J, Bauer, Kaylyn M, Mosbruger, Timothy, Boudina, Sihem, Bronner, Mary, Round, June L, Drummond, Micah J, O'Connell, Ryan M

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Discovery of TRPV1 antagonist ABT-116 von Brown, Brian S, Keddy, Ryan, Perner, Richard J, DiDomenico, Stanley, Koenig, John R, Jinkerson, Tammie K, Hannick, Steven M, McDonald, Heath A, Bianchi, Bruce R, Honore, Prisca, Puttfarcken, Pamela S, Moreland, Robert B, Marsh, Kennan C, Faltynek, Connie R, Lee, Chih-Hung

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In Vitro Structure−Activity Relationship and In Vivo Characterization of 1-(Aryl)-3-(4-(amino)benzyl)urea Transient Receptor Potential Vanilloid 1 Antagonists von Perner, Richard J, DiDomenico, Stanley, Koenig, John R, Gomtsyan, Arthur, Bayburt, Erol K, Schmidt, Robert G, Drizin, Irene, Zheng, Guo Zhu, Turner, Sean C, Jinkerson, Tammie, Brown, Brian S, Keddy, Ryan G, Lukin, Kurill, McDonald, Heath A, Honore, Prisca, Mikusa, Joe, Marsh, Kennan C, Wetter, Jill M, St. George, Karen, Jarvis, Michael F, Faltynek, Connie R, Lee, Chih-Hung

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Bis[(para-methoxy)benzyl] phosphonate prodrugs with improved stability and enhanced cell penetration von Dang, Qun, Liu, Yan, Rydzewski, Robert M., Brown, Brian S., Robinson, Edward, van Poelje, Paul D., Colby, Timothy J., Erion, Mark D.

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Structure–activity studies of a novel series of 5,6-fused heteroaromatic ureas as TRPV1 antagonists von Drizin, Irene, Gomtsyan, Arthur, Bayburt, Erol K., Schmidt, Robert G., Zheng, Guo Zhu, Perner, Richard J., DiDomenico, Stanley, Koenig, John R., Turner, Sean C., Jinkerson, Tammie K., Brown, Brian S., Keddy, Ryan G., McDonald, Heath A., Honore, Prisca, Wismer, Carol T., Marsh, Kennan C., Wetter, Jill M., Polakowski, James S., Segreti, Jason A., Jarvis, Michael F., Faltynek, Connie R., Lee, Chih-Hung

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The Routledge Companion to Health Humanities von Crawford, Paul, Brown, Brian, Charise, Andrea

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5-Aminopyrazoles as Dienophiles in the Inverse Electron Demand Diels−Alder Reactions of 2,4,6-Tris(ethoxy- carbonyl)-1,3,5-triazine:  Syntheses of Pyrazolopyrimidines von Dang, Qun, Brown, Brian S, Erion, Mark D

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Deciphering the transcriptional network of the dendritic cell lineage von Miller, Jennifer C, Brown, Brian D, Shay, Tal, Gautier, Emmanuel L, Jojic, Vladimir, Cohain, Ariella, Pandey, Gaurav, Leboeuf, Marylene, Elpek, Kutlu G, Helft, Julie, Hashimoto, Daigo, Chow, Andrew, Price, Jeremy, Greter, Melanie, Bogunovic, Milena, Bellemare-Pelletier, Angelique, Frenette, Paul S, Randolph, Gwendalyn J, Turley, Shannon J, Merad, Miriam

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