Advances in therapeutic peptides targeting G protein-coupled receptors von Davenport, Anthony P., Scully, Conor C. G., de Graaf, Chris, Brown, Alastair J. H., Maguire, Janet J.

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Crystal structure of the GLP-1 receptor bound to a peptide agonist von Jazayeri, Ali, Rappas, Mathieu, Brown, Alastair J. H., Kean, James, Errey, James C., Robertson, Nathan J., Fiez-Vandal, Cédric, Andrews, Stephen P., Congreve, Miles, Bortolato, Andrea, Mason, Jonathan S., Baig, Asma H., Teobald, Iryna, Doré, Andrew S., Weir, Malcolm, Cooke, Robert M., Marshall, Fiona H.

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Extra-helical binding site of a glucagon receptor antagonist von Jazayeri, Ali, Doré, Andrew S., Lamb, Daniel, Krishnamurthy, Harini, Southall, Stacey M., Baig, Asma H., Bortolato, Andrea, Koglin, Markus, Robertson, Nathan J., Errey, James C., Andrews, Stephen P., Teobald, Iryna, Brown, Alastair J. H., Cooke, Robert M., Weir, Malcolm, Marshall, Fiona H.

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Acetylcholine prioritises direct synaptic inputs from entorhinal cortex to CA1 by differential modulation of feedforward inhibitory circuits von Palacios-Filardo, Jon, Udakis, Matt, Brown, Giles A., Tehan, Benjamin G., Congreve, Miles S., Nathan, Pradeep J., Brown, Alastair J. H., Mellor, Jack R.

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Glucagon-Like Peptide-1 and Its Class B G Protein-Coupled Receptors: A Long March to Therapeutic Successes von Graaf, Chris de, Donnelly, Dan, Wootten, Denise, Lau, Jesper, Sexton, Patrick M, Miller, Laurence J, Ahn, Jung-Mo, Liao, Jiayu, Fletcher, Madeleine M, Yang, Dehua, Brown, Alastair J H, Zhou, Caihong, Deng, Jiejie, Wang, Ming-Wei

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Structures of G protein-coupled receptors reveal new opportunities for drug discovery von Cooke, Robert M., Brown, Alastair J.H., Marshall, Fiona H., Mason, Jonathan S.

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Structure-Based Drug Discovery of N‑((R)‑3-(7-Methyl‑1H‑indazol-5-yl)-1-oxo-1-(((S)‑1-oxo-3-(piperidin-4-yl)-1-(4-(pyridin-4-yl)piperazin-1-yl)propan-2-yl)amino)propan-2-yl)-2′-oxo... von Bucknell, Sarah J, Ator, Mark A, Brown, Alastair J. H, Brown, Jason, Cansfield, Andrew D, Cansfield, Julie E, Christopher, John A, Congreve, Miles, Cseke, Gabriella, Deflorian, Francesca, Jones, Christopher R, Mason, Jonathan S, O’Brien, M. Alistair, Ott, Gregory R, Pickworth, Mark, Southall, Stacey M

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Regional characterisation of TRPV1 and TRPA1 signalling in the mouse colon mucosa von Evans, Caryl, Howells, Kathryn, Suzuki, Rie, Brown, Alastair J.H., Cox, Helen M.

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Differential Signaling by Splice Variants of the Human Free Fatty Acid Receptor GPR120 von Watson, Sarah-Jane, Brown, Alastair J.H., Holliday, Nicholas D.

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Roles of GPR41 and GPR43 in leptin secretory responses of murine adipocytes to short chain fatty acids von Zaibi, Mohamed S., Stocker, Claire J., O’Dowd, Jacqueline, Davies, Alison, Bellahcene, Mohamed, Cawthorne, Michael A., Brown, Alastair J.H., Smith, David M., Arch, Jonathan R.S.

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Can residence time offer a useful strategy to target agonist drugs for sustained GPCR responses? von Hothersall, J. Daniel, Brown, Alastair J., Dale, Ian, Rawlins, Philip

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Author Correction: Acetylcholine prioritises direct synaptic inputs from entorhinal cortex to CA1 by differential modulation of feedforward inhibitory circuits von Palacios-Filardo, Jon, Udakis, Matt, Brown, Giles A., Tehan, Benjamin G., Congreve, Miles S., Nathan, Pradeep J., Brown, Alastair J. H., Mellor, Jack R.

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Cholinergic muscarinic M 1 and M 4 receptors as therapeutic targets for cognitive, behavioural, and psychological symptoms in psychiatric and neurological disorders von Erskine, Daniel, Taylor, John-Paul, Bakker, Geor, Brown, Alastair J H, Tasker, Tim, Nathan, Pradeep J

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Cholinergic muscarinic M1 and M4 receptors as therapeutic targets for cognitive, behavioural, and psychological symptoms in psychiatric and neurological disorders von Erskine, Daniel, Taylor, John-Paul, Bakker, Geor, Brown, Alastair J.H., Tasker, Tim, Nathan, Pradeep J.

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A novel somatostatin receptor ligand for human ACTH - and GH -secreting pituitary adenomas von Regazzo, Daniela, Avallone, Serena, MacSweeney, Cliona P, Sergeev, Eugenia, Howe, David, Godwood, Alex, Bennett, Kirstie A, Brown, Alastair J H, Barnes, Matt, Occhi, Gianluca, Barbot, Mattia, Faggian, Diego, Tropeano, Maria Pia, Losa, Marco, Lasio, Giovanni, Scaroni, Carla, Pecori Giraldi, Francesca

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Structural and functional determination of peptide versus small molecule ligand binding at the apelin receptor von Williams, Thomas L., Verdon, Grégory, Kuc, Rhoda E., Currinn, Heather, Bender, Brian, Solcan, Nicolae, Schlenker, Oliver, Macrae, Robyn G. C., Brown, Jason, Schütz, Marco, Zhukov, Andrei, Sinha, Sanjay, de Graaf, Chris, Gräf, Stefan, Maguire, Janet J., Brown, Alastair J. H., Davenport, Anthony P.

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From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease von Brown, Alastair J H, Bradley, Sophie J, Marshall, Fiona H, Brown, Giles A, Bennett, Kirstie A, Brown, Jason, Cansfield, Julie E, Cross, David M, de Graaf, Chris, Hudson, Brian D, Dwomoh, Louis, Dias, João M, Errey, James C, Hurrell, Edward, Liptrot, Jan, Mattedi, Giulio, Molloy, Colin, Nathan, Pradeep J, Okrasa, Krzysztof, Osborne, Greg, Patel, Jayesh C, Pickworth, Mark, Robertson, Nathan, Shahabi, Shahram, Bundgaard, Christoffer, Phillips, Keith, Broad, Lisa M, Goonawardena, Anushka V, Morairty, Stephen R, Browning, Michael, Perini, Francesca, Dawson, Gerard R, Deakin, John F W, Smith, Robert T, Sexton, Patrick M, Warneck, Julie, Vinson, Mary, Tasker, Tim, Tehan, Benjamin G, Teobald, Barry, Christopoulos, Arthur, Langmead, Christopher J, Jazayeri, Ali, Cooke, Robert M, Rucktooa, Prakash, Congreve, Miles S, Weir, Malcolm, Tobin, Andrew B

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Resilience of benthic deep-sea fauna to mining activities von Gollner, Sabine, Kaiser, Stefanie, Menzel, Lena, Jones, Daniel O.B., Brown, Alastair, Mestre, Nelia C., van Oevelen, Dick, Menot, Lenaick, Colaço, Ana, Canals, Miquel, Cuvelier, Daphne, Durden, Jennifer M., Gebruk, Andrey, Egho, Great A., Haeckel, Matthias, Marcon, Yann, Mevenkamp, Lisa, Morato, Telmo, Pham, Christopher K., Purser, Autun, Sanchez-Vidal, Anna, Vanreusel, Ann, Vink, Annemiek, Martinez Arbizu, Pedro

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Respiratory response of the deep-sea amphipod Stephonyx biscayensis indicates bathymetric range limitation by temperature and hydrostatic pressure von Brown, Alastair, Thatje, Sven

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Hyperoxia during venoarterial ECMO: Culprit or co-variate? A comment from the BLENDER investigators von Premraj, Lavienraj, Brown, Alastair, Burrell, Aidan, Fraser, John F, Pilcher, David

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