Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides von Bressi, Jerome C., Jennings, Andy J., Skene, Robert, Wu, Yiqin, Melkus, Robert, Jong, Ron De, O’Connell, Shawn, Grimshaw, Charles E., Navre, Marc, Gangloff, Anthony R.

Volltext

Benzimidazole and imidazole inhibitors of histone deacetylases: Synthesis and biological activity von Bressi, Jerome C., Jong, Ron de, Wu, Yiqin, Jennings, Andy J., Brown, Jason W., O’Connell, Shawn, Tari, Leslie W., Skene, Robert J., Vu, Phong, Navre, Marc, Cao, Xiaodong, Gangloff, Anthony R.

Volltext

Adenosine Analogues as Selective Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase of Trypanosomatidae via Structure-Based Drug Design von Bressi, Jerome C, Verlinde, Christophe L. M. J, Aronov, Alex M, Shaw, My Le, Shin, Sam S, Nguyen, Lisa N, Suresh, Stephen, Buckner, Frederick S, Van Voorhis, Wesley C, Kuntz, Irwin D, Hol, Wim G. J, Gelb, Michael H

Volltext

Conformational changes in Leishmania mexicana glyceraldehyde-3-phosphate dehydrogenase induced by designed inhibitors von Suresh, Stephen, Bressi, Jerome C, Kennedy, Kevin J, Verlinde, Christophe L.M.J, Gelb, Michael H, Hol, Wim G.J

Volltext

A disubstituted NAD+ analogue is a nanomolar inhibitor of trypanosomal glyceraldehyde-3-phosphate dehydrogenase von KENNEDY, Kevin J, BRESSI, Jerome C, GELB, Michael H

Volltext

A bisubstrate analog induces unexpected conformational changes in phosphoglycerate kinase from Trypanosoma brucei von Bernstein, Bradley E, Williams, David M, Bressi, Jerome C, Kuhn, Peter, Gelb, Michael H, Blackburn, G.Michael, Hol, Wim G.J

Volltext

Protein structure-based design of anti-protozoal drugs von Verlinde, Christophe L. M. J., Bressi, Jerome C., Choe, Jungwoo, Suresh, Stephen, Buckner, Frederick S., Van Voorhis, Wesley C., Michels, Paul A. M., Gelb, Michael H., Hol, Wim G. J.

Volltext

Adenosine Analogues as Inhibitors of Trypanosoma brucei Phosphoglycerate Kinase:  Elucidation of a Novel Binding Mode for a 2-Amino-N6-Substituted Adenosine von BRESSI, Jerome C., CHOE, Jungwoo, HOUGH, Melinda T., BUCKNER, Frederick S., VAN VOORHIS, Wesley C., VERLINDE, Christophe L. M. J., HOL, Wim G. J., GELB, Michael H.

Volltext

A new prodrug of paclitaxel: synthesis of Protaxel von Seligson, Allen L, Terry, Ronald C, Bressi, Jerome C, Douglass, James G, Sovak, Milos

Volltext

INHIBITEURS DE L'HISTONE DEACETYLASE von KWOK, LILY, BRESSI, JEROME C, GANGLOFF, ANTHONY R

Volltext bestellen

Adenosine Analogues as Inhibitors of Trypanosoma b rucei Phosphoglycerate Kinase:  Elucidation of a Novel Binding Mode for a 2-Amino-N 6 -Substituted Adenosine von Bressi, Jerome C., Choe, Jungwoo, Hough, Melinda T., Buckner, Frederick S., Van Voorhis, Wesley C., Verlinde, Christophe L. M. J., Hol, Wim G. J., Gelb, Michael H.

Volltext

inibidores de cmet von Zhiyuan Zhang, John D. Lawson, Lily Kwok, Michael B. Wallace, Jeffrey A. Stafford, Sanjib Das, Jerome C. Bressi, Mallareddy Komandla, Philip Erickson, Shaosong Chu

Volltext bestellen

cMET INHIBITORS von BRESSI, JEROME, C, KWOK, LILY, LAWSON, JOHN, D, CHU, SHAOSONG, KOMANDLA, MALLAREDDY, ERICKSON, PHILIP, STAFFORD, JEFFREY, A, ZHANG, ZHIYUAN, DAS, SANJIB, WALLACE, MICHAEL, B

Volltext bestellen

Histone deacetylase inhibitors von Bressi, Jerome C, Gangloff, Anthony R, Kwok, Lily

Volltext bestellen

Histone deacetylase inhibitors von BRESSI JEROME C, GANGLOFF ANTHONY R, KWOK LILY

Volltext bestellen

Histone deacetylase inhibitors von Bressi, Jerome C, Gangloff, Anthony R, Kwok, Lily

Volltext bestellen

Histone deacetylase inhibitors von BRESSI JEROME C, GANGLOFF ANTHONY R, KWOK LILY

Volltext bestellen

Histone deacetylase inhibitors von BRESSI, JEROME C, GANGLOFF, ANTHONY R, KOWK, LILY

Volltext bestellen

cMET inhibitors von KWOK, LILY, LAWSON, JOHN D, WALLACE, MICHAEL B, BRESSI, JEROME C, CHU, SHAOSONG, KOMANDLA, MALLAREDDY, ERICKSON, PHILIP, STAFFORD, JEFFREY A, ZHANG, ZHIYUAN, DAS, SANJIB

Volltext bestellen

HISTONE DEACETYLASE INHIBITORS von BRESSI JEROME C, GANGLOFF ANTHONY R, KWOK LILY

Volltext bestellen