Neurokinin A (NK 2) receptor revisited with SR 48968, a potent non-peptide antagonist von Advenier, C., Rouissi, N., Nguyen, Q.T., Emonds-Alt, X., Breliere, J-C., Neliat, G., Naline, E., Regoli, D.

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Biochemical and pharmacological characterisatioN OF SR141716A, the first potent and selective brain cannabinoid receptor antagonist von Rinaldi-Carmona, Murielle, Barth, Francis, Héaulme, Michel, Alonso, Richard, Shire, David, Congy, Christian, Soubrié, Philippe, Brelière, Jean-Claude, Le Fur, Gérard

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Characterization of the Binding Sites of [3H]SR 48968, a Potent Nonpeptide Radioligand Antagonist of the Neurokinin-2 Receptor von Emondsalt, X., Golliot, F., Pointeau, P., Lefur, G., Breliere, J.C.

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Neuropharmacological profile of a novel and selective ligand of the sigma site: SR 31742A von Poncelet, M., Santucci, V., Paul, R., Gueudet, C., Lavastre, S., Guitard, J., Steinberg, R., Terranova, J.P., Brelière, J.C., Soubrié, P., Le Fur, G.

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Neuropharmacological characterization of SR 140333, a non peptide antagonist of NK1 receptors von JUNG, M, CALASSI, R, LE FUR, G, MARUANI, J, BARNOUIN, M. C, SOUILHAC, J, PONCELET, M, GUEUDET, C, EMONDS-ALT, X, SOUBRIE, P, BRELIERE, J. C

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Evidence for a common molecular mode of action for chemically distinct nonpeptide antagonists at the neurokinin-1 (substance P) receptor von GETHER, U, EMONDS-ALT, X, BRELIERE, J.-C, FUJII, T, HAGIWARA, D, PRADIER, L, GARRET, C, JOHANSEN, T. E, SCHWARTZ, T. W

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Blockade of cannabinoid (CB1) receptors by SR 141716 selectively antagonizes drug-induced reinstatement of exploratory behaviour in gerbils von PONCELET, M, BARNOUIN, M.-C, BRELIERE, J.-C, LE FUR, G, SOUBRIE, P

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Biochemical and pharmacological activities of SR 144190, a new potent non-peptide tachykinin NK2 receptor antagonist von EMONDS-ALT, X, ADVENIER, C, PROIETTO, V, VAN BROECK, D, VILAIN, P, SOUBRIE, P, LE FUR, G, MAFFRAND, J. P, BRELIERE, J. C, COGNON, C, CROCI, T, DAOUI, S, DUCOUX, J. P, LANDI, M, NALINE, E, NELIAT, G, PONCELET, M

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Repeated administration of SR 46349B, a selective 5-hydroxytryptamine2 antagonist, up-regulates 5-hydroxytryptamine2 receptors in mouse brain von Rinaldi-Carmona, M, Congy, C, Simiand, J, Oury-Donat, F, Soubrie, P, Breliere, J C, Le Fur, G

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Synthesis and structures of hypervalent species of silicon and germanium: toward heptacoordination? von Breliere, C, Carre, F, Corriu, R. J. P, Royo, G

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Enhancement of SiH bond reactivity in pentacoordinated structures von Boyer, J., Breliere, C., Corriu, R.J.P., Kpoton, A., Poirier, M., Royo, G.

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Studies on the chronic phase of adjuvant arthritis: effect of SR 41319, a new diphosphonate von Barbier, A, Breliére, J C, Remandet, B, Roncucci, R

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Allosteric modulation of peripheral sigma binding sites by a new selective ligand: SR 31747 von Paul, Raymond, Lavastre, Serge, Floutard, Daniel, Floutard, Régine, Canat, Xavier, Casellas, Pierre, Le Fur, Gérard, Brelière, Jean-Claude

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Development of tetrazole bioisosteres in angiotensin II antagonists von Ferrari, B., Taillades, J., Perreaut, P., Bernhart, C., Gougat, J., Guiraudou, P., Cazaubon, C., Roccon, A., Nisato, D., Le Fur, G., Brelière, J.C.

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Effect of substance P on cytokine production by human astrocytic cells and blood mononuclear cells: characterization of novel tachykinin receptor antagonists von Derocq, Jean-Marie, Ségui, Michel, Blazy, Chantal, Emonds-Alt, Xavier, Le Fur, Gérard, Brelière, Jean-Claude, Casellas, Pierre

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Two nonpeptide tachykinin antagonists act through epitopes on corresponding segments of the NK1 and NK2 receptors von U Gether, Y Yokota, X Emonds-Alt, J C Brelière, J A Lowe, 3rd, R M Snider, S Nakanishi, T W Schwartz

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Pentacoordinate silicon and germanium derivatives: molecular structure von Breliere, C., Carre, F., Corriu, R.J.P., De Saxce, A., Poirier, M., Royo, G.

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Effects of SR140333, a selective non-peptide NK1 receptor antagonist, on trigemino-thalamic nociceptive pathways in the rat von Michaud, JC, Alonso, R, Gueudet, C, Fournier, M, Calassi, R, Brelière, JC, Le Fur, G, Soubrié, P

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Immunopharmacological profile of SR 31747: In vitro and in vivo studies on humoral and cellular responses von Casellas, Pierre, Bourrié, Bernard, Canat, Xavier, Carayon, Pierre, Buisson, Isabelle, Paul, Raymond, Brelière, Jean-Claude, Le Fur, Gérard

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A potent and selective non-peptide antagonist of the neurokinin a (NK 2) receptor von Emonds-Alt, X., Vilain, P., Goulaouic, P., Proietto, V., Van Broeck, D., Advenier, C., Naline, E., Neliat, G., Le Fur, G., Breliére, J.C.

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