Novel library synthesis of 3,4-disubstituted pyridin-2(1 H )-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature von Pierre, Romain, Brethon, Anne, Jacques, Sylvain A, Blond, Aurélie, Chambon, Sandrine, Talano, Sandrine, Raffin, Catherine, Musicki, Branislav, Bouix-Peter, Claire, Tomas, Loic, Ouvry, Gilles, Morgentin, Rémy, Hennequin, Laurent F, Harris, Craig S

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Synthesis and in vitro evaluation of novel highly potent coumarin inhibitors of gyrase B von Laurin, Patrick, Ferroud, Didier, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav

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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists von Ouvry, Gilles, Bouix-Peter, Claire, Ciesielski, Fabrice, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, Duvert, Denis, Feret, Christophe, Harris, Craig S., Lamy, Laurent, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Pascau, Jonathan, Parnet, Véronique, Perrin, Agnès, Pierre, Romain, Polge, Gaëlle, Raffin, Catherine, Rival, Yves, Taquet, Nathalie, Thoreau, Etienne, Hennequin, Laurent F.

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Route scouting and optimization of a potent sulfoximine-based inverse agonist of RORγt von Lafitte, Guillaume, Parnet, Veronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Musicki, Branislav, Tomas, Loic, Bouix-Peter, Claire, Ouvry, Gilles, Daver, Sebastien, Arlabosse, Jean-Marie, Boiteau, Jean-Guy, Gerfaud, Thibaud, Harris, Craig S.

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Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma von Fournier, Jean-François, Bhurruth-Alcor, Yushma, Musicki, Branislav, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Bouquet, Karinne, Chantalat, Laurent, Delorme, Marion, Drean, Bénédicte, Duvert, Gwenaelle, Fleury-Bregeot, Nicolas, Gauthier, Blanche, Grisendi, Karine, Harris, Craig S., Hennequin, Laurent F., Isabet, Tatiana, Joly, Florence, Lafitte, Guillaume, Millois, Corinne, Morgentin, Rémy, Pascau, Jonathan, Piwnica, David, Rival, Yves, Soulet, Catherine, Thoreau, Étienne, Tomas, Loïc

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Early Development Scale-Up of a Novel CXCR Antagonist: Focus on Racemic and Stereoselective Routes of a Key Intermediate von Tabet, Samuel, Rodeville, Nicolas, Mathieu, Arnaud, Raffin, Catherine, Millois-Barbuis, Corinne, Musicki, Branislav, Muller, Franck, Gerfaud, Thibaud, Boiteau, Jean-Guy, Cardinaud, Isabelle

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Sulfoximines as potent RORγ inverse agonists von Ouvry, Gilles, Bihl, Franck, Bouix-Peter, Claire, Christin, Olivier, Defoin-Platel, Claire, Deret, Sophie, Feret, Christophe, Froude, David, Hacini-Rachinel, Feriel, Harris, Craig S., Hervouet, Catherine, Lafitte, Guillaume, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Parnet, Veronique, Pascau, Coralie, Pascau, Jonathan, Pierre, Romain, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent F.

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Process Development and Good Manufacturing Practice Production of a Tyrosinase Inhibitor via Titanium-Mediated Coupling between Unprotected Resorcinols and Ketones von Gerfaud, Thibaud, Martin, Cédric, Bouquet, Karinne, Talano, Sandrine, Millois-Barbuis, Corinne, Musicki, Branislav, Boiteau, Jean-Guy, Cardinaud, Isabelle

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A convenient one-pot synthesis of boroxoles from diboronic acid von Lafitte, Guillaume, Kunihiro, Kana, Bonneaud, Céline, Dréan, Bénédicte, Gaigne, Frédéric, Parnet, Véronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Fournier, Jean-François, Musicki, Branislav, Ouvry, Gilles, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.

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Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis von Ouvry, Gilles, Atrux‐Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix‐Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie‐Josée, Defoin‐Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean‐François, Froude, David, Hacini‐Rachinel, Fériel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Hélène, Lafitte, Guillaume, Luzy, Anne‐Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Véronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent François

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Synthesis of the 4’-desmethoxy analogue of RU79115 von Musicki, Branislav, Periers, Anne-Marie, Tessot, Nicole, Klich, Michel

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Structure of the light emitter in krill (Euphausia pacifica) bioluminescence von Nakamura, Hideshi, Musicki, Branislav, Kishi, Yoshito, Shimomura, Osamu

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Improved antibacterial activities of coumarin antibiotics bearing 5′,5′-dialkylnoviose: biological activity of RU79115 von Musicki, Branislav, Periers, Anne-Marie, Laurin, Patrick, Ferroud, Didier, Benedetti, Yannick, Lachaud, Sylvette, Chatreaux, Fabienne, Haesslein, Jean-Luc, Iltis, Alain, Pierre, Christine, Khider, Jean, Tessot, Nicole, Airault, Marlene, Demassey, Jacques, Dupuis-Hamelin, Claudine, Lassaigne, Patrice, Bonnefoy, Alain, Vicat, Pascale, Klich, Michel

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Chemokine CXCR1 and CXCR2 receptor antagonist compounds, and use thereof in the treatment of chemokine-mediated pathologies von Musicki, Branislav, Bhurruth-Alcor, Yushma

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Noviose mimics of the coumarin inhibitors of gyrase B von Musicki, Branislav, Periers, Anne-Marie, Piombo, Laurent, Laurin, Patrick, Klich, Michel, Dupuis-Hamelin, Claudine, Lassaigne, Patrice, Bonnefoy, Alain

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NOVEL JAK INHIBITOR COMPOUNDS, METHOD FOR SYNTHESIZING SAME AND USE THEREOF von OUVRY, Gilles, MUSICKI, Branislav, HARRIS, Craig, THOREAU, Etienne

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NOVEL JAK INHIBITOR COMPOUNDS, METHODS FOR SYNTHESIZING SAME AND USE THEREOF von OUVRY, Gilles, MUSICKI, Branislav, Thoreau, Etienne, HARRIS, Craig

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NOVEL JAK INHIBITOR COMPOUNDS, METHOD FOR SYNTHESIZING SAME AND USE THEREOF von OUVRY, Gilles, MUSICKI, Branislav, HARRIS, Craig, THOREAU, Etienne

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NOVEL JAK INHIBITOR COMPOUNDS, METHOD FOR SYNTHESIZING SAME AND USE THEREOF von OUVRY, Gilles, MUSICKI, Branislav, GEORGE, Nicolas, FOUCHET, Marie-Hélène, HARRIS, Craig, BOUIX-PETER, Claire

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Structure-activity relationship in two series of aminoalkyl substituted coumarin inhibitors of gyrase B von Laurin, Patrick, Ferroud, Didier, Schio, Laurent, Klich, Michael, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav

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